11

DAY BY DAY PROGRAM

July 30 (Mon)

8:45 – 11:00	Opening ceremony & Plenary Lectures (Main Hall)

8:45 – 9:00	OPENING CEREMONY

9:00	Chair: S. M. Weinreb (Penn State University, USA)
*30-PL-1*	B. M. Trost Stanford University, USA
	Transition Metal Catalysis for Synthesis of Bioactive Heterocycles

10:00	Chair: S. E. Denrnark (University of IlIinois at Urbana-Champaign, USA)
*30-PL-2*	K. Fuji - Kyoto University, Japan
.	Asymmetric Induction Based on the Dynamic Chirality of Enolates

11:00 – 11:30	BREAK

11:30 – 12:05	Invited Lectures (Section A, B, C, D)

SECTION A	(Room 301)- - - - Chair: M. Miyashita (Hokkaido University, Japan)
*30-IL-1*	V. H. Rawal The University of Chicago, USA V. Huang, T. Iwama The University of Chicago, USA
	Catalytic Asymmetric Diels-Alder Reactions: Novel Routes to Bioactive Alkaloid Natural Products
		96

SECTION B	(Room 302)- - - - Chair: Y. Nagao (University of Tokushima, Japan)
*30-IL-2*	S. Ma Shanghai Institute of Organic Chemistry, China
	Recent Advances on New Synthetic Methodologies for Furan Derivatives	97

SECTION C	(Room 303)- - - - Chair: M. Node (Kyoto Pharmaceutical University, Japan)
*30-IL-3*	S.E. Denmark University of Illinois, USA
	New Directions in the Tandem Cycloaddition Chemistry of Nitroalkenes	98

SECTION D	(Room 304)- - - - Chair: M. Yamaguchi (Tohoku University, Japan)
*30-IL-4*	K. Ogura Chiba University, Japan
	Facile Formation of Metal-Lustrous Crystals from l-Aryl-2-(5-tricyanoethenyl-2-thienyl)-5-(2-thienyl)pyrroles
		99
12:05 – 12:40	Invited Lectures (Section A, B, C, D)

SECTION A	(Room 301)- - - - Chair: M. Miyashita (Hokkaido University, Japan)
*30-IL-5*	B. Yu Shanghai Institute of Organic Chemistry, China B. Li, J. Xie, H. Yu, G. Xing, S. Lu, Y. Hui Shanghai Institute of Organic Chemistry, China
	"One Pot" Assembly of Plant Glycosides	100

SECTION B	(Room 302)- - - - Chair: Y. Nagao (University of Tokushima, Japan)
*30-IL-6*	D. W. C. MacMillan California Institute of Technology, USA C.J. Borths, W.S. Jen, J. S. Wiener, N.A. Paras, R. Wilson California Institute of Technology, USA
	Enantioselective Organocatalysis: A New and Broadly Useful Strategy for Enantioselective Synthesis using Organic Catalysts	101

SECTION C	(Room 303)- - - - M. Node (Kyoto Pharmaceutical University, Japan)
*30-IL-7*	N. Yasuda Merck Research Laboratories, USA Y. Hisao, M. Palucki, K. Wells, M.S. Jensen, N. Rivera, C. Yang, J. Yau, D. L. Hughes, P. J. Reider Merck Research Laboratories, USA
	Efficient Practical Syntheses for Drug Candidates	102

SECTION D	(Room 304)- - - - Chair: M. Yamaguchi (Tohoku University, Japan)
*30-IL-8*	C. L. Raston University of Leeds, UK M. Hardie University of Leeds, UK P.J. Nichols, N. Malic Monash University, Australia
	Ni(II) Macrocycles as Divergent Receptors: An Entry to New Supramolecular Arrays
		103

12:40 – 14:10	LUNCH
14:10 – 17:00	Oral Sessions (Section A, B, C, D)
17:00 – 19:00	Poster Session

July 31 (Tue)

9:00- 11 :00	Plenary Lectures (Main Hall)

9:00	Chair: A. Dondoni (University of Ferrarn, Italy)
*31-PL-3*	A. Fiirstner Max-Planck-Institut fGr Kohlenforschung, Germany
	Catalysis Based Syntheses of Bioactive Heterocycles

10:00	Chair: K. Koga (Nara Institute of Science and Technology, Japan)
*31-PL-4*	S. Murahashi Okayama Universiry of Science, Japan Y.lmada Osaka University, Japan
	Flavin-mimic Catalytic Oxidation and Application to Organic Synthesis

11:00 – 11:30	BREAK

11:30 – 12:05	Invited Lectures (Section A, B, C, D)
SECTION A	(Room 301)- - - - Chair: J. Kobayashi (Hokkaido University, Japan)
*31-IL-9*	W. Steglich Ludwig-Maximilians-Universität Munchen, Germany
	Biosyntheses and Syntheses of Alkaloids from Fungi and Marine Organisms	104

SECTION B	(Room 302)- - - - Chair: S. Hashimoto (Hokkaido University, Japan)
*31-IL-10*	S. Chandrasekaran Indian Institute of Science, India K.R. Prabhu, N. Devan Indian Institute of Science, India
	Novel Synthesis of Heterocycles Mediated by Tetrathiomolybdate	105

SECTION C	(Room 303)- - - - Chair: T. Honda (Hoshi University, Japan)
*31-IL-11*	R.-S. Liu National Tsing-Hua University, Taiwan M. Chen, L. Shu, C. Li National Tsing-Hua University, Taiwan
	Synthesis of Natural Oxygen Heterocycles via Tungsten-Mediated Cyclization Reactions
		106

SECTION D	(Room 304)- - - - Chair: M. Mori (Hokkaido University, Japan)
*31-IL-12*	M. Lautens University of Toronto, Canada
	Rhodium Catalyzed C-C and C-X Bond Formation	107

12:05 – 12:40	Invited Lectures (Section A, B, C, D)

SECTION A	(Room 301)- - - - Chair: J. Kobayashi (Hokkaido University, Japan)
*31-IL-13*	T. Nakata RIKEN, Japan
	Synthetic Studies towards Marine Polycyclic Ethers	108

SECTION B	(Room 302)- - - - Chair: S. Hashimoto (Hokkaido University, Japan)
*31-IL-14*	E. P. Kündig University of Geneva, Switzerland
	V. Alezra, G. Bernardinelli, C. Saudan, F. Viton University of Geneva, Switzerland
	Single Site Chiral Iran and Ruthenium Lewis Acids as Catalysts for Asymmetric Cycloaddition Reactions
		109

SECTION C	(Room 303)- - - - Chair: T. Honda (Hoshi University, Japan)
*31-IL-15*	J. Martens Universität Oldenburg, Germany
	Synthesis of Heterocyclic Imines and Their Application in the Synthesis of Bioactive Compounds
		110

SECTION D	(Room 304)- - - - Chair: M. Mori (Hokkaido University, Japan)
*31-IL-16*	B. H. Kim Pohang University of Science and Technology, Korea G.T. Hwang, V.J. Vun, S.K. Kim Pohang University of Science and Technology, Korea

	Heterocyclic Photo-and Self-responsive Molecules: Design, Synthesis and Evaluation
		111

12:40 – 14:10	LUNCH
14:10 – 15:20	Oral Sessions (Section A, B, C, D)
15:20 – 17:50	Poster Session

August 1 (Wed)

9:00- 11 :00	Plenary Lectures (Main Hall)

9:00	Chair: A. Padwa (Emory University, USA)
*1-PL-5*	J. A. Ellman University of California Berkeley, USA
	New Methods in Synthesis Based Upon Metal-Nitrogen Coordination

10:00	Chair: S. Murai (Osaka University, Japan)
*1-PL-6*	L. S. Liebeskind Emory University, USA A. Alcudia, R. Arrayas, H. Malinakoja, C. Shu, J. Vin Emory University, USA
	High Enantiopurity Scaffolds for Heterocycle Synthesis

11:00 – 11:30	BREAK

11:30 - 12 30	Plenary Lectures (Main Hall)

11:30	Chair: T. Livinghouse (Montana State University, USA)
*1-PL-7*	T. Shioiri Nagoya City University, Japan
	Exploitation of New Synthetic Reagents and Their Application to Novel Construction of Heterocyc1ic Natural Products

12:30	LUNCH

13:30	EXCURSION

August 2 (Thu)

9:00- 11 :50	Award Lectures (Main Hall)

9:10	Chair: S. Lang (Elitra Pharmaceuticals, USA)
*2-AL-1*	V. Snieckus Queen's University, Canada
	*The Directed ortho* Metalation Reaction in Heterocyc1ic Synthesis. A Guided Tour**

11:10	Announcement of the forthcoming 19th ICHC
	R. M. Williams (Colorado State University, USA)

10:20 – 10:50	BREAK

10:50	Chair: C. O. Kappe (Karl-Franzens-University Graz, Austria)
*2-AL-2*	W. H. Pearson University of Michigan, USA
	[3+2] Cycloadditions of 2-Azaallylic Species: Applications to Alkaloid Synthesis

11:50 – 13:10	LUNCH

13:10 – 13:45	Invited Lectures (Section A, B, C, D)
SECTION A	(Room 301)- - - - Chair: M. Somei (Kanazawa University, Japan)
*2-IL-17*	R. M. Williams Colorado State University, USA
	Extraordinarily Versatile Amino Acids Templates for the Total Synthesis of Natural Products, Peptide Isosteres and Amino Acids
		112

SECTION B	(Room 302)- - - - Chair: A. Nishida (Chiba University, Japan)
*2-IL-18*	S. Kim Korea Advanced Institute of Science and Technology, Korea
	Synthetic Applications of N-Aziridinylimines	113

SECTION C	(Room 303)- - - - Chair: M. Ochiai (University of Tokushima, Japan)
*2-IL-19*	K.Narasaka The University of Tokyo, Japan
	Synthesis of Nitrogen-Heterocycles by Radical Cyclization of Oximes	114

SECTION D	(Room 304)- - - - Chair: M. Ihara (Tohoku University, Japan)
*2-IL-20*	E. Kimura Hiroshima University, Japan S. Aoki, M. Shiro Hiroshima University/Rigaku Corporation X-Ray Research Laboratory, Japan
	Cuboctahedral Supramolecular Nanocapsules in Aqueous Solution	115

13:45 – 14:20	Invited Lectures (Section A, B, C, D)

SECTION A	(Room 301)- - - - Chair: M. Somei (Kanazawa University, Japan)
*2-IL-21*	Y. Kita Osaka University, Japan
	Organic Synthesis Using Hypervalent Iodine Reagent: Novel Synthesis of Heterocycles and Its Application
		116

SECTION B	(Room 302)- - - - Chair: A. Nishida (Chiba University, Japan)
*2-IL-22*	S. Kanemasa Kyushu University, Japan
	Enantioselective 1,3-Dipolar Cycloaddition Reactions Catalyzed by Tolerant Chiral Lewis Acid Catalysts. Nitrone and Nitronate Cycloaddition Reactions
		117

SECTION C	(Room 303)- - - - Chair: M. Ochiai (University of Tokushima, Japan)
*2-IL-23*	H. N. C. Wong The Chinese University of Hong Kong, China K. Chan The Chinese University of Hong Kong, China
	Synthetic Applications of Chiral Furanboronates	118

SECTION D	(Room 304)- - - - Chair: M. Ihara (Tohoku University, Japan)
*2-IL-24*	D. Yang The University of Hong Kong, China
	Ketone-Catalyzed Oxidation Reactions	119

14:30 – 16:00	Oral Sessions (Section A, B, C, D)
16:30 – 18:30	Poster Session

August 3 (Fri)

9:00- 13 :00	Plenary Lectures & Closing Ceremony (Main Hall)

9:00	Chair: H. Neunhoeffer (Darmstadt University of Technology, Germany)
*3-PL-8*	R. Grigg Leeds University, UK
	Palladium and Bimetallic Catalysed Cascade Reactions. Routes to Potentially Bioactive Complex Heterocycles

10:00	Chair: O. Yonemitsu (Okayama University of Science, Japan)
*3-PL-9*	G. Queguiner Institute of Research in Fine Organic Chemistry of Normandy, France
	Keys for Metallation of Pyridines, Quinolines and Diazunes (Pyrimidines, Pyridazines, Pyrazines)

11:30	Chair: A. R. Katritzky (University of Florida, USA)
*3-PL-10*	V. Kishi Harvard University, USA
	Stereochemical Assignment of (Acyclic) Molecules through Organic Synthesis - Universal NMR Oatabase Approach -

12:30	CLOSING CEREMONY

ORAL AND POSTER SESSION PROGRAM
July 30 (Mon)				Oral Presentation
14:10 - 15:20			SECTION A (Room 301)
Chair: R. Göttlich (Universität Münster, Germany)
*A-1*	Synthesis of the Quinone-type Antimicrobial Natural Products Dehydroherbarin and Mimosamycin
					120
	N. De Kimpe, B. Kesteleyn, T. Nguyen Van, L. Van Puyvelde (University of Ghent, Belgium)
	Program No.: 30-OP-1 Poster No.: 30-PO-1

*A-2*	Epoxide Hydrolases: A Versatile Tool for the Synthesis of Heterocyclic Natural Products
					121
	A. Steinreiber, S. F. Mayer, S. M. Glück, K. Faber (KF University Graz, Austria)
	Program No.: 30-OP-5 Poster No.: 30-PO-2

*A-3*	Asymmetric Total Synthesis of 11-Deoxytetrodotoxin				122
	T. Nishikawa, M. Asai, M. Isobe (Nagoya University, Japan)
	Program No.: 30-OP-9 Poster No.: 30-PO-3

*A-4*	Daphnezomines, Novel Alkaloids from Daphniphyllum				123
	H. Morita, N. Yoshida, J. Kobayashi (Hokkaido University, Japan)
	Program No.: 30-OP-13 Poster No.: 30-PO-4

*A-5*	*Total Synthesis of Thiazole-Containing Cyclic Peptides, cis,cis-* Ceratospongamide and Lyngbyabellin A**
					124
	F. Yokokawa, H. Sameshima, T. Shioiri (Nagoya City University, Japan)
	Program No.: 30-OP-17 Poster No.: 30-PO-5

*A-6*	Total Synthesis of Phytotoxins, Solanapyrones D and E				125
	H. Hagiwara, K. Kobayashi, S. Miya, T. Hoshi, T. Suzuki, M. Ando (Niigata University, Japan)
	Program No.: 30-OP-21 Poster No.: 30-PO-6

*A-7*	Synthesis and Biological Activities of Epolactaene and Related Compounds				126
	S. Nagata, Y. Matsubara, K. Kuramchi, H. Uchiro, J. Nakai, M. Ikekita, S. Kobayashi (Science University of Tokyo, Japan)
	Program No.: 30-OP-25 Poster No.: 30-PO-7

15:50 - 17:00		SECTION A (Room 301)
Chair: M. Toyota (Tohoku University, Japan)
*A-8*	Synthetic Studies on Biologically Active Polyketides with Tetramic Acid Moiety				127
	N. Satoyoshi, S. Doishita, Y. Fukuda, M. Shindo, K. Shishido (University of Tokushima, Japan)
	Program No.: 30-OP-29 Poster No.: 30-PO-8

*A-9*	Studies Towards the Total Synthesis of Zoanthamine Alkaloids				128
	H. Oguri, G. Hirai, S. M. Moharram, Y. Koizumi, M. Hirama (Tohoku University / CREST, Japan Science and Technology Corporation (JST), Japan)
	Program No.: 30-OP-33 Poster No.: 30-PO-9

*A-10*	Rhodium-Catalyzed Carbonylation at sp³ C-H Bonds Adjacent to a Nitrogen Atomin Alkylamines				129
	N. Chatani, T. Asaumi, T. Ikeda, F. Kakiuchi, S. Murai (Osaka University, Japan)
	Program No.: 30-OP-37 Poster No.: 30-PO-10
*A-11*	Synthesis of Nitrogen Containing Heterocycles Using Ring Closing Metathesis (RCM)
					130
	M. Arisawa, H. Kaneko, C. Theeraladanon, A. Nishida, M. Nakagawa (Chiba University, Japan)
	Program No.: 30-OP-41 Poster No.: 30-PO-11

*A-12*	Improved Process for the Asymmetric Strecker Synthesis and its Application to the Synthesis of Natural Products
					131
	T. Shinada, M. Kawasaki, K. Namba, S. Iwama, Y. Ohfune (Osaka City University, Japan)
	Program No.: 30-OP-45 Poster No.: 30-PO-12

*A-13*	*Catalytic Asymmetric Allylic Alkylation in Water with a Recyclable Amphiphilic Resin-Supported P, N-Chelating Palladium Complex*
					132
	Y. Uozumi, K. Shibatomi (Institute for Molecular Science, Japan)
	Program No.: 30-OP-49 Poster No.: 30-PO-13

*A-14*	Intramolecular [2+2] Photocycloadditions as an Approach Towards the Right-Hand Side of Solanoeclepin A
					133
	R. H. Blaauw, J.-F. Brière, R. De Jong, J. C. J. Benningshof, A. E.Van Ginkel, H. Hiemstra (University of Amsterdam, The Netherlands)
	Program No.: 30-OP-53 Poster No.: 30-PO-14

14:10 - 15:20		SECTION B (Room 302)
	Chair: H. Kotsuki (Kochi University, Japan)
*B-1*	(Het)arylacetonitriles and Arylsulfonylacetonitriles in Synthesis of Condensed Heterocycles and Heterocyclic b-Enaminoketones
					134
	Y. M. Volovenko, A. V. Tverdokhlebov, T. A. Volovnenko, T. V. Shokol (Kiev National Taras Shevchenko University, Ukraine)
	Program No.: 30-OP-2 Poster No.: 30-PO-34

*B-2*	Preparation and Reactivities of Novel (Diacetoxyiodolarenes Bearing Heteroaromatics
					135
	H. Togo, T. Nabana (Chiba University, Japan)
	Program No.: 30-OP-6 Poster No.: 30-PO-35

*B-3*	Anionically Activated Trifluoromethyl Group in Heterocyclic Synthesis				136
	A. S. Kiselyov (ImClone Systems Incorporated, USA)
	Program No.: 30-OP-10 Poster No.: 30-PO-36

*B-4*	New Route for the Synthesis of Fused Pyrimidine by Annelation of an Imidazo Moiety
					137
	A. Z. M. S. Chowdhury, Y. Shibata (National Institute for Environmental Studies, Japan)
	Program No.: 30-OP-14 Poster No.: 30-PO-37

*B-5*	Synthesis of the Azepinoindole Stenine Using a Linked Pummerer-Cycloaddition Strategy
					138
	A. Padwa, J. D. Ginn, S. M. Lynch (Emory University, USA)
	Program No.: 30-OP-18 Poster No.: 30-PO-38

*B-6*	Synthesis of 4,5-Dihydro-1,2,4-triazin-6-ones via Tandem Iminoacylation/Cycloacylation of Amino Acid Esters and Hydrazonyl Bromides				139

	D. M. Wilson, M. Ramirez-Weinhouse, L. Mao, V. Molteni, A. Termin (Du Pont Pharmaceuticals Research Laboratories, USA)
	Program No.: 30-OP-22 Poster No.: 30-PO-39

*B-7*	Thermal Ring Expansion Reactions of 2-Halo-2H-Azirines: Synthesis of 4‑Haloisoxazoles
					140
	T. M. V. D. Pinho e Melo, C. S. J. Lopes, A. M. d'A. Rocha Gonsalves (University of Coimbra, Portugal)
	Program No.: 30-OP-26 Poster No.: 30-PO-40

15:50 - 17:00		SECTION B (Room 302)
Chair: M. Otsuka (Kumamoto University, Japan)
*B-8*	*Synthesis of Azacycles and Oxacycles via* Tandem Radical Addition-Cyclization**				141
	T. Naito, H. Miyabe, K. Fujii (Kobe Pharmaceutical University, Japan)
	Program No.: 30-OP-30 Poster No.: 30-PO-41

*B-9*	*A Novel Entry into the Fischer Indole Synthesis via* Thermal Cyclization of N-Trifluoroacetyl Enehydrazine**
					142
	O. Miyata, Y. Kimura, K. Muroya, T. Naito (Kobe Pharmaceutical University, Japan)
	Program No.: 30-OP-34 Poster No.: 30-PO-42

*B-10*	Thermal and Photochemical Transformations with 4-Isoxazolines: 3-, 5-and 7-Membered N-Heterocycles via Azomethine Ylide Intermediates
					143
	W. Eberbach, W. Friebolin (University of Freiburg, Germany)
	Program No.: 30-OP-38 Poster No.: 30-PO-43

*B-11*	Synthesis of Heterocycles Using Lanthanide. Triflate/TMSCI				144
	A. Nishida, M. Yamanaka, M. Kawahara, R. Tsuji, M. Arisawa, M. Nakagawa (Chiba University, Japan)
	Program No.: 30-OP-42 Poster No.: 30-PO-44

*B-12*	Asymmetric Synthesis of Oxazolines Using a Chiral Nitridomanganese Complex				145
	S. Minakata, M. Nishimura, T. Takahashi, M. Komatsu (Osaka University, Japan)
	Program No.: 30-OP-46 Poster No.: 30-PO-45

*B-13*	The Chemistry of 1-Hydroxyindoles				146
	K. Noguchi, A. Goto, T. Hayashi, F. Yamada, K. Yamada, M. Somei (Kanazawa University, Japan)
	Program No.: 30-OP-50 Poster No.: 30-PO-46

*B-14*	Cinchona Alkaloid Catalyzed Asymmetric Baylis-Hillman Reaction and ItsApplication
					147
	Y. Iwabuchi, M. Furukawa, T. Sugihara, M. Ushiyama, M. Nakatani, T. Esumi, S. Hatakeyama (Nagasaki University, Japan)
	Program No.: 30-0P-54 Poster No.: 30-PO-47

14:10 - 15:20		SECTION C (Room 303)
	Chair: S. Hatakeyama (Nagasaki University, Japan)
*C-1*	Synthesis, Antithrombin Activity, and Acute Toxicity of Substituted 3,5‑Dihydroxy-3,5-Dihydro-2-Pyrrolones
					148
	E. A. Goun, D. H. Miles (University of Central Florida, USA) O. P. Krasnykh, S. J. Solodnikov, A. N. Masliwets, N. A. Konjuhova (Perm State University, Russia)
	Program No.: 30-OP-3 Poster No.: 30-PO-69

*C-2*	Synthesis of Nucleosides with Four-membered Heterocyclic Sugars as Potential Antiviral Agents
					149
	E. Ichikawa (The University of Tokyo, Japan), S.Yamamura (Keio University, Japan) Y. Terada (Meijyo University, Japan) K. Kato (Nippon Kayaku Co.Ltd., Japan)
	Program No.: 30-OP-7 Poster No.: 30-PO-70

*C-3*	Mechanistic Insights and Synthesis of Novel Lactam and Peptide based Templates for Serine Protease Inhibition
					150
	J. Seibel, R. Wilmouth, C. Schofield (University of Oxford, United Kingdom)
	Program No.: 30-OP-11 Poster No.: 30-PO-71

*C-4*	Aldol and Arylmethylene Derivatives of 4-Piperiodones				151
	M. J. Turmuchanova, G. S. Litvinenko, D. G. Kim (The Al-Farabi Kazakh State University, Kazakhstan) J. R. Dimmock (University of Saskatchewan, Canada)
	Program No.: 30-OP-15 Poster No.: 30-PO-72

*C-5*	Synthesis of Purines with Inhibitory Activity against Mycobacterium Tuberculosis				152
	A. K. Bakkestuen, A. Bråthe, L-L Gundersen, G. Langli, J. Nolsøe (University of Oslo, Norway)
	Program No.: 30-OP-19 Poster No.: 30-PO-73

*C-6*	*Solid-Phase Synthesis of Dihydropyrimidones via N-Acyliminium Ion-Based* α-Ureidoalkylations
					153
	D. Dallinger, M. G. Valverde, C. O. Kappe (Karl-Franzens-University Graz, Austria)
	Program No.: 30-OP-23 Poster No.: 30-PO-74

*C-7*	Selective Electroreductive Cyclization of Nitrogen-Containing Nonconjugated Enonesand Ynones
					154
	I. Nishiguchi, S. Goda, H. Maekawa (Nagaoka University of Technology, Japan)
	Program No.: 30-OP-27 Poster No.: 30-PO-75

15:50 - 17:00		SECTION C (Room 303)
Chair: I. Nishiguchi (Nagaoka University of Technology, Japan)
*C-8*	Polymer Supported Oligosaccharide Synthesis by Use of Real Time Reaction Monitoring Method
					155
	S. Manabe, H. Ando, Y. Nakahara, Y. Ito (RIKEN (The Institute of Physical and Chemical Research), Japan)
	Program No.: 30-OP-31 Poster No.: 30-PO-76

*C-9*	Synthesis of Fluorine-Containing Heterocycles for Agrochemicals, Pharmaceutical and Polymers
					156
	J. S. Ji, P. Q. Lu, R. Y.Yang (Shanghai High Victory Science & Technology Co., Ltd., China)
	Program No.: 30-OP-35 Poster No.: 30-PO-77

*C-10*	Synthesis, Chemistry, and Applications of Heterocyclic Cage Compounds(V)				157
	H. Wu, H. Lin, Z. Wang, C. Wu (National Chiao Tung University, Taiwan)
	Program No.: 30-OP-39 Poster No.: 30-PO-78

*C-11*	Regioselective Synthesis of Alkynylbenzotriazoles				158
	T. Kitamura, N. Tashi, H. Chen, Y. Fujiwara (Kyushu University, Japan)
	Program No.: 30-OP-43 Poster No.: 30-PO-79

*C-12*	Efficient Anodic Synthesis of 2-Fluoro and 2, 3-Difluorobenzofuran Derivatives				159
	K. M. Dawood (Tokyo Institute of Technology, Japan/ Cairo University, Egypt) H. Ishii, T. Fuchigami (Tokyo Institute of Technology, Japan)
	Program No.: 30-OP-47 Poster No.: 30-PO-80

*C-13*	2H-Pyran-2-ones as Synthons for the Synthesis of α,b-Didehydro-α-amino Acid Derivatives
					160
	L. Vraničar, S. Polanc, M. Kočevar (University of Ljubljana, Slovenia)
	Program No.: 30-OP-51 Poster No.: 30-PO-81

*C-14*	2-Heteroaryl-1,4-Dihydropyrimidines-Novel and Potent Non-Nucleosidic Inhibitors of Hepatitis B Virus (HBV)
					161
	S. Goldmann, J. Stoltefuss, U. Niewöhner, T. Krämer, E. Graef, S. Lottmann, K. Deres, R. Masantschek, D. Koletzki, O. Weber, A. Paessens (BAYER AG, Germany)
	Program No.: 30-OP-55 Poster No.: 30-PO-82

14:10 - 15:20		SECTION D (Room 304)
Chair: R. Shirai (Nara Institute of Science and Technology, Japan)
D-1	C-Phosphorylation of Heteroaromatic Compounds in Synthesis of Novel Phosphorus-Containing Heterocycles
					162
	A. A. Tolmachev, A. Kostyuk (National Academy of Sciences of Ukraine, Ukraine)
	Program No.: 30-OP-4 Poster No.: 30-PO-102

*D-2*	Neighboring Effect of Heteroaromatic Rings for the π-Facial Selectivity				163
	T. Kobayashi, T. Tsuzuki, K. Miki, Y. Tayama (Shinshu University, Japan)
	ProgramNo.: 30-OP-8 Poster No.: 30-PO-103

D-3	Formation of Iminosubstituted Propadienethiones by Thermal (FVP) and Electron Impact Induced Fragmentation of Multisulfur Heterocycles
					164
	C. T. Pedersen (USD, Odense University, Denmark) R. Flammang (University of Mons-Hainaut, Belgium) E. Fanghanel (Martin Luther University, Halle Wittenberg, Germany)
	Program No.: 30-OP-12 Poster No.: 30-PO-104

*D-4*	1,4,5,8-Tetraazafulvalenes - New Starting Material for Functional Dyes				165
	R. Beckert, C. Käpplinger, D. Müller (Friedrich-Schiller-University, Germany)
	Program No.: 30-OP-16 Poster No.: 30-PO-105

*D-5*	Anomalous Carbon Insertion into a Benzene Ring in Bischler-Napieralski Reaction				166
	T. Ishikawa, K. Shimooka, T. Narioka (Chiba University, Japan)
	Program No.: 30-OP-20 Poster No.: 30-PO-106

*D-6*	Synthesis and Properties of Pyrroles and Porphyrins Fused with Rigid Bicyclic Ring
					167
	H. Uno, S. Ito, K. Nakamoto, H. Watanabe, M. Wada, N. Ochi, N. Ono (Ehime University, Japan)
	Program No.: 30-OP-24 Poster No.: 30-PO-107

*D-7*	Photochromic Imidazole: A Novel Material				168
	A. K. Padhy (National Institute of Science & Technology, India)
	Program No.: 30-OP-28 Poster No.: 30-PO-108

15:50 - 17:00		SECTION D (Room 304)
Chair:H.Takahashi (TeikyoUniversity, Japan)
*D-8*	New Approach to Synthesis of 4-Piperidones				169
	D. Kim (The Atyrau Institute of Scientific and Technical Problems, Kazakhstan)
	Program No.: 30-OP-32 Poster No.: 30-PO-109

*D-9*	Chiral Relay Auxilliaries				170
	V. K. Tandon, S. Rai (Lucknow University, India)
	Program No.: 30-OP-36 Poster No.: 30-PO-110

*D-10*	Synthesis of Benzolactones and Benzolactams by Aryl Radical Carbonylation				171
	K. Orito, T. Tatsuzawa, R. Harada, M. Tokuda (Hokkaido University, Japan)
	Program No.: 30-OP-40 Poster No.: 30-PO-111

*D-11*	A New Method for the Preparation of Enantiomerically Pure α-Substituted Pyrrolidines
					172
	T. Maki, Y. Ishida, K. Shirai, O. Onomura, Y. Matsumura (Nagasaki University, Japan)
	Program No.: 30-OP-44 Poster No.: 30-PO-112

*D-12*	The Isolation of the First Stable Atropisomers in Proximity-Screened NZ, NZ-diazasesquinorbornanes (N²[2]polynorbornanes)
					173
	R. N. Warrener, G. Sun (Central Queensland University, Australia)
	Program No.: 30-OP-48 Poster No.: 30-PO-113

*D-13*	Synthesis of Novel, Axially Chiral 1,8-Disubstituted Naphthalenes				174
	A. V. Bedekar, S. Yoshikawa, K.Tanaka (University of Shizuoka, Japan)
	Program No.: 30-OP-52 Poster No.: 30-PO-114

*D-14*	Synthesis of Pyridine Derivatives Using Aminoacroleins as an Equivalent of Malonaldehydes
					175
	H. Suda, H. Saitoh, K. Umihara, Y. Furugori, I. Itoh (Sankio Chemical Co., Lld., Japan)
	Program No.: 30-OP-56 Poster No.: 30-PO-115

July 30 (Mon)		Poster Presentation
17:00 - 19:00

*30-PO-1*	Synthesis of the Quinone-type Antimicrobial Natural Products, Dehydroherbarin and Mimosamycin
			120
	N. De Kimpe, B. Kesteleyn, T. Nguyen Van, L. Van Puyvelde (University of Ghent, Belgium)
	Program No.: 30-OP-1 (A-1)

30-PO-2	Epoxide Hydrolases: A Versatile Tool for the Synthesis of Heterocyclic Natural Products
			121
	A. Steinreiber, S. F. Mayer, S. M.Gluck, K. Faber (KF University Graz, Austria)
	Program No.: 30-OP-5 (A-2)

*30-PO-3*	Asymmetric Total Synthesis of 11-Deoxytetrodotoxin		122
	T. Nishikawa, M. Asai, M. Isobe (Nagoya University, Japan)
	Program No.: 30-OP-9 (A-3)

*30-PO-4*	Daphnezomines, Novel Alkaloids from Daphniphyllum humile		123
	H. Morita, N. Yoshida, J. Kobayashi (Hokkaido University, Japan)
	Program No.: 30-OP-13 (A-4)

*30-PO-5*	*Total Synthesis of Thiazole-Containing Cyclic Peptides, cis,cis-Ceratospongamide and Lyngbyabellin A*
			124
	F. Yokokawa, H. Sameshima, T. Shioiri (Nagoya City University, Japan)
	Program No.: 30-OP-17 (A-5)

*30-PO-6*	Total Synthesis of Phytotoxins, Solanapyrones D and E		125
	H. Hagiwara, K. Kobayashi, S. Miya, T. Hoshi, T. Suzuki, M. Ando (Niigata University, Japan)
	Program No.: 30-OP-21 (A-6)

30-PO-7	Synthesis and Biological Activities of Epolactaene and Related Compounds		126
	S. Nagata, Y. Matsubara, K. Kuramchi, H. Uchiro, J. Nakai, M. Ikekita, S. Kobayashi (Science University of Tokyo, Japan)
	Program No.: 30-OP-25 (A-7)

30-PO-8	Synthetic Studies on Biologically Active Polyketides with Tetramic Acid Moiety
			127
	N. Satoyoshi, S. Doishita, Y. Fukuda, M. Shindo, K. Shishido (University of Tokushima, Japan)
	Program No.: 30-OP-29 (A-8)

*30-PO-9*	Studies Towards the Total Synthesis of Zoanthamine Alkaloids		128
	H. Oguri, G. Hirai, S. M. Moharram, Y. Koizumi, M. Hirama (Tohoku University / CREST / Japan Science and Technology Corporation (JST), Japan)
	Program No.: 30-OP-33 (A-9)

*30-PO-10*	Rhodium-Catalyzed Carbonylation at sp³ C-H Bonds Adjacent to a Nitrogen Atom in Alkylamines
			129
	N. Chatani, T. Asaumi, T. Ikeda, F. Kakiuchi, S. Murai (Osaka University, Japan)
	Program No.: 30-OP-37 (A-10)

*30-PO-11*	Synthesisof Nitrogen Containing Heterocycles Usino Ring Closing Metathesis (RCM)
			130
	M. Arisawa, H. Kaneko, C. Theeraladanon, A. Nishida, M. Nakagawa (Chiba University, Japan)
	Program No.: 30-OP-41 (A-11)

*30-PO-12*	Improved Process for the Asymmetric Strecker Synthesis and its Application to the Synthesis of Natural Products
			131
	T. Shinada, M. Kawasaki, K. Namba, S. Iwama, Y. Ohfune (Osaka City University, Japan)
	Program No.: 30-OP-45 (A-12)

*30-PO-13*	*Catalytic Asymmetric Allylic Alkylation in Water with a Recyclable Amphiphilic Resin-Supported P, N-Chelating Palladium Complex*
			132
	Y. Uozumi, K.Shibatomi (Institute for Molecular Science, Japan)
	Program No.: 30-OP-49 (A-13)

*30-PO-14*	Intramolecular [2+2] Photocycloadditions as an Approach Towards the Right-Hand Side of Solanoeclepin A
			133
	R. H. Blaauw, J.-F. Brière, R. De Jong, J. C. J. Benningshof, A. E. Van Ginkel, H. Hiemstra (University of Amsterdam, The Netherlands)
	Program No.: 30-OP-53 (A-14)

*30-PO-15*	Asymmetric Addition of Me₃SiCN to Chiral Heterocyclic Aldimines		176
	E. Lukevics, I. Iovel, L. Golomba, J. Popelis (Latvian Institute of Organic Synthesis, Latvia)
*30-PO-16*	Concise Enantiospecific Synthesis of a Coccinellid Alkaloid, (-)-Adalinine		177
	T. Honda, M. Kimura (Hoshi University, Japan)

*30-PO-17*	*Synthesis of Some Oxidative Derivatives of Mitragynine, An Indole Alkaloid in Mitragyna speciosa,* and Their Opioid Agonistic Activity**
			178
	H. Takayama, H. Ishikawa, M. Kitajima, N. Aimi (Chiba University, Japan)

*30-PO-18*	C₂-Symmetric 2,6-Diallylpiperidine as Chiral Building Stock		179
	H. Takahata, M. Ichinose, H. Nemoto (Toyama Medical and Pharmaceutical University, Japan)

*30-PO-19*	Concise Route to (-)-Morphine		180
	H. Nagata, N. Miyazawa, K. Ogasawara (Tohoku University, Japan)

*30-PO-20*	Synthetic Studies of Imbiline 1 and Plakinidine C		181
	Y. Kitahara, M. Mochii, M. Mori, T. Mizuno, A. Kubo (Meiji Pharmaceutical University, Japan)

*30-PO-21*	Synthetic Approaches to Homochelidonine		182
	M. Yoshida, T. Watanabe, T. Ishikawa (Chiba University, Japan)

*30-PO-22*	Oxidative Cyclization-Methoxycarbonylation of Cyclic and Acyclic-4-yn-1-ols under Mild Condition
			183
	K. Kato, A. Nishimura, M. Tanaka, Y. Yamamoto, H. Akita (Toho University, Japan)

*30-PO-23*	*Total Synthesis of Dragmacidins A-C via* Indolylglycines**		184
	T. Kawasaki, H. Enoki, K. Matsumura, K. Ohno, M. Sakamoto (Meiji Pharmaceutical University, Japan)

*30-PO-24*	*Erythrinan Alkaloids from Two Erythrina* Plants**		185
	H. Tanaka (Meijo University, Japan) H. Etoh (Shizuoka University, Japan)

*30-PO-25*	Synthesis of Optically Active γ-Butyrolactone and Tetrahydrofuran Lignans
			186
	S. Yamauchi, Y. Kinoshita (Ehime University, Japan)

*30-PO-26*	Stereoselective Synthesis of Mucocin, an Antitumor Agent, Based on a Sml₂- Induced Reductive Cyclization
			187
	S. Takahashi, (RIKEN (Synthetic Organic Chemistry Lab.), Japan) A. Kubota, T. Nakata (RIKEN (The Institute of Physical and Chemical Research), Japan)

*30-PO-27*	Synthetic Study of the Mycalamides: Efficient Synthesis of the Right Half Segment
			188
	Y. Nishii, (RIKEN (Synthetic Organic Chemistry Lab.), Japan) S. Takahashi, T. Nakata (RIKEN (The Institute of Physical and Chemical Research), Japan)

*30-PO-28*	Synthetic Studies on Blasticidin S		189
	Y. Ichikawa, M. Ohbayashi, K. Hirata, M. Isobe (Nagoya University, Japan)
*30-PO-29*	Synthetic Studies on Cyclomarin A, an Antiinflammatory Cyclic Peptide from a Marine Bacterium
			190
	H. Sugiyama, F. Yokokawa, T. Shioiri (Nagoya City University, Japan)

*30-PO-30*	Synthetic Approaches toward Ecteinascidin Marine Natural Products		191
	N. Saito, R. Seki, N. Kameyama, A. Kubo (Meiji Pharmaceutical University, Japan)

*30-PO-31*	Synthesis of Fagaridine by Palladium-assisted Internal Biaryl Coupling Reaction
			192
	T. Sato, Y. Nakano, T. Harayama (Okayama University, Japan)

*30-PO-32*	Synthesis and Studies on Some b-Lactam and Thiazolidine Compounds		193
	H. A. Soleiman (South Valley University, Egypt)

*30-PO-33*	Regioselective Cleavage of Cyclic Ethereal Bond of 7-Oxabicyclo [2.2.1]heptane Derivatives Mediated by Samarium(II)Iodide
			194
	A. Yoshida, H. Takayama (Teikyo University, Japan)

*30-PO-34*	(Het)arylacetonitriles and Arylsulfonylacetonitriles in Synthesis of Condensed Heterocycles and Heterocyclic b-Enaminoketones
			134
	Y. M. Volovenko, A. V. Tverdokhlebov, T. A. Volovnenko, T. V. Shokol (Kiev National Taras Shevchenko University, Ukraine)
	Program No.: 30-OP-2 (B-1)

*30-PO-35*	Preparation and Reactivities of Novel (Diacetoxyiodo)arenes Bearing Heteroaromatics
			135
	H.Togo, T. Nabana (Chiba University, Japan)
	Program No.: 30-OP-6 (B-2)

*30-PO-36*	Anionically Activated Trifluoromethyl Group in Heterocyclic Synthesis		136
	A. S. Kiselyov (ImClone Systems Incorporated, USA)
	Program No.: 30-OP-10 (B-3)

*30-PO-37*	New Route for the Synthesis of Fused Pyrimidine by Annelation of an Imidazo Moiety
			137
	A. Z. M. S. Chowdhury, Y. Shibata (National Institute for Environmental Studies, Japan)
	Program No.: 30-OP-14 (B-4)

*30-PO-38*	Synthesis of the Azepinoindole Stenine Using a Linked Pummerer-Cycloaddition Strategy
			138
	A. Padwa, J. D. Ginn, S. M. Lynch (Emory University, USA)
	Program No.: 30-OP-18 (B-5)

*30-PO-39*	Synthesis of 4,5-Dihydro-1,2,4-triazin-6-ones via Tandem Iminoacylation/Cycloacylation of Amino Acid Esters and Hydrazonyl Bromides
*30-PO-39*			139
	D.M. Wilson, M. Ramirez-Weinhouse, L. Mao, V. Molteni, A. Termin (DuPont Pharmaceuticals Research Laboratories, USA)
	Program No.: 30-OP-22 (B-6)

*30-PO-40*	Thermal Ring Expansion Reactions of 2-Halo-2H-Azirines: Synthesis of 4-Haloisoxazoles
*30-PO-40*			140
	T. M. V. D. Pinho e Melo, C. S.J. Lopes, A. M. d' A. Rocha Gonsalves (University of Coimbra, Portugal)
	Program No.: 30-OP-26 (B-7)

*30-PO-41*	*Synthesis of Azacycles and Oxacycles via* Tandem Radical Addition-Cyclization**
*30-PO-41*			141
	T. Naito, H. Miyabe, K. Fujii (Kobe Pharmaceutical University, Japan)
	Program No.: 30-OP-30 (B-8)

*30-PO-42*	*A Novel Entry into the Fischer Indole Synthesis via* Thermal Cyclization of N-Trifluoroacetyl Enehydrazine**
			142
	O. Miyata, Y. Kimura, K. Muroya, T. Naito (Kobe Pharmaceutical University, Japan)
	Program No.: 30-OP-34 (B-9)

*30-PO-43*	Thermal and Photochemical Transformations with 4-Isoxazolines: 3-, 5- and 7-Membered N-Heterocycles via Azomethine Ylide Intermediates
			143
	W. Eberbach, W. Friebolin (University of Freiburg, Germany)
	Program No.: 30-OP-38 (B-10)

*30-PO-44*	Synthesis-of Heterocycles Using Lanthanide Triflate/TMSCI		144
	A. Nishida, M. Yamanaka, M. Kawahara, R. Tsuji, M. Arisawa, M. Nakagawa (Chiba University, Japan)
	Program No.: 30-OP-42 (B-11)

*30-PO-45*	Asymmetric Synthesis of Oxazolines Using a Chiral Nitridomanganese Complex
			145
	S. Minakata, M. Nishimura, T. Takahashi, M. Komatsu (Osaka University, Japan)
	Program No.: 30-OP-46 (B-12)

*30-PO-46*	The Chemistry of 1-Hydroxyindoles		146
	K. Noguchi, A. Goto, T. Hayashi, F. Yamada, K. Yamada, M. Somei (Kanazawa University, Japan)
	Program No.: 30-OP-50 (B-13)

*30-PO-47*	Cinchona Alkaloid Catalyzed Asymmetric Baylis-Hillman Reaction and its Application
*30-PO-47*			147
	Y. Iwabuchi, M. Furukawa, T. Sugihara, M. Ushiyama, M. Nakatani, T. Esumi, S. Hatakeyama (Nagasaki University, Japan)
	Program No.: 30-OP-54 (B-14)

*30-PO-48*	Reaction of Cyanopyridinium Salts with Active Methylene Compounds		195
	R. Fujita, W. Sato (Tohoku Pharmaceutical University, Japan)

*30-PO-49*	Synthesis of Some 5-Substituted Pyrano[3,4-c]coumarin Derivatives		196
	M. A. Khalil (South Valley University, Egypt)

*30-PO-50*	Asymmetric [2,3] Witting Rearrangement of Crotyl Furfuryl Ethers		197
	M. Tsubuki, T. Kamata, M. Nakatani, K. Yamazaki, T. Matsui, T. Honda (Hoshi University, Japan)

*30-PO-51*	Synthesis and Properties of Some Five-, Six-, Seven-, Eight-Membered Nitrogen-Containing Heterocycles Condensed with 9,10-Anthraquinone Nucleus
*30-PO-51*			198
	L. M. Gornostaev, E. V. Arnold, N. A. Bulgakova, I. V. Kalashnikova, T. I. Lavrikova, R. V. Mitrokhin, O. V. Podvyazny (Krasnoyarsk State Pedagogical University, Russia)

*30-PO-52*	A Regiospecific Synthesis of 1-Heterocyclic Substituted 1,2,4-Triazoles via Base Catalytic Reaction of 1,2,4- Triazole withFunctionalized Carbodiimide
			199
	M.-W. Ding, G.-P. Zeng, Z.-J. Liu (Central China Normal University, China)

*30-PO-53*	Stereodivergent Process for the Synthesis of Dendrobates Alkaloids		200
	N. Toyooka, M. Okumura, H. Nemoto (Toyama Medical and Pharmaceutical University, Japan)

*30-PO-54*	Construction of Novel Heterocyclic Switching Molecules		201
	A. Kakehi, S. Ito, H. Suga, T. Mori, T. Kako (Shinshu University, Japan)

*30-PO-55*	Enantioselective Cyanosilylation of Ketones Promoted by Lewis Acid-Lewis Base Bifunctional Catalyst
*30-PO-55*			202
	M. Kanai, Y. Hamashima, M. Shibasaki (The University of Tokyo, Japan)

*30-PO-56*	Enantioselective Reissert-Type Reaction Promoted by Lewis Acid-Lewis Base Bifunctional Catalyst
*30-PO-56*			203
	K. Funabashi, M. Takamura, M. Kanai, M. Shibasaki (The University of Tokyo, Japan)

*30-PO-57*	Intramolecular Alkyl Migration Reaction in Indolylborates		204
	M. Ishikura, H. Kato, N. Ohnuki (Health Sciences University of Hokkaido, Japan)

*30-PO-58*	Quinolone Analogues. Synthesis of 3-Heteroaryl-1,4-dihydro-1-methylpyridazino[3,4-b]quinoxalin-4-ones
*30-PO-58*			205
	Y. Kurasawa (Kitasato University, Japan)

*30-PO-59*	Three-Step Total Synthesis of Luotonin A and Six-Step Formal Synthesis of Mappicine by Intramolecular Hetero Diels-Alder Reaction
*30-PO-59*			206
	M. Toyota, C. Komori, M. Ihara (Tohoku University, Japan)

*30-PO-60*	Application of Dimeric 1,2,4-Triazines in the Synthesis of Symmetrical and Unsymmetrical Biheteroaromatic Systems
*30-PO-60*			207
	A. Rykowski, D. Branowska, J. Kielak (University of Podlasie, Poland)

*30-PO-61*	The Haloform Synthesis of 1,3,3,5,5-Penta-alkyl-piperazin-2-ones: Correction of the Important Byproduct Structure
			208
	P. Nesvadba (Ciba Specialty Chemicals Inc., Switzerland)

*30-PO-62*	Heterocyclization of [60]Fullerene		209
	M. Ohno (Toyota Technological Institute, Japan) H. Ishida, K. Itoh (Nagoya University, Japan)

*30-PO-63*	Novel Synthesis of 4H-1,3-Thiazines and 4H-1,3-Oxazines from 3‑N‑Acylamino Alcohols
*30-PO-63*			210
	T. Nishio, Y. Konno, E. Kimura, M. Ori (University of Tsukuba, Japan)

*30-PO-64*	Synthesis of Heterocycle-fused Azulenes from 1-Acetyl- and 1-Formyl substituted 2-Methoxyazulenes
*30-PO-64*			211
	D.-L. Wang, H. Tanaka, K. Imafuku (Kumamoto University, Japan)

*30-PO-65*	Cycloaddition of N-Aryl Substituted Ketenimines under High Pressure		212
	M. Shimizu, A. Oishi, Y. Taguchi, Y. Gama, I. Shibuya (National Institute of Advanced Industrial Science and Technology(AIST), Japan)

*30-PO-66*	Synthesis: of Pyran-4-ones from Isoxazoles		213
	C. S. Li, E. Lacasse (Merck Frosst Canada & Co, Canada)

*30-PO-67*	Regio- and Diastereoselective Cycloaddition Reaction of N-Methyl Nitrones Derived from 3-(Allylamino)propionaldehydes
			214
	M. Noguchi, J. Hikata, M. Tanaka, H. Yamamoto (Yamaguchi University, Japan)

*30-PO-68*	Synthetic Studies on Polycyclic Guanidine Alkaloids		215
	K. Nagasawa (The University of Tokyo, / RIKEN (The Institute of Physical and Chemical Research), Japan) A. Georgieva, T. Ishiwata, H. Koshino, T. Nakata (RIKEN (The Institute of Physical and Chemical Research), Japan) Y. Hashimoto (The University of Tokyo, Japan)

*30-PO-69*	Synthesis, Antithrombin Activity, and Acute Toxicity of Substituted 3,5-Dihydroxy-3,5-dihydro-2-pyrrolones
			148
	E. A. Goun, D. H. Miles (University of Central Florida, USA) O. P. Krasnykh, S. J. Solodnikov, A. N: Masliwets, N. A. Konjuhova (Perm State University, Russia)
	Program No.: 30-OP-3 (C-1)

*30-PO-70*	Synthesis of Nucleosides with Four-membered Heterocyclic Sugars as Potential Antiviral Agents
			149
	E. Ichikawa (The University of Tokyo, Japan) S. Yamamura (Keio University, Japan), Y. Terada (Meijyo University, Japan), K. Kato (Nippon Kayaku Co.Ltd., Japan)
	Program No.: 30-OP-7 (C-2)

*30-PO-71*	Mechanistic Insights and Synthesis of Novel Lactam and Peptide based Templates for Serine Protease Inhibition
			150
	J. Seibel, R. Wilmouth, C. Schofield (University of Oxford, UK)
	Program No.: 30-OP-11 (C-3)

*30-PO-72*	Aldol and Arylmethylene Derivatives of 4-Piperiodones		151
	M. J. Turmuchanova, G. S. Litvinenko, D. G. Kim (The Al-Farabi Kazakh State University, Kazakhstan) J. R. Dimmock (University of Saskatchewan, Canada)
	Program No.: 30-OP-15 (C-4)

*30-PO-73*	Synthesis of Purines with Inhibitory Activity against Mycobacterium Tuberculosis
			152
	A. K.Bakkestuen, A. Bråthe, L-L. Gundersen, G. Langli, J. Nolsøe (University of Oslo, Norway)
	Program No.: 30-OP-19 (C-5)

*30-PO-74*	*Solid-Phase Synthesis of Dihydropyrimidones via N-Acyliminium Ion Based α-Ureidoalkylations*
			153
	D. Dallinger, M. Gercía Valverde, C. O. Kappe (Karl-Franzens-University Graz, Austria)
	Program No.: 30-OP-23 (C-6)

*30-PO-75*	Selective Electroreductive Cyclization of Nitrogen-Containing Nonconjugated Enones and Ynones
*30-PO-75*			154
	I. Nishiguchi, S. Goda, H. Maekawa (Nagaoka University of Technology, Japan)
	Program No.: 30-OP-27 (C-7)

*30-PO-76*	Polymer Supported Oligosaccharide Synthesis by Use of Real Time Reaction Monitoring Method
*30-PO-76*			155
	S. Manabe, H. Ando, Y. Nakahara, Y. Ito (RIKEN (The Institute of Physical and Chemical Research), Japan)
	Program No.: 30-OP-31 (C-8)

*30-PO-77*	Synthesis of Fluorine-Containing Heterocycles for Agrochemicals, Pharmaceutical and Polymers
*30-PO-77*			156
	J. S. Ji, P. O. Lu, R. Y. Yang (Shanghai High Victory Science & Technology Co.,Ltd., China)
	Program No.: 30-OP-35 (C-9)

*30-PO-78*	Synthesis, Chemistry, and Applications of Heterocyclic Case Compounds(V)		157
	H.-J. Wu, H.-C. Lin, Z. Wang, C.-Y. Wu (National Chiao Tung University, Taiwan)
	Program No.: 30-OP-39 (C-10)

*30-PO-79*	Regioselective Synthesis of Alkynylbenzotriazoles		158
	T. Kitamura, N. Tashi, H. Chen, Y. Fujiwara (Kyushu University, Japan)
	Program No.: 30-OP-43 (C-11)

*30-PO-80*	Efficient Anodic Synthesis of 2-Fluoro and 2, 3-Difluorobenzofuran Derivatives
*30-PO-80*			159
	K. M. Dawood (Tokyo Institute of Technology, Japan/ Cairo University, Egypt) H. Ishii, T. Fuchigami (Tokyo Institute of Technology, Japan)
	Program No.: 30-OP-47 (C-12)

*30-PO-81*	2H-Pyran-2-ones as Synthons for the Synthesis of α,b-Didehydro-α-amino Acid Derivatives
*30-PO-81*			160
	L. Vraničar, S. Polanc, M. Kocevar (University of Ljubljana, Slovenia)
	Program No.: 30-OP-51 (C-13)

*30-PO-82*	2-Heteroaryl-1,4-Dihydropyrimidines-Novel and Potent Non-Nucleosidic Inhibitors of Hepatitis B Virus (HBV)
			161
	S. Goldmann, J. Stoltefuss, U. Niewöhner, T. Krämer, E. Graef, S. Lottmann, K. Deres, R. Masantschek, D. Koletzki, O. Weber, A. Paessens (BAYER AG, Germany)
	Program No.: 30-OP-55 (C-14)

*30-PO-83*	Synthetic Studies of Physiologically Active Natural Product by Using the Novel Lewis Acid Generated from Boron Trifluoride Diethyl Etherate and Trimethylsilyl Triflate

			216
	M. Sato, K. Horita, S. Nishibe (Health Sciences University of Hokkaido, Japan)

*30-PO-84*	Synthesis of b-Carboline Derivatives Linked to N-Methyl-N-nitrosourea at N9 Atom and Improved Minor Groove, Selectivity in Methylation of DNA
			217
	T. Konakahara, Y. Nishida, K. Kobayashi, S. Ohno, N. Sakai (Science University of Tokyo, Japan)

*30-PO-85*	Development of a New-Style Triphase Catalyst and Its Application to Epoxidation of Allylic Alcohols
			218
	Y. M. A. Yamada, M. Ichinohe, H. Takahashi, S. Ikegami (Teikyo University, Japan)

*30-PO-86*	Synthesis of Pyridine Derivatives Using Ketene Dithioacetals. II: Synthesis of 2,2'-Dipyridyl Derivatives with the Fluorescence Property		219
	N. Mizuyama, Y. Tominaga (Nagasaki University, Japan) Y. Shigemitsu (Technology Center of Nagasaki, Japan) S. Hirayama (Sasebo National College of Technology, Japan)

*30-PO-87*	Ruthenium(II)-Catalyzed Cycloaddition of 1,6-Diynes with Heterocumulenes Providing Heterobicycles
			220
	Y. Yamamoto, H. Takagishi, K. Itoh (Nagoya University, Japan)

*30-PO-88*	Chalcogeno-Baylis-Hillman Reactions via Cyclic Sulfonium Ion Intermediates
			221
	T. Kataoka, S. Kinoshita, M. Fujita, H. Kinoshita, T. Iwamura, S. Watanabe (Gifu Pharmaceutical University, Japan)

*30-PO-89*	Synthesis, Fluorescent Properties and Stereoselective Reduction of 3- Aryl-4-methylthiomaleimides
			222
	Y. Shigemitsu (Industrial Technology Centre of Nagasaki, Japan) Y. Tominaga (Nagasaki University, Japan)

*30-PO-90*	Synthesis and Activity of Indoles Substituted by Heteroaromatics at 3-Position
			223
	A. Nishida, M. Fuwa, M. Nakagawa (Chiba University, Japan)

*30-PO-91*	Synthesis of Benzoxazines by the Mannich-type Reaction of Phenols		224
	Y. Tanaka, Y. Irisa, Y.Taruno, M. Morimoto, H. Saimoto, Y. Shigemasa, Y. Okamoto, S. Minami (Tottori University, Japan)


*30-PO-92*	1,2,3-Triazole Derivatives as Carbenoid Source: Formation of Mesoionic 1,3-Oazolium-4-olate and 1,3-Thiazolium-4-olate
*30-PO-92*			225
	H. Nakano, K. Horii, N. Ito (Aichi University of Education, Japan)

*30-PO-93*	A Facile Synthetic Way to Polycyclic Compounds by One-Pot Reactions of Allenes with Palladium Catalysts: Asymmetric Synthesis of Cyclic Indole Compounds

			226
	Y. Hiratsuka, K.Watanabe, I. Abe, F. Kato, M. Hiroi, K. Hiroi (Tohoku Pharmaceutical University, Japan)

*30-PO-94*	Total Syntheses of Riccardin A and Isoplagiochin D by the Intramolecular Pd(0) Catalyzed Stille-Kelly Reaction
			227
	H. Takahashi, N. Sato, T. Mori, H. Yaso, Y. Fukuyama (Tokushima Bunri University, Japan)

*30-PO-95*	Synthesis of [1,2,3]Triazolo[1,5-a]pyrazines		228
	T. Jug, T. Trček, B. Verček (University of Ljubljana, Slovenia)

*30-PO-96*	Formation of Cyclic Polysulfides by the Reaction of 2,4,6-Trisubstituted 5,6-Dihydro-1,3,5-dithiazines with Oxidizing Agents
			229
	Y. Takikawa, K. Suzuki, Y. Fujisawa, S. Aoyagi, K. Shimada (Iwate University, Japan)

*30-PO-97*	Total Syntheses of b-Carboline Alkaloids, Pyridindolol K1, Pyridindolol K2, and Pyridindolol
*30-PO-97*			230
	S. Hibino, N. Kanekiyo, T. Kuwada, J. Nobuhiro, T. Choshi (Fukuyama University, Japan)

*30-PO-98*	Total Syntheses of Carbazole Alkaloids, Carbazomycin G, Murrayaquinone A and Furostifoline		231
	T. Choshi, H. Hagiwara, H. Fujimoto, J. Nobuhiro, S. Hibino (Fukuyama University, Japan)

*30-PO-99*	Hexahydro-1H-Pyrrolo[1,2-c]imidazolone: A Novel Chiral Unit Identified from Parallel Synthetic Libraries of Bicyclic N-Chiral Amines
			232
	Y. Uozumi, K. Yasoshima, K. Shibatomi (Institute for Molecular Science, Japan) K. Mizutani, T. Miyachi, S. Nagai (Nagoya City University, Japan)

*30-PO-100*	Chiral Bis-pyridino-18-crown-6•Lanthanide Triflate Complexes as Effective Catalysts for Asymmetric Aldol Reactions in Aqueous Media
			233
	K. Manabe, T. Hamada, S. Kobayashi (The University of Tokyo, Japan)

*30-PO-101*	Catalytic Asymmetric Reactions of Aldehydes Using a Chiral Zirconium Catalyst
*30-PO-101*			234
	Y. Yamashita, H. Ishitani, H. Shimizu, S. Saito, S. Kobayashi (The University of Tokyo, Japan)

*30-PO-102*	C-Phosphorylation of Heteroaromatic Compounds in Synthesis of Novel Phosphorus-Containing Heterocycles
			162
	A. A. Tolmachev, A. Kostyuk (National Academy of Sciences of Ukraine, Ukraine)
	Program No.: 30-OP-4 (D-1)

*30-PO-103*	Neighboring Effect of Heteroaromatic Rings for the π-Facial Selectivity		163
	T. Kobayashi, T. Tsuzuki, K. Miki, Y. Tayama (Shinshu University, Japan)
	Program No.: 30-OP-8 (D-2)

*30-PO-104*	Formation of Iminosubstituted Propadienethiones by Thermal (FVP) and Electron Impact, Induced Fragmentation of Multisulfur Heterocycles
			164
	C. T. Pedersen (USD, Odense University, Denmark) R. Flammang (University of Mons-Hainaut, Belgium) E. Fanghanel (Martin Luther University, Halle Wittenberg, Germany)
	Program No.: 30-OP-12 (D-3)

*30-PO-105*	1,4,5,8-Tetraazafulvalenes - New Starting Material for Functional Dyes		165
*30-PO-105*	R. Beckert, C. Käpplinger, D. Müller (Friedrich-Schiller-University, Germany)
	Program No.: 30-OP-16 (D-4)

*30-PO-106*	Anomalous Carbon Insertion into a Benzene Ring in Bischler-Napieralski Reaction
*30-PO-106*			166
	T. Ishikawa, K. Shimooka, T. Narioka (Chiba University, Japan)
	Program No.: 30-OP-20 (D-5)

*30-PO-107*	Synthesis and Properties of Pyrroles and Porphyrins Fused with Rigid Bicyclic Rings
*30-PO-107*			167
	H. Uno, S. Ito, K. Nakamoto, H. Watanabe, M. Wada, N. Ochi, N. Ono (Ehime University, Japan)
	Program No.: 30-OP-24 (D-6)

*30-PO-108*	Photochromic Imidazole: A Novel Material		168
	A. K. Padhy (National Institute of Science & Technology, India)
	Program No.: 30-OP-28 (D-7)

*30-PO-109*	New Approach to Synthesis of 4-Piperidones		169
	D. G. Kim (The Atyrau Institute of Scientific and Technical Problems, Kazakhstan)
	Program No.: 30-OP-32 (D-8)

*30-PO-110*	Chiral Relay Auxilliaries		170
*30-PO-110*	V. K. Tandon, S. Rai (Lucknow University, India)
	Program No.: 30-OP-36 (D-9)

*30-PO-111*	Synthesis of Benzolactones and Benzolactams by Aryl Radical Carbonylation
*30-PO-111*			171
	K. Orito, T. Tatsuzawa, R. Harada, M. Tokuda (Hokkaido University, Japan)
	Program No.: 30-OP-40 (D-10)

*30-PO-112*	A New Method for the Preparation of Enantiomerically Purea-Substituted Pyrrolidines
*30-PO-112*			172
	T. Maki, Y. Ishida, K.Shirai, O. Onomura, Y. Matsumura (Nagasaki University, Japan)
	Program No.: 30-OP-44 (D-11)

*30-PO-113*	The Isolation of the First Stable Atropisomers in Proximity-Screened NZ,NZ-diazasesquinorbornanes (N²[2]polynorbornanes)
*30-PO-113*			173
	R. N. Warrener, G. Sun (Central Queensland University, Australia)
	Program No.: 30-OP-48 (D-12)

*30-PO-114*	Synthesis of Novel, Axially Chiral 1,8-Disubstituted Naphthalenes		174
	A. V. Bedekar, S. Yoshikawa, K. Tanaka (University of Shizuoka, Japan)
	Program No.: 30-OP-52 (D-13)

*30-PO-115*	Synthesis of Pyridine Derivatives Using Aminoacroleins as an Equivalent of Malonaldehydes
*30-PO-115*			175
	H. Suda, H. Saitoh, K. Umihara, Y. Furugori, I. Itoh (Sankio Chemical Co., Ltd., Japan)
	Program No.: 30-OP-56 (D-14)

*30-PO-116*	*Synthesis of Pyrrolo- and Thienopyrimidines peri-Fused with Pyrimidine, 1,4-Diazepine and 1,4-Thiazepine Rings*
*30-PO-116*			235
	Z. Sarakauskaite, S. Tumkevicius, V. Masevicius (Vilnius University, Lithuania)

*30-PO-117*	Inhibition of HIV Integrase by 4-Hydroxy Coumarin Dimer Bearing Aniline Mustard Moiety
*30-PO-117*			236
	L-Y. Hsu (National Defense Medical Center, Taiwan) P. C.-M. Mao (Veterans General Hospital Kaohsiung, Taiwan) J.-F. Mouscadet, H. Leh, C. Auclair (Institut Gustave Roussy, France)

*30-PO-118*	The Synthesis and Antimicrobial Activity of New 4,5-Dithiazole Derivatives		237
	L Preda, O. Oniga, B. Tiperciuc (The University of Medicine and Pharmacy "Iuliu Hatieganu” Roumania)

*30-PO-119*	Quaternary Ammonium Compounds with Thiazol Active on Botrytis Cinerea and Fusarium Oxysporum Vegetal Fungi
*30-PO-119*			238
	M. Palage, A. Muresan (The University of Medicine and Pharmacy "Iuliu Hatieganu” Romania) M. Parvu (The University Babes-Bolyai, Roumania)

*30-PO-120*	Selective Suzuki Coupling Reactions at Dibromo-thiophenes		239
	J. Fröhlich, V. Peutsch, C. Hametner (Vienna University of Technology, Austria)

*30-PO-121*	Novel Specific Inhibitors of Puromycin-Sensitive Aminopeptidase		240
	H. Kakuta, H. Takahashi, K. Nagasawa, Y. Hashimoto (The University of Tokyo, Japan)

*30-PO-122*	Design, Synthesis and Bioactivity of Leflunomide Derivatives as Novel Immunomodulatory Agents
*30-PO-122*			241
	W.-H. Huang, A.-R. Lee (National Defense University, Taiwan)

*30-PO-123*	Synthesis and Fungicidal Activity of Novel FlavanoneAnalogues		242
	G. Yang, Y. Ding, X. Jiang (Central China Normal University, China)

*30-PO-124*	*Interactions of Peptides Derived from E.coli* RecA, Protein with Single-stranded Oligonucleotides Containing 5-Formyl-2’-deoxyuridine**
*30-PO-124*			243
	T. Sugiyama, R. Kuroda (The University of Tokyo, Japan) " A. Kittaka, H.Takayama (Teikyo University, Japan) M. Tomioka, Y. Ida (Showa University, Japan)

*30-PO-125*	Introduction of Formyl-bearing Uracil Bases into Oligonucleotides: Effects to Sequence Specific and Non-Specific DNA Binding Proteins
*30-PO-125*			244
	A. Kittaka, H. Takayama (Teikyo University, Japan) T. Sugiyama, R. Kuroda (The University of Tokyo, Japan) M. Kurihara (National Institute of Health Sciences, Japan) J. Inoue (Keio University, Japan)

*30-PO-126*	Synthesis and Biological Activity of Tricyclic Indole Derivatives as Na⁺/H⁺Exchanger Inhibitors
*30-PO-126*			245
	M. Kitano, K. Nakano, K. Matsui, N. Ohashi (Sumitomo Pharmaceuticals Co., Lid., Japan)

*30-PO-127*	A Novel Synthesis of L-Ribose from D-Mannono-1,4-lactone		246
	H. Takahashi, Y. Iwai, Y. Hitomi, S. Ikegami (Teikyo University, Japan)

*30-PO-128*	Facile Synthesis and Structure Elucidation of Novel Spiro-cyclodisaccharides
*30-PO-128*			247
	X. Li, H. Takahashi, H. Ohtake, S. Ikegami (Teikyo University, Japan)

*30-PO-129*	Synthesis of Optically Active TAN-67, Highly Selective Delta Opioid Receptor Agonist, and Investigation of its Pharmacological Properties
*30-PO-129*			248
	H. Fujii, K. Kawai, K. Kawamura, A. Mizusuna, Y. Onoda, M. Murachi T. Tanaka, T. Endoh, H. Nagase (Toray Industries, Inc., Japan) Y. Yajima, M. Narita, J. Kamei, T. Suzuki (Hoshi University, Japan)

*30-PO-130*	Synthesis of Metabolites for Potent Na⁺/H⁺ Exchanger Inhibitor SM-20550		249
	M. Yuri, M. Kitano, K. Matsui, N. Ohashi (Sumitomo Pharmaceuticals Co., Lid., Japan) M. Yabuki, H. Nishibe, H. Kanamaru (Sumitomo Chemical Co., Lid., Japan)

*30-PO-131*	Synthesis of 5-(N'-Sulfonylureido)pyrazole Derivatives and their Endothelin Converting Enzyme Inhibitory Activities
*30-PO-131*			250
	H. Hasegawa, K. Umekawa, Y. Kuribayashi, N. Ohashi (Sumitomo Pharmaceuticals Co., Lid., Japan)

*30-PO-132*	A Nitroisoflavone-Salicoylindole-Ring Transformation		251
	R. Albuschat, S. Tappmeyer, W. Löwe (Freie Universität Berfin, Germany)

*30-PO-133*	Synthesis of (Z)-3-[(4-Oxo-1H-pyridine-2-yl)methylidenyl]indolin-2-one		252
	W. Löwe, A. Lumetzberger, C. Dietrich, M. Weber, P. Luger (Freie Universität Berlin, Germany)

*30-PO-134*	3-Arylaminoalkylamino-5-phenylpyridazines as Novel Substrates for Acyl‑CoA: Cholesterol O-Acyltransferase
*30-PO-134*			253
	D. Barlocco (University of Milan, Italy) M. P. Giovannoni, V. Dal Piaz (University of Florence, Italy) B. M. Kwon, Y. K. Kim (Korea Res. Inst. Biosc. & Biotec., Korea) L. Toma (University of Pavia, Italy)

*30-PO-135*	Tris(2,6-diphenylbenzyl)silyl Group as a New and Highly Effective Protector for Carboxylic Acids and Ketone Carbonyls
*30-PO-135*			254
	S. Shirakawa, A. Iwasaki, K. Maruoka (Kyoto University, Japan)

*30-PO-136*	Mild Air-Oxidation of Activated Carbonyl Compounds with Cesium Salts: Application to the Construction of a Model Ring Unit of Camptothecin
*30-PO-136*			255
	T. Watanabe, T. Ishikawa (Chiba University, Japan)
*30-PO-137*	Synthesis of Cycloalkano-Oligopyrroles and Their Structures		256
*30-PO-137*	Y. Fumoto, H. Uno, N. Ono (Ehime University, Japan)		256

*30-PO-138*	Synthesis and Properties of Thiophene Derivatives Fused with Bicyclo[2.2.2]octadiene
*30-PO-138*			257
	Y. Shimizu, S. Ito, H. Uno, T. Ogawa, N. Ono (Ehime University, Japan)

*30-PO-139*	Application of 2-(3,5,6-Trifluoro-2-hydroxy-4-methoxyphenyl) benzoxazole and -thiazole to Fluorescent Probes Sensing pH and Metal Cation
*30-PO-139*			258
	K. Tanaka, T. Kumagai, H. Aoki, M. Deguchi, S. Iwata (Seikei University, Japan)

*30-PO-140*	Raections of Heterocyclic Quinone Methides		259
	S. Thamarai Salvi, R. Nandha Kumar, T. Suresh, P. S. Mohan

*30-PO-141*	Chemical Behaviour of 5-(2-Phenyl-thiazol-4-yl)-[1,2,4]-triazol-3-thione		260
	V. Zaharia, H. Miresan (University of Medicine and Pharmacy "luliu Hatieganu”; Romania)

*30-PO-142*	Oxidation of 2-Aminomethylpyridine: Synthesis of Symmetrical N‑Heterocycles
*30-PO-142*			261
	Y. Yamaguchi, Y. Okamoto (Kitasato University, Japan)

*30-PO-143*	Synthesis of Peptide-containing 3,5-Dioxa-12-azawurtzitanes		262
	H. Izumi, S. Futamura (National Institute of Advanced Industrial Science and Technology, Japan)

*30-PO-144*	Synthesis of New Functional Compounds Having Ferrocene Moiety Related to π-Extended Tetrathiafulvalenes
*30-PO-144*			263
	A. E.-W. Sarhan, M. Murakami, T. Izumi (Yamagata University, Japan)

*30-PO-145*	Synthesis of Chiral Binaphthyl Ligands Using Enzymatic Amidation		264
	N. Aoyagi, T. Izumi (Yamagata University, Japan)

*30-PO-146*	*Preparation of 2-Alkyl/Arylfuro[3,2-c]quinoline-4(5H)-ones viaMolecular Rearrangement of 4-Alkyl/Aryl-3-bromopyrano[3,2-c]quinoline-2,5(2H,6H)-diones*
*30-PO-146*			265
	A. Klásek, K. Kořistek (Tomas Bata University, Czech Republic) P. Sedmera (Academy of Sciences of the Czech Republic, Czech Republic)

*30-PO-147*	Synthesis and Reactivity of 3-Alkyl/Aryl-3-thiocyanato-2,4(1H,3H)- quinolinediones
*30-PO-147*			266
	A. Klásek, J. Polis (Tomas Bata University, Czech Republic) J. Kosmrlj (University of Ljubljana, Slovenia)

*30-PO-148*	Combinatorial Libraries of Condensed Heterocycles Containing the 2‑Mercapto-4(3H)-pyrimidinone Fragment
*30-PO-148*			267
	A. Ivachtchenko, S. Kovalenko, A. Ilin, A. Drushlyak (Chemical Diversity Labs, Inc., USA)

*30-PO-149*	*Combinatorial Libraries of Benzimidazo[1,2-c]-6(5H)-Quinazolines*		268
	A. Ivachtchenko, S. Kovalenko, A. Drushlyak (Chemical Diversity Labs, Inc., USA)

*30-PO-150*	An Efficient Conversion of Aryl Esters to Benzthiazoles		269
	A. K. Chakraborti, L. Sharma (National Institute of Pharmaceutical Education and Research (NIPER), India)

*30-PO-151*	Synthesis of Thiazoles from Aldehydes in a One-Pot Reaction		270
	A. K. Chakraborti, G. Kaur (National Institute of Pharmaceutical Education and Research (NIPER), India)

*30-PO-152*	Synthesis of 6-Phenyl-1,2,3,4-rahydrodibenzo[b,g][1,8]naphthyridines		271
	G. A. Prakash, S. P. Rajendran (Bharathiar University, India)

*30-PO-153*	Synthesis of 2-Acetyl-3(2'-oxoquinolinyl)-5phenylpyrazolines		272
	S. P. Rajendran, P. Meenasundari (Bharathiar University, India)

*30-PO-154*	Synthesis and Properties of Novel Macrocyclic Thiourea Derivatives		273
	Y. Okumura, N. Matsumura, K. Mizuno (Osaka Prerecture University, Japan)

*30-PO-155*	Synthesis and Ring Modification of [2]Catenane		274
	T. Takata, N. Watanabe, N. Kihara (Osaka Prerecture University, Japan)

*30-PO-156*	Superacidic Media: a New Tool in Medicinal Chemistry VINFLUNINE: the First Exampe of this Use
*30-PO-156*			275
	A. Duflos, J. Fahy, F. Redoules, J. C. Tristani (Pierre Fabre Research Centre of Castres, France) J. C. Jacquesy (University of Poitiers, France)

*30-PO-157*	Synthesis of a New Diels-Alder Quinone Adduct and Its Use in Preparing Thiazolo- and Oxazolo-quinolines
*30-PO-157*			276
	A. S. Hammam, M. S. Kamel, S. M. Radwan, M. A. Abdel Rahman (Assiut University, Egypt)

*30-PO-158*	Enaminone in Heterocyclic Synthesis: New Routes for the Synthesis of Polyfunctionally Substituted Five-and/or Six-membered Heteroaromatics and their Condensed Derivatives
*30-PO-158*			277
	Z. E. Kandeel (Cairo University, Egypt)

*30-PO-159*	Preliminar Theoretical Studies in the Design of Antitumor Drugs: Putrescine Derivatives
*30-PO-159*			278
	M. Legaspi, A. Robinsohn, G. Rodrigo, B. Fernández, S. Sicardi, M. Hedrera (Universidad de Buenos Aires, Argentina)

*30-PO-160*	Design of New Quinoxaline and Benzoquinoxaline Analogs as Antineoplastic Agents
*30-PO-160*			279
	G. Rodrigo, V. Baez, A. Robinsohn, M. Hedrera, S. Sicardi, B. Fernandez (Universidad de Buenos Aires, Argentina)

*30-PO-161*	A Convenient Method for Direct Acylation of Indoles at the 3-Position with Acyl Chlorides in the Presence of Dialkylaluminum Chloride
*30-PO-161*			280
	T. Okauchi, M. Itonaga, H.Matsueda, T. Minami (Kyusyu Institute of Technology, Japan)

*30-PO-162*	*Synthesis of 4,6-Dialkyl-5,7(4H,6H)-furazano[3,4-d]pyrimidinediones Using Sulfilimine*
*30-PO-162*			281
	M. Takahashi, N. Matsumoto (Ibaraki University, Japan)

*30-PO-163*	Anionic Cycloaromatization of (Z)-2-(6-Substituted-3-hexen-1,5- diynyl)benzonitriles Initiated by Methoxide Addition: Synthesis of Phenanthridinones and Benzo[c]phenanthridinones
*30-PO-163*			282
	M.-J. Wu, C.-F. Lin, W.-D. Lu (Kaohsiung Medical University, Taiwan)

*30-PO-164*	*A Novel Synthesis of Substituted 3,6-Dihydro-1H-Benzo[c]oxocines via* Claisen Rearrangement and RCM**
*30-PO-164*			283
	E.-C. Wang, K.-S. Huang, C.-C.Wang, M.-K. Hsu, J.-R. Lin (Kaohsiung Medical University, Taiwan)

July 31 (Tue)			Oral Presentation
14:10 - 15:20		SECTION A (Room 301)
Chair: A. Kubo (Meiji Pharmaceutical Univeristy, Japan)
*A-15*	Synthesis of Some New 1,8-Naphthyridine Derivatives of Expected Biological Activity
				284
	O. A. Fathalla, M. Kamel, M.I. El-Zahar, E. M. M. El-Deen (National Research Centre, Egypt) M. Refai (Ain Shams University, Egypt)
	Program No.: 31-OP-57 Poster No.: 31-PO-1

*A-16*	Enantioselective Synthesis of the Tetracyclic Left-Hand Substructure of Solanoeclepin A
				285
	J. C. J. Benningshof, M. IJsselstijn, S. R. Wallner, R. H. Blaauw, A. E. van Ginkel, F. P. J. T. Rutjes, H. Hiemstra (University of Amsterdam, The Netherlands)
	Program No.: 31-OP-61 Poster No.: 31-PO-2

*A-17*	Enantioselective Total Synthesis of Eudistomin C			286
	H. Tokuyama, T.Yamashita, N. Kawai, T. Fukuyama (The University of Tokyo, Japan)
	Program No.: 31-OP-65 Poster No.: 31-PO-3

*A-18*	Stereoselective Total Synthesis of Zaragozic Acid A			287
	M. Kikuchi, K. Igawa, M. Suzuki, K. Ping-Huai, T. Nakai, K. Tomooka (Tokyo Institute of Technology, Japan)
	Program No.: 31-OP-69 Poster No.: 31-PO-4

*A-19*	Asymmetric Total Synthesis of CDC25A Inhibitor Dysidiolide and Its Potent Analogs
				288
	R. Shirai, K.Dodo, K.Koga (NaraInstitute of Science and Technology, Japan) M. Takahashi, Y. Hashimoto (The University ot Tokyo, Japan)
	Program No.: 31-OP-73 Poster No.: 31-PO-5

*A-20*	Synthetic Study of Ciguatoxin CTX3C			289
	T. Oishi, H. Uehara, M. Maruyama, H. Imai, Y. Nagumo, M. Shoji, K.Maeda, J.-Y. Le Brazidec, M. Kosaka, H. Oguri, M. Hirama (Tohoku University / CREST, Japan)
	Program No.: 31-OP-77 Poster No.: 31-PO-6

*A-21*	Synthesis of Methylcoriandrin			290
	K. Datta, M. Bandyopadhyay, D. Mal (Indian Institute of Technology, India)
	Program No.: 31-OP-81 Poster No.: 31-PO-7

*A-22*	Asymmetric Synthesis of (R)-3-Methylpyrrolidine Alkaloids			291
	X. Zheng, Y. P. Ruan (Xiamen University, China) P. Q. Huang (Lanzhou University/ Xiamen University, China) A. W. M. Lee, W. H. Chan (Hong Kong Baptist University, China)
	Program No.: 31-OP-85 Poster No.: 31-PO-8

*A-23*	Cyanothiocetamide in Heterocyclic Synthesis: Synthesis of Pyridinethione, 2‑S-Alkylpyridine, Thieno[2,3-b]pyridine, Pyrazolo[4,3-c]pyridine and Thiopyrano[2,3-b]pyridine Derivatives
				292
	F.A. Attaby, Y. M. Ibrahim (Cairo University, Egypt)
	Program No.: 31-OP-89 Poster No.: 31-PO-51

14:10 - 15:20		SECTION B (Room 302)
Chair: Y. Yokoyama (Toho University, Japan)
*B-15*	Efficient Cyclization of Ether Ring Using Sml₂			293
	F. Matsuda. H. Tamiya (Hokkaido University, Japan)
	Program No.: 31-OP-58 Poster No.: 31-PO-40

*B-16*	Tetrahydropyrrolo[3,2-c]pyridines. Synthesis and Reactivity			294
	L. G. Voskressensky, A. V. Varlamov, T. N. Borisova (Russian Peoples Friendship University, Russia)
	Program No.: 31-OP-62 Poster No.: 31-PO-41

*B-17*	Studies Directed toward the Total Synthesis of Mycalamides- Stereoselective Construction of the Right- and Left-Half Segments
				295
	M. Toyota, M. Hirota, H. Hirano, N. Kagawa, M. Ihara (Tohoku University, Japan)
	Program No.: 31-OP-66 Poster No.: 31-PO-42

*B-18*	Regioselective BH₃-hydride Reduction of Inosine Derivatives			296
	K. Hirota, R. Hattori, H. Sajiki. Y. Monguchi (Gifu Pharmaceutical University, Japan), O. Muraoka, G. Tanabe (Kinki University, Japan)
	Program No.: 31-OP-70 Poster No.: 31-PO-43

*B-19*	Lithio-1,2,4-triazines-Synthesis, Structure, Synthetic Potential			297
	H. Neunhoeffer, T. Hundsdorf (Darmstadt University of Technology, Germany)
	Program No.: 31-OP-74 Poster No.: 31-PO-44

*B-20*	Novel Carbon-Carbon Bond Formation Reaction of Methoxyallene Oxide Promoted by Til₄
				298
	M. Shimizu, R. Hayakawa, I. Hachiya (Mie University, Japan)
	Program No.: 31-OP-78 Poster No.: 31-PO-45

*B-21*	Enantioselective Coniugate Additions of Thiols and β-Keto Esters Catalyzed by Chiral N-Oxide-Metal Complexes
				299
	M. Nakajima, M. Saito, Y. Yamaguchi, S. Hashimoto (Hokkaido University, Japan)
	Program No.: 31-OP-82 Poster No.: 31-PO-46

*B-22*	Solid/Liquid Phase Synthesis of b-Strand Mimetic Templates via Regioselective 1,3-Dipolar Cycloaddition
				300
	N. Fuchi, T. Doi, T. Takahashi (Tokyo Institute of Technology, Japan) M. Kahn (University of Washington, USA)
	Program No.: 31-OP-86 Poster No.: 31-PO-47

*B-23*	Chemistry of 1,6-Disila[4.4.4]propellane and Related Compounds			301
	A. Toshimitsu, M. Katkevics, A. Sano, M. Asahara, T. Miki, H. Fujimura, H. Tsuji, S. Yamaguchi, K. Tamao (Kyoto University, Japan)
	Program No.: 31-OP-90 Poster No.: 31-PO-147

14:10 - 15:20		SECTION C (Room 303)
Chair: Y. Mori (Meijo University, Japan)
*C-15*	Synthesis and Biological Evaluation of 4,5-Dihydronaphtho[1,2-d]1,2,3-thia- or selenadiazole Derivatives
				302
	M. Daneshtalab (Memorial University of Newroundland, Canada) A. R. Jalilian, M. Binesh-Marvasti, A. Shafiee (Tehran University of Medical Sciences, Iran) S. Sattari (University of Alberta, Canada)
	Program No.: 31-OP-59 Poster No.: 31-PO-92

*C-16*	Fluorescent Rhodacyanine Dyes as Antimalarial Agents: Library Construction and Structure-Activity Relationship
				303
	K. Takasu, H. Inoue, M. Ihara (Tohoku University, Japan) H. -S. Kim, Y. Wataya (Okayama University, Japan)
	Program No.: 31-OP-63 Poster No.: 31-PO-93

*C-17*	Discovery of Novel Aspartyl Ketones as Potent Caspase-3 Inhibitors			304
	Y. Han, A. Giroux, E. L. Grimm, R. Aspiotis, C. I. Bayly, D. J. Mckay, S. Roy, S. Xanthodakis, J. Valancourt, D. M. Rasper, J. Tam, P. Tawa, D. W. Nicholson, R. J. Zamboni (Merck Frosst Canada & Co., Canada) N. A. Thornberry, E. P. Paterson, M. Garcia-Calvo, J. W. Becker, J. Rotonda (Merck Research Laboratories, Merck & Co., Inc., USA)
	Program No.: 31-OP-67 Poster No.: 31-PO-94

*C-18*	Novel Synthesis of Substituted Indoles from 2-Aminophenols			305
	W.-M. Dai, D.-S. Guo, L.-P. Sun(The Hong Kong University of Science and Technology, China)
	Program No.: 31-OP-71 Poster No.: 31-PO-95

*C-19*	Heterocyclic-fused Naphthalimides: Synthesis Via Unusual Pschorr Cyclization, Spectral Properties and Interesting Photocleaving Action to DNA
				306
	X. Qian, J. Cui, R. Zhang (Dalian University of Technology, China) W. Yao, P. Mao (East China University of Science and Technology, China)
	Program No.: 31-OP-75 Poster No.: 31-PO-96

*C-20*	Practical Synthesis of an Indolocarbazole-based DNA Topoisomerase I Inhibitor			307
	A. Kamatani, M. Kawasaki, N. Satake, S. Hiraga, A. Akao, T. Nemoto, T. Iida, T. Mase (Banyu Pharmaceutical Co., Lid., Japan) S. A. Weissman, D. M. Tschaen, R. P. Volante (Merck Research Laboratories, USA)
	Program No.: 31-OP-79 Poster No.: 31-PO-97

*C-21*	Annelated Pyrrolo-Pyrimidines New Tricyclic DNA-Interactive Ring Systems			308
	A. M. Almerico (University of Palermo, Italy) A. Lauria, P. Diana, P. Barraja, A. Montalbano, G. Cirrincione, G. Dattolo (Università degli Studi, Italy)
	Program No.: 31-OP-83 Poster No.: 31-PO-98

*C-22*	Alkyl α-Substituted b-(Dimethylamino)-α, b-didehydro Acid Derivatives and Their Chiral Analogs-Versatile Reagents in the Synthesis of Heterocyclic Systems			309
	B. Stanovnik, J. Svete, U. Bratušek, U. Grošelj, R. Jaksě, L. Jukič Soršak, S. Pirc, S. Rečnik, C. Turk (University of Ljubljana, Slovenia)
	Program No.: 31-OP-87 Poster No.: 31-PO-99

*C-23*	The Reaction of Aldolic Condensation-Means to Obtain α-Dicarbonyls			310
	V. Zaharia, S. Imre (University of Medicine and Pharmacy "Iuliu Hatieganu”: Romania) P. Verite (University of Medicine and Pharmacy, France)
	Program No.: 31-OP-91 Poster No.: 31-PO-103

14:10 - 15:20		SECTION D (Room 304)
Chair: M. Sodeoka (Tohoku University, Japan)
*D-15*	Studies on the Self-Organization Phenomena Involving Pyridone and Phenol Derivatives
				311
	I. Takahashi, M. Wagi, M. Takahashi, H. Kitajima, M. Hatanaka, K. Isa (Fukui University, Japan) S. Hosoi, T. Ohta (Kanazawa University, Japan)
	Program No.: 31-OP-60 Poster No.: 31-PO-120

*D-16*	Synthesis of Chiral Diarylacetylene-Dicobalt Hexacarbonyls			312
	T. Sugihara, C. Harumori, H. Takao, H. Imagawa, M. Nishizawa (Tokushima Bunri University, Japan)
	Program No.: 31-OP-64 Poster No.: 31-PO-121

*D-17*	Tributylmagnesium Ate Complex Mediated Novel Bromine-Magnesium Exchange Reaction: Industrial Synthesis of a Muscarinic M₃ Receptor Antagonist
				313
	T. Iida, T. Wada, K. Tomimoto, T. Mase (Banyu Pharmaceutical Co., Ltd., Japan)
	Program No.: 31-OP-68 Poster No.: 31-PO-122

*D-18*	Introduction of Podand Histidyl Moieties into a Pyridine Scaffold to Induce a Chiral Helicity
				314
	T. Moriuchi, M. Nishiyama, K. Yoshida, T. Ishikawa, T. Hirao (OsakaUniversity, Japan)
	Program No.: 31-OP-72 Poster No.: 31-PO-123

*D-19*	New Polycyclic Aza-heterocycles, Precursors for Persistent Free Polyradicals			315
	I. A. Silberg, C. Cristea, D. Porumb (Babes-Bolyai University, Romania) M. D. Banciu (Polytechnic University, Romania) M. Danila ("C. D. Nenitzescu "Center of Organic Chemistry, Romania)
	Program No.: 31-OP-76 Poster No.: 31-PO-124

*D-20*	Tetrakis(2-thienyl)methane: First Synthesis and Synthetic Utility			316
	M. Oda, H. Nakaminami, M. Sogabe, K. Matsumoto, H. Kurata (Osaka University, Japan)
	Program No.: 31-OP-80c Poster No.: 31-PO-125

*D-21*	Greening of Cephalosporin Chemistry			317
	B. Zwanenburg, G. Kemperman, J. Zhu (University of Nijmegen, The Netherlands)
	Program No.: 31-OP-84 Poster No.: 31-PO-126

*D-22*	New Synthetic Pathways to Indole and Benzimidazole Derizatives			318
	Y. Torisawa, H. Yukawa, T. Nishi, J. Minamikawa (Otsuka Pharmaceutical Co. Ltd., Japan)
	Program No.: 31-OP-88 Poster No.: 31-PO-127

*D-23*	Evaluation of Lipophilicity of Some New Thiazolyl-oxadiazolines by Principal Component Analysis
				319
	B. Tiperciuc, S. Todor, O. Oniga (University of Medicine and Pharmacy "Iuliu Hatieganu", Romania) C. Sarbu (The University of Babes - Bolyai, Romania)
	Program No.: 31-OP-92 Poster No.: 31-PO-28

July 31 (Tue)		Poster Presentation
16:00 - 18:00

*31-PO-1*	Synthesis of Some New 1,8-Naphthyridine Derivatives of Expected Biological Activity
			284
	O. A. Fathalla, M. Kamel, M.I. El-Zahar, E.M. M. El-Deen (National Research Centre, Egypt) M. Refai (Ain Sharns University, Egypt)
	Program No.: 31-OP-57 (A-15)

*31-PO-2*	Enantioselective Synthesis of the Tetracyclic. Left-Hand Substructure of Solanoeclepin A
			285
	J. C. J. Benningshof, M. IJsselstijn, S. R. Wallner, R..H. Blaauw, A. E. Van Ginkel, F. P. J. T. Rutjes, H. Hiemstra (University of Arnsterdam, The Netherlands)
	Program No.: 31-OP-61 (A-16)

*31-PO-3*	Enantioselective Total Synthesis of Eudistomin C		286
	H. Tokuyama, T. Yamashita, N. Kawai, T. Fukuyama (The University of Tokyo, Japan)
	Program No.: 31-OP-65 (A-17)

*31-PO-4*	Stereoselective Total Synthesis of Zaragozic Acid A		287
	M. Kikuchi, K. Igawa, M. Suzuki, K. Ping-Huai, T. Nakai, K. Tomooka (Tokyo Institute of Technology, Japan)
	Program No.: 31-OP-69 (A-18)

*31-PO-5*	Asymmetric Total Synthesis of CDC25A Inhibitor Dysidiolide and Its Potent Analogs
			288
	R. Shirai, K. Dodo, K. Koga (Nara Institute of Science and Technology, Japan) M. Takahashi, Y. Hashimoto (The University of Tokyo, Japan)
	Program No.: 31-OP-73 (A-19)

*31-PO-6*	Synthetic Study of Ciguatoxin CTX3C		289
	T. Oishi, H. Uehara, M. Maruyama, H. Imai, Y. Nagumo, M. Shoji, K. Maeda, J.-Y. Le Brazidec, M. Kosaka, H. Oguri, M. Hirama (Tohoku University / CREST, Japan)
	Program No.: 31-OP-77 (A-20)

*31-PO-7*	Synthesis of Methylcoriandrin		290
	K. Datta, M. Bandyopadhyay, D. Mal (Indian Institute of Technology, Kharagpur, India)
	Program No.: 31-OP-81 (A-21)

*31-PO-8*	Asymmetric Synthesis of (R)-3-Methylpyrrolidine Alkaloids		291
	X. Zheng, Y. P. Ruan (Xiamen University, China) P. Q. Huang (Lanzhou University/ Xiamen University, China) A. W. M. Lee, W. H. Chan (Hong Kong Baptist University, China)
	Program No.: 31-OP-85 (A-22)

*31-PO-9*	Synthetic Studies on (-)-Ephedradine A		320
	W. Kurosawa, T. Kan, T. Fukuyama (The University of Tokyo, Japan)

*31-PO-10*	Synthetic Studies on FR901483		321
	T. Fujimoto, H. Kitaoka, S. Ieda, T. Kan, T. Fukuyama (The University of Tokyo, Japan)

*31-PO-11*	Synthesis of Polyamine Alkaloids by the Condensation of a Chiral SLactam with a Cyclic Imino Ether. Structure and Properties of Azalactams
			322
	H. Matsuyama, A. Matsumoto, N. Ohira, A. Kurosawa, T. Takei, M. Yoshida, M. Iyoda (Tokyo Metropolitan University, Japan)

*31-PO-12*	Novel Synthetic Strategy towards Polysubstituted Cyclohexane Derivatives: Synthetic Studies of (-)-Stenine
			323
	H. Fujioka, N. Kotoku, Y. Nagatomi, T. -I. Wang, T. Fujita, Y. Kita (Osaka University, Japan)

*31-PO-13*	Lipase-Catalyzed Enantioselective Desymmetrization of Prochiral 1,3-Diols: Study on Asymmetric Total Synthesis of Fredericamycin A and Its Analog
			324
	S. Akai, T. Tsujino, T. Naka, N. Fukuda, K. Kawaguchi, K. Higuchi, Y. Kita (Osaka University, Japan)

*31-PO-14*	Seven New Labdane-type Diterpenoids from the Wood of Cunninghamia konishii
			325
	Y.-H. Kuo, Y.-C. Li (National Taiwan University, Taiwan)

*31-PO-15*	Three New Adenine Analogues from the Leaves of Formosan Bridelia balansae
			326
	I.-L. Tsai, Y.-H. Tsai, I.-S. Chen (Kaohsiung Medical University, Taiwan) C.-Y. Duh (National Sun Yat-sen University, Taiwan)

*31-PO-16*	*Enantioselective Total Synthesis of Cyanobacterin Employing (5R)-5-(l-Menthyloxy)-2(5H)-furanone as the Chiral Synthon*
			327
	S. Park, T. Kusano, F. Ishibashi (Nagasaki University, Japan)

*31-PO-17*	Progress toward the Total Synthesis of Pinnatoxins, Aza-Spirocyclic Marine Natural Toxins
			328
	J. Ishihara, S. Tojo, A. Kamikawa, M. Horie, Y. Shimada, A. Murai (Hokkaido University, Japan)

*31-PO-18*	Studies on the Synthesis of Germacranolide Derivatives and Their Rearrangement to Guaianolides
			329
	Y. Higuchi, M. Ando (Niigata University, Japan)

*31-PO-19*	Production of Taxol®, Taxol Analogs, and Some Biologically Active Taxoids by Callus Cultures of Japanese Yew (Taxus cuspidata)
			330
	J. Bai, S. Zhang, J. Sakai, M. Kitabatake, K. Toyoizumi, H. Fujisawa, M. Ando (Niigata University, Japan)

*31-PO-20*	Synthesis of Biologically Active Taxinine NN-1 as Modulators of Multidrug Resistant Tumor Cells and Anticancer Reagent
			331
	S. Zhang, J. Sakai, H. Sasaki, M. Ando (Niigata University, Japan)

*31-PO-21*	Aza-pinacol Rearrangement: Acid-catalyzed Rearrangement of Aziridines to Imines
			332
	Y. Sugihara, S. Iimura, J. Nakayama (Saitama University, Japan)

*31-PO-22*	A Stereoselective Synthesis of Enamides: Synthetic Study on Oximidines		333
	K. Kuramochi, H. Watanabe, T. Kitahara (The University of Tokyo, Japan)

*31-PO-23*	Pyrralic Acids, a Novel Class of Pyrrole Masked Amino Acids from Actinomycetes
			334
	M. Brüning, N. Pöhlmann, A. Zeeck (University of Gotlingen, Germany)

*31-PO-24*	Studies on Total Synthesis of Wortmannin, A Potent Inhibitor of Phosphoinositide3-Kinase
			335
	T. Mizutani, S. Honzawa, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-25*	Enantioselective Total Synthesis of Epothilones and Their Analogues Using Multifunctional Asymmetric Catalysis
			336
	R. Namme, D. Sawada, M. Kanai, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-26*	Enantioselective Total Syntheses of (+)-Decursin and Its Derivatives Using Catalytic Asymmetric Epoxidation of Enones and Structural Determination of the Asymmetric Catalyst
			337
	T. Nemoto, T. Ohshima, M. Shibasaki (The University of Tokyo, Japan) K. Yamaguchi (Chiba University, Japan)

*31-PO-27*	A Formal Synthesis of 4-Demethoxydaunomycin Using Catalytic Asymmetric Ring Opening Reaction of meso-Epoxides with Anilines
			338
	A. Sekine, T. Ohshima, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-28*	Evaluation of Lipophilicity of Some New Thiazolyl-oxadiazolines by Principal Component Analysis
			319
	B. Tiperciuc, S. Todor, O. Oniga (University of Medicine and Pharmacy "Iuliu Hatieganu”, Romania) C. Sarbu (The University of Babes - Bolyai, Romania)
	Program No.: 31-OP-92 (D-23)

*31-PO-29*	Synthetic Study of Guanofosfocin-Preparation of 8-(Mannosyloxy)inosine Derivative
			339
	H. Sugimura, Y. Natsui (Yokohama National University, Japan)

*31-PO-30*	Synthetic Studies on Papuamides, Novel Cyclodepsipeptide with Anti-HIV and Cytotoxic Activities
			340
	N. Okamoto, K. Kobayashi, O. Hara, K. Makino, Y. Hamada (Chiba University, Japan)

*31-PO-31*	Total Synthesis of Spicamycin		341
	T. Suzuki, S. T. Suzuki, I. Yamada, Y. Koashi, K. Yamada, N. Chida (Keio University, Japan)

*31-PO-32*	New Findings in Reissert Indole Synthesis and Total Synthesis of Picrasidine V
			342
	H. Suzuki, H. Yamada, H. Gyoutoku, Y. Murakami (Toho University, Japan)

*31-PO-33*	Synthetic Studies on an Antitumor Cyclic Peptide, Ustiloxin A		343
	M. Nakada, H. Ichinose, A. Tada (Waseda University, Japan)

*31-PO-34*	Sesquiterpene Pyridine Alkaloids from Hippocratea excelsa		344
	T. Uchiyama, M. Furukawa, M. Makino, K. Ishimi, Y. Ichinohe, Y. Fujimoto (Nihon University, Japan)

*31-PO-35*	A Concise Construction of an Erythrinane Skeleton Using Mn(III/Cu(II)-Mediated Oxidative Radical Cyclization of α-Methylthio Amides
			345
	S. Chikaoka, A. Toyao, Y. Takeda, O. Tamura, H. Ishibashi (Kanazawa University, Japan) O. Muraoka, G. Tanabe (Kinki University, Japan)

*31-PO-36*	Synthetic Study on Ecteinascidin 743		346
	A. Endo, S. Tohma, T. Kan, T. Fukuyama (The University of Tokyo / CREST/ The Japan Science and Technology Corporation (JST), Japan)

*31-PO-37*	Synthetic Studies on (+)-Lysergic Acid		347
	T. Kurokawa, T. Fukuyama (The University of Tokyo / CREST / The Japan Science and Technology Corporation (JST), Japan)

*31-PO-38*	Total Synthesis of (+)-Gelsemine		348
	S. Vokoshima, H. Tokuyama, T. Fukuyama (The University of Tokyo/CREST, Japan)

*31-PO-39*	Synthetic Studies on FR-900482		349
	M. Kambe, E. Arai, M. Suzuki, H. Tokuyama, T. Fukuyama (The University of Tokyo, Japan)

*31-PO-40*	Efficient Cyclization of Ether Ring Using Sml₂		293
	F. Matsuda, H. Tamiya (Hokkaido University, Japan)
	Program No.: 31-OP-58 (B-15)

*31-PO-41*	Tetrahydropyrrolo[3,2-c]pyridines. Synthesis and Reactivity		294
	L. G. Voskressensky, A. V. Varlamov, T. N. Borisova (Russian Peoples Friendship University, Russia)
	Program No.: 31-OP-62 (B-16)

*31-PO-42*	Studies Directed toward the Total Synthesis of Mycalamides-Stereoselective Construction of the Right- and Leh-Half Segments
			295
	M. Toyota, M. Hirota, H. Hirano, N. Kagawa, M. Ihara (Tohoku University, Japan)
	Program No.: 31-OP-66 (B-17)

*31-PO-43*	Regioselective BH₃-hydride Reduction of Inosine Derivatives		296
	K. Hirota, R. Hattori, H. Sajiki, Y. Monguchi (Gifu Pharmaceutical University, Japan) O. Muraoka, G. Tanabe (Kinki University, Japan)
	Program No.: 31-OP-70 (B-18)

*31-PO-44*	Lithio-1,2,4-triazines-Synthesis, Structure, Synthetic Potential		297
	H. Neunhoeffer, T. Hundsdorf (Darmstadt University of Technology, Germany)
	Program No.: 31-OP-74 (B-19)

*31-PO-45*	Novel Carbon-Carbon Bond Formation Reaction of Methoxyallene Oxide Promotedby Til₄
			298
	M. Shimizu, R. Hayakawa, I. Hachiya (Mie University, Japan)
	Program No.: 31-OP-78 (B-20)

*31-PO-46*	Enantioselective Coniugate Additions of Thiols and b-Keto Esters Catalyzed by Chiral N-Oxide-Metal Complexes
			299
	M. Nakajima, M. Saito, Y. Yamaguchi, S. Hashimoto (Hokkaido University, Japan)
	Program No.: 31-OP-82 (B-21)

*31-PO-47*	Solid/Liquid Phase Synthesis of b-Strand Mimetic Templates via Regioselective 1,3-Dipolar Cycloaddition
			300
	N. Fuchi, T. Doi, T. Takahashi (Tokyo Institute of Technology, Japan) M. Kahn (University of Washington, USA)
	Program No.: 31-OP-86 (B-22)

*31-PO-48*	*Lewis Acid-Catalyzed Ring-Opening Reactions of Semicyclic N,O-Acetals: Application to Piperidine Alkaloid Syntheses*
			350
	M. Sugiura, S. Kobayashi (The University of Tokyo, Japan)

*31-PO-49*	Nickel and Palladium Catalyzed Synthesis of Heterocycles		351
	Y. Tamaru, M. Kimura, S. Tanaka (Nagasaki University, Japan)

*31-PO-50*	Regioisomeric Formation of 1,2,4-Triazolo[4',3':2,3][1,2,4]triazino-[5,6-b]indole of Its Angular Isomer from 3-Hydrazino-1,2,4-triazino[5,6-b]indole Derivatives
			352
	E. S. H. El Ashry, H. Abdel Hamid, A El Nemr, A Mousaad, E. S. Ramadan (Alexandria University, Egypt) Y. A Al-Soud (Al-Albeit University, Jordan)

*31-PO-51*	Cyanothiocetamide in Heterocyclic Synthesis: Synthesis of Pyridinethione, 2‑S-Alkylpyridine, Thieno[2,3-b]pyridine, Pyrazolo[4,3-c]pyridine and Thiopyrano[2,3-b]pyridine Derivatives
			292
	F. A. Attaby, Y. M. Ibrahim (Cairo University, Egypt)
	Program No.: 31-OP-89 (A-23)

*31-PO-52*	Design and Synthesis of New Structures Related to Indole Alkaloids and otherNatural Products
			353
	D. S. Black, M. F. Channon, G. C. Condie, P. S. R. Mitchell, R. Rezaie (The Universiry of New South Wales, Australia)

*31-PO-53*	An Efficient Method for the Syntheses of 2-Substituted-2-oxazolines and 2H‑2-oxazolines: Condensation of Ortho Esters with Amino Alcohols under Environment Friendly Conditions
			354
	R. S. Gulhane, A. K. Chakraborti (National Institute of Pharmaceutical Education and Research (NIPER), India)

*31-PO-54*	Novel Synthesis of 3-Alkyl-2,5-diaryl-1,4-oxathiepin-7-ones		355
	B. S. Kim, K. Kim (Seoul National University, Korea)

*31-PO-55*	Synthesis and Toxicity to PC12 Cells of 1-Alkyl-1,2,3,4-tetrahydroisoquinolines
			356
	T, Saitoh, M. Ishikawa, Y. Horiguchi, T. Sano (Showa Phamiaceutical University, Japan) M. Nakatani, S. Shimazu, N. Sato, F. Yoneda (Fujimoto Pharmaceulical Co., Japan)

*31-PO-56*	Synthesis and Electroluminescent Applications of Ortho-fused Heterocyclic Compounds
			357
	N. Tsujiuchi, H. Osuga, M. Hisamoto, K. Tanaka (Wakayama University, Japan)

*31-PO-57*	Cycloaddition Reaction of Styrene Derivatives Using Iron Salt Catalyst: Fe(BF₄)₂ Mediated Reaction in the Ionic Liquid Solvent System
			358
	H. Ohara, H. Kiyokane, T. Itoh (Okayama University, Japan)

*31-PO-58*	The First Catalytic Asymmetric Nitro-Mannich Reaction		359
	K. Yamada, H. Gröger, S. J. Harwood, G. Moll, N. Tsuritani, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-59*	Catalytic Asymmetric Aldol Reaction of Ketones and Aldehydes Using Chiral Calcium Alkoxides
			360
	M. Shibasaki (The University of Tokyo, Japan) T. Suzuki, N. Yamagiwa (The University of Tokyo / Nagoya University, Japan) Y. Matsuo, R. Noyori (Nagoya University, Japan) S. Sakamoto, K. Yamaguchi (Chiba University, Japan)

*31-PO-60*	Direct Catalytic Asymmetric Aldol Reactions Promoted by Heterobimetallic Catalysts
			361
	N. Yoshikawa, N. Kumagai, S. Matsunaga, T. Ohshima, T. Suzuki, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-61*	Immobilization of Asymmetric Multifunctional Catalysts on an Insoluble Polymer
			362
	S. Matsunaga, R. G. Franzén, T. Ohshima, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-62*	Highly Regioselective Synthesis of Cyclic Enol Silyl Ethers Using Ring-Closing Metathesis
			363
	A. Okada, T. Ohshima, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-63*	*Direct Catalytic Asymmetric Aldol Reaction: Synthesis of Syn-1,2-diols Using Zn-Zn-Linked BINOL Complex*
			364
	N. Kumagai, N. Yoshikawa, S. Matsunaga, T. Ohshima, T. Suzuki, M. Shibasaki (The University of Tokyo, Japan)

*31-PO-64*	Beckmann Rearrangement vs. Carbonyl Compound Regeneration from Cyclohexanone Oxime		365
	G. C. Penieres, A. T. Cecilio, N. C. Olivia, G. E. José Guadalupe, C. S. José Luis, A. M. Rubén (Universidad Nacional Autónoma, México)

*31-PO-65*	The Tandem Michael/Aldol: Reaction as a Tool of Syntheses of Heterocycles		366
	A. Kamimura, K. Matsuura, Y. Omata, H. Mitsudera (Yamaguchi University, Japan)

*31-PO-66*	Enantioselectivity in Chiral Lewis Acid-catalyzed Cycloadditions of Carbonyl Ylides
			367
	H. Suga, K. Inoue, A. Kakehi, S. Ito (Shinshu University, Japan) T. Ibata (Osaka University, Japan)

*31-PO-67*	Synthesis of Donor-Acceptor Substituted 2,2'-Bithiophenes and Reactivity Studies
			368
	M. M. Marques Raposo (Universidade do Minho, Portugal) G. Kirsch (Université de Metz, France)

*31-PO-68*	Stereoselective b-Glycosylation of 2,3-Dideoxyribofuranose Derivatives Controlled by Phosphonothioate Functionality
			369
	T. Yokomatsu, T. Murano, T. Sada, S. Shibuya (Tokyo University of Pharmacy & Lire Science, Japan)

*31-PO-69*	Dynamic Kinetic Resolution of Carbonates of the Serinol; Asymmetric Synthesis of the 4-Hydroxymethyl-2-oxazolidinone
			370
	S. Sugiyama, S. Watanabe, T. Inoue, K. Ishii (Mevi Pharmaceutical University, Japan)

*31-PO-70*	Faceselective Addition to Cation-π Complexes of Pyridinium Salts: Stereoselective Synthesis of 1,2- and 1,4-Dihydropyridines
			371
	M. Saitoh, T. Misono, S. Yamada (Ochanomizu University, Japan)

*31-PO-71*	Stereoselective Synthesis of Medium-Sized Cyclic Compounds by Tandem Reactions of Cyclic Oxosulfonium Vlides with b-Acetoxy-α-Methylene Ketone Derivatives

			372
	H. Akiyama, A. Nabeshima, T. Fujimoto, K. Ohshima, I. Yamamoto, Kakehi, R. Iriye (Shinshu University, Japan)

*31-PO-72*	Novel Palladium-catalyzed Oxazolidone Synthesis		373
	S. Tanimori, U. Inaba, M. Kirihata (Osaka Prerecture University, Japan)

*31-PO-73*	Stereoselective Photocyclization of Enamide Derivatives in Polymer Matrix		374
	T. Tsuno, Y. Uchida, K. Sugiyama (Nihon University, Japan)

*31-PO-74*	Lactam Synthesis Based on Amine Trap of Acyl Radicals		375
	T. Fukuyama, M. Tojino, Y. Uenoyama, I. Ryu (Osaka Prerecture University, Japan)

*31-PO-75*	*Total Syntheses of (±)-7-Oxokaurenolide and (±)-Methyl Gummiferolate via* Radical Cyclization**
			376
	M. Toyota, M. Yokota, M. Ihara (Tohoku University, Japan)

*31-PO-76*	Regioselective Alkylation of 2,4-Diaminopyrimidine Systems		377
	K. Kazaoka, H. Sajiki, M. Sako, K. Hirota (Giru Pharmaceutical University, Japan)

*31-PO-77*	Enantioselective Diels-Alder Reaction Catalyzed by Bispyrazolylalkanes		378
	C. Kashima, Y. Miwa. S. Shibata, Y. Yokoyama (University of Tsukuba, Japan)

*31-PO-78*	Regio -and Stereoselective Cyclization of Epoxy Alcohols Using Magnesium Halides
			379
	M. Karikomi, Y. Kimura. S. Watanabe, T. Uyehara (Utsunomiya University, Japan)

*31-PO-79*	Solid State and Solution Structure of Some Novel Pentavalent Organogermanium Compounds
			380
	Y. Takeuchi, M. Nishikawa, K. Tanaka (Kanagawa University, Japan) A. Kalman. L. Parkanyi (Hungarian Academy of Sciences, Hungary) G. Yamamoto (Kitasato University, Japan)

*31-PO-80*	Study of Asymmetric Tandem Michael-HWE Reactions		381
	D. Monguchi, K.Tanaka (University of Shizuoka, Japan)

*31-PO-81*	Synthesis of Polysubstituted Furans by Iridium-Catalyzed Intermolecular Couplings
			382
	T. Makino, I. Matsuda, K. Itoh (Nagoya University, Japan)

*31-PO-82*	Chiral Amidomonophosphine-Rhodium(I) Catalyst for Asymmetric 1,4-Addition of Arylboronic Acids to Cycloalkenones
			383
	M. Kuriyama, K. Tomioka (Kyoto University, Japan)

*31-PO-83*	Copper-Catalyzed Asymmetric Alkylation of Imines with Diethylzinc.		384
	K. Nagai, H. Fujihara. K. Tomioka (Kyoto University, Japan)

*31-PO-84*	Synthesis and Reaction of 1-Azaazulene N-ylide		385
	H. Fujii, K. Iwafuji. N. Abe (Yamaguchi University, Japan) Kakehi (Shinshu University, Japan)

*31-PO-85*	Rearrangement Reaction of Fused 3-(2-Bromoethyl)pyrimidine Derivatives with Amines
			386
	K. Sasaki, T. Tagata. F. Tanaka, K. Okuda. T. Hirota (Okayama University, Japan)

*31-PO-86*	A Simple Synthetic Method for Fluorine-Containing Heterocycles Having Quinoline Skeleton
			387
	E. Okada, T. Ashida.T. Sakaemura, T. Mori (Kobe University, Japan)

*31-PO-87*	*Synthesis of 3-Fluorinated* Quinoline Derivatives via Intramolecular Substitution of o-Substituted b,b-Difluorostyrenes**
			388
	J. Ichikawa, Y. Wada. T. Mori (The University of Tokyo, Japan)

*31-PO-88*	*Development of a General Methodology towards Synthesis of Amaryllidaceae* Alkaloids: Application to the Total Synthesis of (-)Brunsvigine**
			389
	C.-K. Sha, A.-W. Hong, C.-M. Huang, T.-H. Jeng (National Tsing Hua University, Taiwan)

*31-PO-89*	*Synthesis of 3-Benzazepine Derivatives via* The Ring-Expansion Reaction of Isoquinolines**
			390
	H. Sato, H. Ozawa, Y. Koseki, T. Nagasaka (Tokyo University of Pharrnacy and Life Science, Japan)

*31-PO-90*	A Stereocontrolled Construction of b-Glycosidic Linkages Using Mannopyranosyl and 2-Azido-2-deoxyglucopyranosyl Donors Carrying Phosphorus-Containing Leaving Groups
			391
	T. Tsuda, S. Sato, S. Nakamura, S. Hashimoto (Hokkaido University, Japan)

*31-PO-91*	Enantiocontrol in Tandem Allylic Onium Vlide Generation and Rearrangement Catalyzed by Chiral Dirhodium(II) Complexes
			392
	S. Kitagaki, H. Tsutsui, Y. Yanamoto, H. Okubo, S. Hashimoto (Hokkaido University, Japan)

*31-PO-92*	Synthesis and Biological Evaluation of 4,5-Dihydronaphtho [1,2-d]1,2,3-thia- or selenadiazole Derivatives
			302
	M. Daneshtalab (Memorial University of Newroundland, Canada) A. R. Jalilian, M. Binesh-Marvasti, A. Shafiee (Tehran University of Medical Sciences, Iran) S. Sattari (University of Alberta, Canada)
	Program No.: 31-OP-59 (C-15)

*31-PO-93*	Fluorescent Rhodacyanine Dyes as Antimalarial Agents: Library Construction and Structure-Activity Relationship
			303
	K. Takasu, H. Inoue, M. Ihara (Tohoku University, Japan) H.-S. Kim, Y. Wataya (Okayama University, Japan)
	Program No.: 31-OP-63 (C-16)

*31-PO-94*	Discovery of Novel Aspartyl Ketones as Potent Caspase-3 Inhibitors		304
	Y. Han, A. Giroux, E. L. Grimm, R. Aspiotis, C. I. Bayly, D. J. Mckay, S. J. Roy, S. Xanthodakis, J. Valancourt, D. M. Rasper, J. Tam, P. Tawa, D. W. Nicholson, R. J. Zamboni (Merck Frosst Canada & Co., Canada) N. A. Thornberry, E. P. Paterson, M. Garcia-Calvo, J. W. Becker, J. Rotonda (Merck Research Laboratories, Merck & Co., Inc., USA)
	Program No.: 31-OP-67 (C-17)

*31-PO-95*	Novel Synthesis of Substituted Indoles from 2-Aminophenols		305
	W.-M. Dai, D.-S. Guo, L.-P. Sun (The Hong Kong University of Science and Technology, China)
	Program No.: 31-OP-71 (C-18)

*31-PO-96*	Heterocyclic-fused Naphthalimides: Synthesis Via Unusual Pschorr Cyclization, Spectral Properties and Interesting Photocleaving Action to DNA
			306
	X. Qian, J. Cui, R. Zhang (Dalian University of Technology, China) W. Yao, P. Mao (East China University of Science and Technology, China)
	Program No.: 31-OP-75 (C-19)

*31-PO-97*	Practical Synthesis of an Indolocarbazole-based DNA, Topoisomerase I Inhibitor
			307
	A. Kamatani, M. Kawasaki, N. Satake, S, Hiraga, A. Akao, T. Nemoto, T. Iida, T. Mase (Banyu Pharmaceutical Co., Lid., Japan) S. A. Weissman, D. M. Tschaen, R. P. Volante (Merck Research Laboratories, USA)
	Program No.: 31-OP-79 (C-20)

*31-PO-98*	Annelated Pyrrolo-Pyrimidines New Tricyclic DNA-Interactive Ring Systems
			308
	A. M. Almerico (University of Palermo, Italy) A. Lauria, P. Diana, P. Barraja, A. Montalbano, G. Cirrincione, G. Dattolo (Università degli Studi, Italy)
	Program No.: 31-OP-83 (C-21)

*31-PO-99*	Alkyl α-Substituted b-(Dimethylamino)-α, b-didehydro Acid Derivatives and Their Chiral Analogs--Versatile Reagents in the Synthesis of Heterocyclic Systems
			309
	B. Stanovnik, J. Svete, U. Bratušek, U. Grošelj. R. Jakše, L. Jukić Soršak, S. Pirc, S. Rečnik, C. Turk (University of Ljubljana, Slovenia)
	Program No.: 31-OP-87 (C-22)

*31-PO-100*	Synthesis of 2',5'-isoDNA Mimic Chiral Peptide Nucleic Acids		393
	M. A.-A. Osman, T. Yamasaki, M. Otsuka (Kumamoto University, Japan)

*31-PO-101*	Potent Estrogen Agonists and Antagonists Sased on Carborane as a Hydrophobic Skeletal Structure
			394
	T. Yoshimi, T. Iijima, Y. Yamakoshi, H. Fukasawa, Y. Endo (The University of Tokyo, Japan)

*31-PO-102*	Novel 2-(N-Cyanoimino) thiazolidin-4-one Derivatives: Synthesis and Hypolipidemic Activities in Rodents
			395
	M. Watanabe, T. Ando, T. Yasusa, K. Urabe, S. Muraoka, F. Yoneda (Fujimoto Pharmaceutical Corp., Japan)

*31-PO-103*	The Reaction of Aldolic Condensation-Means to Obtain α-Dicarbonyls		310
	V. Zaharia, S. Imre(University of Medicine and Pharmacy "Iuliu Hatieganu", Romania) P. Verite (University of Medicine and Pharmacy, France)
	Program No.: 31-OP-91 (C-23)

*31-PO-104*	Retinoid Synergistic Dibenzodiazepine and Pryrimidine Derivatives		396
	B. Takahashi, M. Ebisawa, K. Ohta, E. Kawachi, H. Fukasawa, Y. Hashimoto, H. Kagechika (The University of Tokyo, Japan)

*31-PO-105*	Use of Phenyl 2-Selenoketosides of N-Acetylneuraminic Acid as a Glycosyl Donor for the Glycosylation Reactions
			397
	K. Ikeda, M. Sato, K. Tanaka (University of Shizuoka, Japan)

*31-PO-106*	Synthesis and Evaluation 3,4-Epoxypiperidine Derivatives as a Novel Alkylating Agent
			398
	K. Miyashita, S. Adachi, M. Park, T. Imanishi (Osaka University, Japan)

*31-PO-107*	Synthesis and Evaluation of Antibacterial Fluoroquinolones		399
	C:-C. Tzeng, Y.-L –Chen, K.-C. Fang, J.-Y. Sheu, S.-L. Hsu (Kaohsiung Medical University, Taiwan)

*31-PO-108*	New Cytotoxic Butanolides from Litsea acutivena		400
	I.-S. Chen, H.-I. Cheng, I.-L. Tsai (Kaohsiung Medical University, Taiwan) C.-Y. Duh (National Sun Yat-sen University, Taiwan) K.-H. Lee.. (University of North Carolina, USA)

*31-PO-109*	Structural Features of Aliphatic N-Nitrosamines of 7‑Azabicyclo[2.2.1]heptanes That Facilitate N-NO Bond Cleavage
			401
	T. Ohwada (The University of Tokyo, Japan)

*31-PO-110*	Production of Novel Bioactive Dehydro Cyclic Dipeptides by Microbial Enzyme System
			402
	H. Kanzaki, S. Yanagisawa, K. Akazawa, T. Nitoda (Okayama University, Japan)

*31-PO-111*	Microbial Metabolism of a Bioactive Diketopiperazine		403
	K. Miyoshi, N. Mizuta, T. Nitoda, H. Kanzaki (Okayama University, Japan)

*31-PO-112*	*Synthesis and In Vitro* Anti-Measles and Anti-Rhino Viral Activities of Several "Fat" Nucleosides Containing the Imidazo[4,5-e][1,3]diazepine Ring System**
			404
	N. Zhang, H. -M. Chen, R. S. Hosmane (University of Maryland, USA) R. Sood (Nabi, USA)

*31-PO-113*	*Synthesis and Potent In Vitro* Anti-Epstein-Barr Virus (Anti-EBV) Activity of a 3'-Deoxy "Fat" Nucleoside Containing the Imidazo[4,5-e][1,3]diazepine Ring System**
			405
	R. Sood, V. S. Bhadti (Nabi, USA) R. S. Hosmane (University of Maryland, USA)

*31-PO-114*	Theoretical Approach to Stereospecific Heterocyclization of Carbohydrate Derivatives
			406
	A. Robinsohn, G. Rodrigo, M. Hedrera, B. Fernández (Universidad de Buenos Aires, Argentina) M. M. Alho, N. D’Accorso (FCEN, Universidad de Buenos Aires, Argentina)

*31-PO-115*	Systemic Activity of Oxazolones Derived from Ketones		407
	R. K. Sandhar, R. C. Sharma, M. R. Manrao (Punjab Agricultural University, India)

*31-PO-116*	Nucleophilic Reactions in Indole Series: Displacement of Bromine under Phase Transfer Catalysis
			408
	G. Cirrincione (University of Palermo, Italy) P. Barraja, P. Diana, A. Lauria, A. Montalbano, A. M. Almerico, G. Dattolo (Università degli Study, Italy)

*31-PO-117*	"Interrupted" Diazotization of 3-Aminoindoles and 3-Aminopyrroles		409
	G. Cirrincione (University of Palermo, Italy) P. Barraja, P. Diana, A. Lauria, A. Montalbano, A. M. Almerico, G. Dattolo (Università degli Study, Italy)

*31-PO-118*	Exploitation of Benzimidazoles as Nematicides		410
	M. Rai, G. Kaur, V. K. Kaul(Punjab Agricultural University, India)

*31-PO-119*	Bioactive Heterocycles: Synthesis and Fungitoxicity of Mercapto Substituted 4-Thiazolidinones
			411
	M. Jolly, B. Surendranath, J. R. Sharma, M. R. Manrao (Punjab Agricultural University, India)

*31-PO-120*	Studies on the Self-Organization Phenomena Involving Pyridone and Phenol Derivatives
			311
	I. Takahashi, M. Wagi, M. Takahashi, H. Kitajima, M. Hatanaka, K. Isa (Fukui University, Japan) S. Hosoi, T. Ohta (Kanazawa University, Japan)
	Program No.: 31-OP-60 (D-15)

*31-PO-121*	Synthesis of Chiral Diarylacetylene-Dicobalt Hexacarbonyls		312
	T. Sugihara, C. Harumori, H. Takao, H. Imagawa, M. Nishizawa (Tokushima Bunri University, Japan)
	Program No.: 31-OP-64 (D-16)

*31-PO-122*	Tributylmagnesium Ate Complex Mediated Novel Bromine-Magnesium Exchange Reaction: Industrial Synthesis of a Muscarinic M₃ Receptor Antagonist
			313
	T. Iida, T. Wada, K. Tomimoto, T. Mase (Banyu Pharmaceutical Co., Lid., Japan)
	Program No.: 31-OP-68 (D-17)

*31-PO-123*	Introduction of Podand Histidyl Moieties into a Pyridine Scaffold to Induce a Chiral Helicity
			314
	T. Moriuchi, M. Nishiyama, K. Yoshida, T. Ishikawa, T. Hirao (Osaka University, Japan)
	Program No.: 31-OP-72 (D-18)

*31-PO-124*	New Polycyclic Aza-heterocycles, Precursors for Persistent Free Polyradicals		315
	I. A. Silberg, C. Cristea, D. Porumb (Babes-Bolyai University, Romania) M. D.Banciu (Polytechnic University, Romania) M. Danila (“C.D. Nenitzescu" Center of Organic Chemistry, Romania)
	Program No.: 31-OP-76 (D-19)

*31-PO-125*	Tetrakis(2-thienyl)methane: First Synthesis and Synthetic Utility		316
	M. Oda, H. Nakaminami, M. Sogabe, K. Matsumoto, H. Kurata (Osaka University, Japan)
	Program No.: 31-OP-80 (D-20)

*31-PO-126*	Greening of Cephalosporin Chemistry		317
	B. Zwanenburg, G. Kemperman, J. Zhu (University of Nijmegen, The Netherlands)
	Program No.: 31-OP-84 (D-21)

*31-PO-127*	New Synthetic Pathways to Indole and Benzimidazole Derizatives		318
	Y. Torisawa, H. Yukawa, T. Nishi, J. Minamikawa (Otsuka Pharmaceutical Co. Lid., Japan)
	Program No.: 31-OP-88 (D-22)

*31-PO-128*	Electronic Effects of Icosahedral Carboranes on Solvolysis		412
	Y. Taoda, T. Sawabe, Y. Endo (The University of Tokyo, Japan)

*31-PO-129*	Synthesis of 2-Pyridylpyridines via Diels-Alder Reactions between 3-Pyridyl-1,2,4-triazines and Some Dienophiles
			413
	F. Ikeuchi, T. Shinto, H. Suda. Y. Furugori, I. Itoh (Sankio Chemical Co., Lid., Japan)

*31-PO-130*	Development and Biological Applications of Novel Zinc Fluorescent Probes: ZnAFs
			414
	T. Hirano, K. Kikuchi, T. Nagano (The University of Tokyo, Japan) N. Matsumoto, Y. Kudo (Tokyo University of Pharmacy and Life Science, Japan)

*31-PO-131*	Selective Sensing of Zinc Ion with TPEN Moiety on a Magnetic Resonance lmaging Contrast Agent
			415
	K. Hanaoka, K. Kikuchi, T. Nagano (The University of Tokyo, Japan)

*31-PO-132*	Inositol 1,4,5-Trisphosphate Analogues Modified at 1-Phosphate		416
	W. Nakanishi, K. Kikuchi, K. Hirose, M. Iino, T. Nagano (The University of Tokyo, Japan)

*31-PO-133*	Design and Synthesis of a Enzyme Cleavable Sensor Molecule for Phosphodiesterase Activity Based on Fluorescence Resonance Energy Transfer
			417
	H. Takakusa, K. Kikuchi, T. Nagano (The University of Tokyo, Japan)

*31-PO-134*	A Fluorescent Sensor for Anions in Neutral Aqueous Solution		418
	S. Mizukami, K.Kikuchi, T. Nagano (The University of Tokyo, Japan) A. Odani (Nagoya University, Japan)

*31-PO-135*	Development of Novel Fluorescence Probes for Hydroxyl Radical		419
	K. Setsukinai, Y. Urano, T. Nagano (The University of Tokyo, Japan)

*31-PO-136*	Multiple Active Intermediate in Cytochrome P450: Reaction Mechanism Analysis by Synthetic Heme-Thiolate
			420
	N. Suzuki, T. Nagano (The University of Tokyo, Japan) T. Higuchi (Nagoya City University, Japan)

*31-PO-137*	Fluorescence Off/On Switching Mechanism of Fluorescein-Based Fluorescence Probes
			421
	T. Miura, K. Tanaka. Y. Urano, T. Nagano (The University of Tokyo, Japan)

*31-PO-138*	Small Molecule-based Laser Inactivation of Inositol 1,4,5-Trisphosphate Receptor
			422
	T. Inoue, K. Kikuchi, T. Nagano (The University of Tokyo, Japan) K. Hirose. M. Iino (The University of Tokyo / CREST / Japan Science and Technology Corporation (JST), Japan)

*31-PO-139*	Nanoscale Supramolecular Architecture by Self-Assembly of Multinuclear Zinc(II) Complexes in Aqueous Solution
			423
	S. Aoki, E. Kimura (Hiroshima University, Japan) M. Shiro (Rigaku Corporation X-Ray Research Laboratory, Japan)

*31-PO-140*	*Enhanced Chemiluminescence of Cypridina* Luciferin Analogue, 6-(p-Methoxyphenyl)imidazo[1,2-α]pyrazin-3(7H)-one**
			424
	K. Teranishi, S. Tanabe (Mie University, Japan)

31-PO-141	High-Pressure-Promoted Uncatalyzed Condensation of Phenylisothiocyanates with Amiopyridine Derivatives
			425
	H. Kotsuki, K., Kumamoto (Koehi University, Japan) Y. Kubo, Y. Misawa (Saitama University, Japan)

*31-PO-142*	Synthesis and Photochromism of Fluorescent Diarylethenes Having a 2,4,5-Triphenylimidazole Chromophore
			426
	K. Yagi, M. Irie (Kyushu University / CREST / Japan Science and Teehnology Corporation (JST), Japan)

*31-PO-143*	Preparation, Fluorescence, and Liquid Crystalline Properties of 4,7-Diaryl-1,2,5-benzothiadiazole
			427
	H. Gorohmaru, N. Matsumoto, T. Thiemann, S. Mataka (Kyushu University/ CREST/ Japan Science and Teehnology Corporation (JST), Japan)

*31-PO-144*	*Formation and Characterization of Dihydrocyclopent[2,1-c]azete Derivative on Irradiation of 2,5-di-tert-Butyl-3H-azepine*
			428
	K. Satake, Y. Tawada (Okayama University, Japan) S. Yakami, M. Kimura (Kyushu University, Japan)

*31-PO-145*	Dipolar Cycloaddition of Mesoionic Compounds with Buckminsterfullerene: Intriguing Thermal and Photochemical Reactions of the Adducts
			429
	Y. Kawamura, K. Akaishi, S. Sato, M. Nishiuchi, M. Tsukayama (The University of Tokushima, Japan)

*31-PO-146*	*Fulvalene Formation via* a Reaction of Nucleophilic Carbenes with Buckminsterfullerene of Electron Acceptors**
			430
	Y. Kawamura, K. Takeda, M. Nishiuchi, M. Tsukayama (The University of Tokushima, Japan)

*31-PO-147*	Chemistry of 1,6-Disila[4.4.4]propellane and Related Compounds		301
	A. Toshimitsu, M. Katkevics, A. Sano, M. Asahara, T. Miki, H. Fujimura, H. Tsuji, S. Yamaguchi, K. Tamao (Kyoto University, Japan)
	Program No.: 31-OP-90 (B-23)

*31-PO-148*	New Scaffolds Containing the Quinoline-6-sulphonamide Moiety for Combinatorial Synthesis
			431
	A. Ivachtchenko, V. Kobak (Chemical Diversity Labs, Inc., USA)

*31-PO-149*	Asymmetric Total Synthesis of (+)-Brefeldin A from (S)-Lactate by Triple Chirality Transfer Process and Nitrile Oxide Cycloadditions
			432
	D. Kim, J. Lee, P. J. Shim, J. I. Lim, S. Kim (Seoul National University, Korea) T. Doi (Tokyo Institute of Technology, Japan)

*31-PO-150*	Synthesis of 3-Oxo-2,3-dihydro prazolo[3,4-b]quinolines		433
	S. P. Rajendran, K. M. Rani (Bharathiar University, India)

*31-PO-151*	Isocyanatophosphoric Acid Dichlorides in Synthesis of Carboxyimidophosphates and Heterocyclic Nitriles
			434
	A. Chaykovskaya, R. Smaliy, A. Tolmachev (National Aeademy of Sciences of Ukraine, Ukraine)

*31-PO-152*	The New Approach to the Synthesis of Polymethylene Derivatives of 1,3-Diazaheterocycles
			435
	K. Nazarenko, T. Shyroka, K. Shvidenko, A. Tolmachev (National Academy of Sciences of Ukraine, Ukraine)

*31-PO-153*	Reactions of 1,3-Benzothiazines and 1,4-Benzothiazepines with Dimethyl Acetylenedicarboxylate
			436
	L. Fodor (University of Szeged/ Central Laboratory Country Hospital, Hungary) G. Bernath (University of Szeged, Hungary) P. SoMr (Eötvös Loránd University) A. Kámán, G. Argay (Hungarian Academy of Sciences, Hungary)

*31-PO-154*	Synthesis, NMR, MS and X-ray Investigation of Homoadanantane-fused Pyridopyrimidines and Related Saturated Heterocycles
			437
	G. Bernáth, P. Csomós, Z. Gyarmati (University of Szeged, Hungary) G. Argay, A. Kálmán (Hungarian Academy of Sciences, Hungary) K. Pihlaja (University of Turku, Finland)

*31-PO-155*	Total Synthesis of (-)-Tubifoline by Palladium-Catalyzed Asymmetric Allylic Substitution
			438
	M. Nakanishi, D. Kajishima, Y. Sato, M. Mori (Hokkaido University, Japan)

*31-PO-156*	Preparation and Tautomerism of 3-Methyl-1-p-substituted phenyl pyrazolin-5-thiol
			439
	Y. Tagawa, Y. Goto (Fukuoka University, Japan) T. Yoshida, M. Yasuda, M. Nakashima (RRF Research Inc., Japan)

*31-PO-157*	The Synthesis of New Optically Active C₃-Symmetric Trisamides		440
	R. D. Ionescu, T. Frejd (Lund University, Sweden)

*31-PO-158*	Modulatory Activity of Protein Kinase C by Xanthone Derivatives		441
	L. Saraiva, E. Scusa, E. Pinto, P. Fresco, M. Pinto, J. Gonçalves (University of Porto, Portugal)

*31-PO-159*	Synthesis and Bioactivity of Novel Difused Helerocyclic Compounds		442
	G. Yang (Central China Normal University, China)

*31-PO-160*	Synthesis and Study of 4-Alkoxy-3-alkoxycabonyl-1(2H) isoquinolones and Related 1,6- and 1,7-Naphthyridines
			443
	M. M. Bianco, G. Levin, C. B. Schapira, I. A. Perillo (Universidad de Buenos Aires, Argentina)

*31-PO-161*	Synthesis of Dioxa-Cage Compounds as a New Probe for the Stereochemistry of the Bisadducts of p-Benzoquinone with 1,3-Cyclodienes
			444
	H.-J. Wu, C.-B. Tsao, T.-Y. Tsai (Chiao Tung University, Taiwan)

*31-PO-162*	Diels-Alder Reactions of 6-Hydroxy-2H-pyran-3(6H)-ones with Cyclopentadiene and Its Application for the Synthesis of New Skeletal Oxa-Cage Compounds
			445
	H.-J. Wu, H.-C. Lin, L. Cheng (Chiao Tung University, Taiwan)

August 2 (Thu)			Oral Presentation
14:30 - 16:00		SECTION A (Room 301)
Chair: H. Sasai (Osaka University, Japan)
*A-24*	New Concept for Blue Flower Color Development by Metal Complex			446
	K. Yoshida, M. Mori, K. Oyama, T. Kondo (Nagoga University, Japan). Y. Toyama (Sugigama Jogakuen University, Japan)
	Program No.: 2-OP-89 Poster No.: 2-PO-1

*A-25*	Inhibition and Structural Studies of the Enzyme Porphobilinogen Synthase			447
	F. Stauffer, E. Zizzari, C. Jarret, R. Neier (University of Neuchâtel, Switzerland)
	Program No.: 2-OP-93 Poster No.: 2-PO-2

*A-26*	Chemoselective Palladium Catalyzed Reaction in Aqueous Media: Selectivity in the Reaction of Bromoaniline with Allylalcohol
				448
	Y. Yokoyama, H. Hikawa, Y. Murakami (Toho University, Japan)
	Program No.: 2-OP-97 Poster No.: 2-PO-3

*A-27*	Axial Chirality due to an Acyclic Imide-Ar Bond: a Study of Steric and Electronic Effects of Acyl Groups on Racemization
				449
	K. Kondo, T. Iida, H. Fujita, T. Suzuki, Y. Murakami (Toho University, Japan) K. Yamaguchi (Chiba University, Japan)
	Program No.: 2-OP-101 Poster No.: 2-PO-4

*A-28*	Use of Bis(acylketene) in Heterocycle Synthesis			450
	M. Sato, K. Kondo, T. Katsumata, K. Iwamoto (University of Shizuoka, Japan)
	Program No.: 2-OP-105 Poster No.: 2-PO-5

*A-29*	Generation and Reaction of Metal-Containing Carbonyl Ylides: Tandem [3+2]-Cycloaddition-Carbene Insertion Leading to Novel Polycyclic Compounds
				451
	N. Iwasawa, M. Shido, H. Kusama (Tokgo Institute of Technology, Japan)
	Program No.: 2-OP-109 Poster No.: 2-PO-6

*A-30*	Chiral Aziridine-2-carboxylates: Preparation and Utilization for the Synthesis of Phenylalanine and Homophenylalanine
				452
	H.-J. Ha (Hankuk University of Foreign Studies/ ChembioNex Co., Ltd, HUFS BI, Korea), H.-J. Yoo, C. S. Park (Sogang University, Korea) W. K. Lee (Sogang University/ Chembio Nex Co., Lld, HUFS B/, Korea) Y. H. Lim (Chembio Nex Co., Ltd, HUFS BI, Korea)
	Program No.: 2-OP-113 Poster No.: 2-PO-7

*A-31*	Nitrile in Heterocyclic Synthesis: New Routes for the Synthesis of Novel 9‑Fluorenone, Indenopyridazine, Indenopyridine and Indenopyrazolotriazine Derivatives
				453
	A. Z. A. E.-B. Hassanien (Suez Canal University, Egypt) Z. E. Kandeel (Cairo University, Egypt)
	Program No.: 2-OP-120 Poster No.: 2-PO-148

*A-32*	Selectivity Control During the Nucleophilic Opening of Epoxides as Key Step in the Syntheses of Pharmaceuticals
				454
	A. K. Chakraborti (National Institute of Pharamaceutical Education and Research, India)
	Program No.: 2-OP-122 Poster No.: 2-PO-150

14:30 - 16:00		SECTION B (Room 302)
Chair: A. Kittaka (Teikyo University, Japan)
*B-24*	A Novel Chiral Phosphole and Its Derivatives: Application of a Chiral Phosphino-Phosphaferrocene to Palladium-Catalyzed Asymmetric Allylic Alkylation
				455
	M. Ogasawara, K. Yoshida, T. Hayashi (Kyoto University, Japan)
	Program No.: 2-OP-90 Poster No.: 2-PO-38

*B-25*	Stereoselective Synthesis of Pyrrolidines and Piperidines via Catalytic Aminyl-radical Reactions
				456
	R. Göttlich (Universität Münster, Germany)
	Program No.: 2-OP-94 Poster No.: 2-PO-39

*B-26*	Catalytic Asymmetric Epoxidation of Conjugated Olefins with (Salen) ruthenium Complex under Photoirradiation
				457
	T. Takeda, K. Nakata, R. Irie, T. Katsuki (Kyushu University, Japan)
	Program No.: 2-OP-98 Poster No.: 2-PO-40

*B-27*	A Novel Synthesis of Pyridine Derivatives via Self-condensation of Cyclic Ketones in aq NH₄Cl under Hydrothermal Conditions
				458
	B. K. Mehta, K. Yanagisawa, H. Kotsuki (Kochi University, Japan)
	Program No.: 2-OP-102 Poster No.: 2-PO-41

*B-28*	Direct and Regioselective Preparation of Pyridyltitanium Compounds from Acetylenes, a Nitrile, and (η²-Propene)Ti(O-i-Pr)₂
				459
	D. Suzuki, H. Urabe, F. Sato (Tokyo Institute of Technology, Japan)
	Program No.: 2-OP-106 Poster No.: 2-PO-42

*B-29*	Intramolecular Alkene Hydroaminations Catalyzed by Simple Amido Derivatives of the Group 3 Metals
				460
	Y. K. Kim, T. Livinghouse (Montana State University, USA) J. E. Bercaw (Califomia Institute of Technology, USA)
	Program No.: 2-OP-110 Poster No.: 2-PO-43

*B-30*	Stereoselective Synthesis of Piperidones and Mannich-Type Products			461
	K. Ishimaru, T. Kojima (The National Defense Academy, Japan)
	Program No.: 2-OP-114 Poster No.: 2-PO-44

*B-31*	Synthesis of New Benzodiazepines NNRT Inhibitors of HIV			462
	A. J. CoGuzza. D. M. Bilder, D. R. Chidester, J. D. Rodgers, C. S. Brosz, G. A. Cain, E. R. Holler, J. L. Hytrek, J. H. Sun, J. -S. Yan, M. X. Xia, C. A. Teleha (DuPont Pharmaceuticals Company, USA)
	Program No.: 2-OP-117 Poster No.: 2-PO-45

*B-32*	*Novel Strategies for Heterocyclic Construction via* Multicomponent Reactions**			463
	V. Nair, A. U. Vinod, S. Bindu, L. Balagopal, C. Rajesh (Regional Research Laboratory, India)
	Program No.: 2-OP-123 Poster No.: 2-PO-155

14:30 - 16:00		SECTION C (Room 303)
Chair: H. Takahata (Tohoku Pharmaceutical University, Japan)
*C-24*	The Generation of Isobenzofuran and its Cycloaddition with Multiple Bond			464
	H. Ohmura, K. Mikami (Tokyo Institute of Technology, Japan)
	Program No.: 2-OP-91 Poster No.: 2-PO-75

*C-25*	The Synthesis of b-Nitropyridines and Their Use in Organic Synthesis			465
	J. M. Bakke, I. Sletvold, H. Svensen (Norwegian University of Science and Technology, Norway)
	Program No.: 2-OP-95 Poster No.: 2-PO-76

*C-26*	Enantioselective Acceleration in Kinetic Resolution with a Chiral Nucleophilic Catalyst
				466
	T. Kawabata, Y. Momose, K. Yamamoto, K. Fuji (Kyoto University, Japan)
	Program No.: 2-OP-99 Poster No.: 2-PO-77

*C-27*	Stereoselective Cyclization Using Palladium (II) Catalyst via Hemiacetal Intermediates
				467
	M. Miyazawa, Y. Hirose, T. Nakano, H. Yokoyama, S. Yamaguchi, Y. Hirai (Toyama University, Japan)
	Program No.: 2-OP-103 Poster No.: 2-PO-78

*C-28*	The Aza-ene Reaction of Heterocyclic Ketene Aminals			468
	I.-T. Huang, M.-X. Wang, J.-H. Zhang, X.-P. Nie (The Chinese Academy of Sciences, China)
	Program No.: 2-OP-107 Poster No.: 2-PO-79

*C-29*	Scale up Synthesis of Natural Compound Analogs from Acetylene, Ketones, Carbon Dioxide and Primary Amines
				469
	N. B. Chernysheva, I. Y. Titov, A. A. Bogolyubov, V. V. Semenov (Zelinsky Institute of Organic Chemistry / Chemical Block Ltd., Russia)
	Program No.: 2-OP-111 Poster No.: 2-PO-80

*C-30*	Exoxides and Azirdines in Organic Synthesis: Total Synthesis of (-)-Boronolide and (-)-Muricatacin. A Simple Approach to Chiral Diamine and other related Ligands
				470
	V. K. Singh, M. Chandrasekhar, K. L. Chandra (Indian Institute of Technology Kanpur, India)
	Program No.: 2-OP-115 Poster No.: 2-PO-81

*C-31*	*Site Directed DNA Cross-linking by Novel Nucleoside Analog via* Synchronous Activation within Duplex**
				471
	T. Kawasaki, F. Nagatsugi, N. Tokuda, M. Maeda, S. Sasaki (Kyushu University, Japan)
	Program No.: 2-OP-118 Poster No.: 2-PO-82

*C-32*	Transfer Reagents: The Synthesis of 3,6-Di(2-Pyridyl)-Pyridazino Norbornadiene and its Use in the Synthesis of bis-dppn Ligands
				472
	D. Margetic, D. N. Butler, R. N. Warrener (Central Queensland University, Australia)
	Program No.: 2-OP-124 Poster No.: 2-PO-156

14:30 - 16:00		SECTION D (Room 304)
Chair: K. Takeda (Hiroshima University, Japan)
*D-24*	New Approach in Synthesis of Heterocycles-Rearrangements of 1,2,3-Triazoles and 1,2,3-Thiadiazoles
				473
	Y. Y. Morzherin, T. V. Glukhareva, V. A. Bakulev (Urals State Technical University, Russia)
	Program No.: 2-OP-92 Poster No.: 2-PO-112

*D-25*	Selective Synthesis of New Tetrazine Derivatives			474
	J. Faragó, Z. Novák, A. Kotschy (Eötvös University, Hungary)
	Program No.: 2-OP-96 Poster No.: 2-PO-113

*D-26*	Synthesis and Cycloaddition of Novel Zwitterionic Pyridine Derivatives			475
	G. Hajós, Z. Riedl, P. Kövér, A. Messmer (Chemical Research Center, Hungary)
	Program No.: 2-OP-100 Poster No.: 2-PO-114

*D-27*	Preparation and Reactivity of D-heterocycle-triosmium Clusters			476
	Q. Lin, W. Leong (National University of Singapore, Singapore)
	Program No.: 2-OP-104 Poster No.: 2-PO-115

*D-28*	Synthetic Applications of N-Phenacylpyridinium Salts Bearing Leaving Group at alpha-Position
				477
	E. Babaev (Moscow State University, Russia)
	Program No.: 2-OP-108 Poster No.: 2-PO-116

*D-29*	Intramolecular 1,3-Dipolar Cycloaddition Initiated by Microwaves			478
	M. Potáček, J. Pospfsil (Masaryk University of Brno, Czech Republic)
	Program No.: 2-OP-112 Poster No.: 2-PO-117

*D-30*	Synthesis using Unprotected Amno Acids; One-Step Synthesis of N-Acetyltryptophan from Indole and Serine
				479
	Y. Hiroki (Chiba University, Japan) Y. Yokoyama. M. Mitsuhashi. Y. Murakami (Toho University, Japan)
	Program No.: 2-OP-116 Poster No.: 2-PO-118

*D-31*	New Class of DNA Binders Based on BisTHF, Bisfuran and Bispyrrole Scaffold
				480
	T. Shibata, F. Nagatsugi, Y. Shibata, M. Maeda, S. Sasaki (Kyushu University, Japan) H. Torigoe (RIKEN (The Institute of Physical and Chemical Research), Japan)
	Program No.: 2-OP-119 Poster No.: 2-PO-119

*D-32*	Dopamine-selective Membrane Potential Changes by Hexahomotrioxacalix[3]arene Hosts Equipped with a Defined Structure for Tripodal Hydrogen Bonding
				481
	K. Odashima, N. Shirai, R. Tanaka, Y. Murakami, J. Miyake, Y. Wasada-Tsutsui (Nagoya City University, Japan) K. Ozaku, S. Amemiya (The University of Tokyo, Japan)
	Program No.: 2-OP-121 Poster No.: 2-PO-149

August 2 (Thu)		Poster Presentation
16:00 - 18:30
*2-PO-1*	New Concept for Blue Flower Color Development by Metal Complex		446
	K. Yoshida, M. Mori, K. Oyama, T. Kondo (Nagoya University, Japan) Y. Toyama (Sugiyama Jogakuen University, Japan)
	Program No.: 2-OP-89 (A-24)

*2-PO-2*	Inhibition and Structural Studies of the Enzyme Porphobilinogen Synthase		447
	F. Stauffer, E. Zizzari, C. Jarret, R. Neier (University of Neuchdtel, Switzerland)
	Program No.: 2-OP-93 (A-25)

*2-PO-3*	Chemoselective Palladium Catalyzed Reaction in Aqueous Media: Selectivity in the Reaction of Bromoaniline with Allylalcohol
			448
	Y. Yokoyama, H. Hikawa. Y. Murakami (Toho University, Japan)
	Program No.: 2-OP-97 (A-26)

*2-PO-4*	Axial Chirality due to an Acyclic Imide-Ar Bond: a Study of Steric and Electronic Effects of Acyl Groups on Racemization
			449
	K. Kondo, T. Iida. H. Fujita, T. Suzuki. Y. Murakami (Toho University, Japan) K. Yamaguchi (Chiba University, Japan)
	Program No.: 2-OP-101 (A-27)

*2-PO-5*	Use of Bis(acylketene) in Heterocycle Synthesis		450
	M. Sato, K. Kondo, T. Katsumata, K. Iwamoto (University of Shizuoka, Japan)
	Program No.: 2-OP-105 (A-28)

*2-PO-6*	Generation and Reaction of Metal-Containing Carbonyl Ylides: Tandem [3+2]-Cycloaddition-Carbene Insertion Leading to Novel Polycyclic Compounds
			451
	N. Iwasawa, M. Shido. H. Kusama (Tokyo Institute of Technology, Japan)
	Program No.: 2-OP-109 (A-29)

*2-PO-7*	Chiral Aziridine-2-carboxylates: Preparation and Utilization for the Synthesis of Phenylalanine and Homophenylalanine
			452
	H.-J. Ha (Hankuk University of Foreign Studies/ ChembioNex Co.,Ltd, HUFS BI, Korea) H.-J. Yoo, C. Park (Sogang University, Korea) W. Lee (Sogang University/ ChembioNex Co., Ltd, HUFS BI Korea) Y. Lim (ChembioNex Co., Ltd, HUFS BI, Korea)
	Program No.: 2-OP-113 (A-30)

*2-PO-8*	4-Nitro-5-Isoxazolone: A Useful Synthetic Reagent for Polyfunctionalized Systems
			482
	N. Nishiwaki, M. Tamura. K. Hori, Y. Tohda. M. Ariga (Osaka Kyoiku University, Japan)

*2-PO-9*	A Column-Free Synthesis of Various Amides, Carbamates, and Ureas Using Polymer-Bound N-hydroxysuccinimide
			483
	M. Katoh, M. Sodeoka (Tohoku University/Japan Science and Technology Corporation, Japan) Y. Baba, T. Shimizu (Tohoku University, Japan)

*2-PO-10*	Synthesis, Molecular Structure and Fluxional Behavior of (R)-7-p-Tolyldinaphtho[2,1-b;1',2'-d]stibole
			484
	S. Yasuike, T. Iida, J. Kurita (Hokuriku University, Japan) K. Yamaguchi, H. Seki (Chiba University, Japan)

*2-PO-11*	Synthesis of Pyrrolidine and Piperidine Derivatives by Photoinduced Electron Transfer Reaction
			485
	T. Takahashi, Y. Yamamura, S. Hirokami (Toyama Medical & Pharmaceutical University, Japan)

*2-PO-12*	Synthetic Studies on GE3: Stereocontrolled Construction of the Acyl Side Chain and the Piperazic Acid Derivatives
			486
	K. Makino, Y. Henmi, M. Terasawa, Y. Hamada (Chiba University, Japan)

*2-PO-13*	Synthetic Studies on Martinelline and Martinellic Acid, Novel G-Protein Linked Receptor Antagonists
			487
	O. Hara, K. Sugimoto, Y. Hamada (Chiba University, Japan)

*2-PO-14*	Preparation and Reactions of 1-Benzoselenopyrylium Salts		488
	M. Yoshida, H. Minamida, K. Yamamoto, H. Sashida (Hokuriku University, Japan)

*2-PO-15*	*Ring Transformations of Dihydroselenines via* Selenonium Ylides**		489
	E. Honda, T. Iwamura, S. Watanabe, T. Kataoka (Giru Pharmaceutical University, Japan)

*2-PO-16*	A One-Pot Intramolecular and Regioselective Cyclization of Nitrile with Styryl Carbon-Carbon Double Bond to Form 3-Substituted Isoindolin-1-one Derivatives
			490
	F. T. Luo, C. H. Chen (Academia Sinica, Taiwan)

*2-PO-17*	(+) and H-4,5-Dialkoxy-2-oxazolidinones as New Class of Chiral Synthons for Optically Pure α-Amino Aldehydes and α-Amino Acids
			491
	H. Matsunaga, T. Morita, T. Kunieda (Kumamoto University, Japan)

2-PO-18	Synthesis and Reaction of Indolizine-1,2-dicarboxylic Anhydride		492
	Y. Miki, R.Yamakawa, H. Hachiken, H. Hibino (Kinki University, Japan)

*2-PO-19*	Alkylation of Metalated O-Silyl Cyanohydrins of b-Silyl-α,b-epoxyaldehydes via Tandem Ring Opening-Brook Rearrangement-Allylic Rearrangement
			493
	E. Kawanishi, M. Sasaki, K. Takeda (Hiroshima University, Japan)

2-PO-20	Synthesis and Reaction of Indolo[1,2-b]indazoles		494
	Y.-M. Zhu, K. Kaneko, K. Shiono, T. Sato, H. Katayama (Niigata College of Pharmacy, Japan)

*2-PO-21*	Indium(I)-mediated Stereoselective Synthesis of 1,3-Amino Alcohols Bearing Three Chiral Centers by Umpolung of Chiral 2-Ethynylaziridines
			495
	H. Ohno, H. Hamaguchi, T. Tanaka (Osaka University, Japan)

*2-PO-22*	Application of Optically Active Ligands Possessing Pro N-Ar Axial Chirality to Transition Metal-Catalyzed Asymmetric Reactions
			496
	K. Kondo, K. Kazuta, H. Fujita, Y. Sakamoto, Y. Murakami (Toho University, Japan)

*2-PO-23*	Development of Chemoselective and Enantioselective N-Acylation Reagents		497
	Y. Murakami, K. Kondo (Toho University, Japan)

*2-PO-24*	Synthesis and Charge Transfer Complexation of Chiral Polynitrohelicenes		498
	D. Nakano, S. Anzai, H. Okubo, M. Yamaguchi (Tohoku University, Japan)

*2-PO-25*	Synthetic Studies of Pseurotin A, a Highly Functionalized γ-Lactam Natural Product
			499
	S. Aoki, T. Ohi, K.Takao, K. Tadano (Keio University, Japan)

*2-PO-26*	A Facile Synthesis of Fluoromethylated Heterocyclic Compounds		500
	M. Suzuki, M. Mori, Y. Suzuki, M. Sato (University of Shizuoka, Japan)

*2-PO-27*	Introduction of Carbon Substituent to Dehydroacetic Acid at the 5-Position by Stille Coupling Reaction
			501
	Y. Katsumata, K. Iju, K. Ikeda, M. Sato (University of Shizuoka, Japan)

*2-PO-28*	Syntheses of Chiral Helicenepolyamines		502
	H. Okubo, S. Anzai, S. Honzawa, M. Yamaguchi (Tohoku University, Japan)

*2-PO-29*	Asymmetric Syntheses of Nepetalactones Utilizing Biocatalysis		503
	T. Katoh, K. Okamoto, H. Tanaka, M. Node (Kyoto Pharmaceutical University, Japan)

*2-PO-30*	Enantiodivergent Synthesis of (+)- and (-)-Ferruginine Utilizing PLE-catalyzed Asymmetric Dealkoxycarbonylation
			504
	T. Katoh, T. Nakai, K. Kakiya, S. Nakamura, M. Node (Kyoto Pharmaceutical University, Japan)

*2-PO-31*	Construction of Heterocyclic Compounds by Use of α-Diazophosphonates: New One-pot Syntheses of Indole and Isocoumarin
			505
	Y. Nakamura, T. Ukita (Tanabe Seiyaku Co., Ltd., Japan)

*2-PO-32*	Regioselective Sulfonation at the C-2 Hydroxyl Group of Cyclodextrins by the Combination of Sulfonyl Imidazole and Molecular Sieves
			506
	K. Teranishi, K. Watanabe, F. Ueno (Mie University, Japan)

*2-PO-33*	Asymmetric Aerobic Oxidative Cyclization Catalyzed by (Salen) ruthenium Complexes
			507
	K. Masutani, T. Uchida, R. Irie, T. Katsuki (Kyushu University, Japan)

*2-PO-34*	Highly Enantioselective Hetero Diels-Alder Reaction Catalyzed by Metaliosalen Complexes
			508
	K. Aikawa, Y. Matsuoka, R. Irie, T. Katsuki (Kyushu University, Japan)

*2-PO-35*	Selective Nuclephilic Substitutions on 3-Nitropyridines		509
	H. Svensen, J. M. Bakke (Organic Chemistry Laboratories, Norway)

*2-PO-36*	*Tetrahydrofuranylation of Alcohols with Hypervalent tert-Butylperoxyiodane in the Presence of Carbon Tetrachloride*
			510
	T. Sueda, M. Ochiai (University of Tokushima, Japan)

*2-PO-37*	Synthesis and Photodynamic Activities of Monoazaporphyrins and its Azoniasalt
			511
	S. Kai, S. Hiramitsu, M. Suzuki, Y. Masaki (Gifu Pharmaceutical University, Japan)

*2-PO-38*	A Novel Chiral Phosphole and Its Derivatives: Application of a Chiral Phosphino-Phosphaferrocene to Palladium-Catalyzed Asymmetric Allylic Alkylation
			455
	M. Ogasawara, K. Yoshida, T. Hayashi (Kgoto University, Japan)
	Program No.: 2-OP-90 (B-24)

*2-PO-39*	Stereoselective Synthesis of Pyrrolidines and Piperidines via Catalytic Aminyl-radical Reactions
			456
	R. Gottlich (Universität Münster, Germany)
	Program No.: 2-OP-94 (B-25)

*2-PO-40*	Catalytic Asymmetric Epoxidation of Conjugated Olefins with (Salen) ruthenium Complex under Photoirradiation
			457
	T. Takeda, K. Nakata, R. Irie, T. Katsuki (Kgushu University, Japan)
	Program No.: 2-OP-98 (B-26)

*2-PO-41*	A Novel Synthesis of Pyridine Derivatives via Self-condensation of Cyclic Ketones in aq NH₄Cl under Hydrothermal Conditions
			458
	B. K. Mehta, K. Yanagisawa, H. Kotsuki (Kochi University, Japan)
	Program No.: 2-OP-102 (B-27)

*2-PO-42*	Direct and Regioselective Preparation of Pyridyltitanium Compounds from Acetylenes, a Nitrile, and (η²-Propene)Ti(O-i-Pr)₂
			459
	D. Suzuki, H. Urabe, F. Sato (Tokyo Institute of Technology, Japan)
	Program No.: 2-OP-106 (B-28)

*2-PO-43*	Intramolecular Alkene Hydroaminations Catalyzed by Simple Amido Derivatives of the Group 3 Metals
			460
	Y. K. Kim, T. Livinghouse (Montana State University, USA) J. E. Bercaw (California Institute of Technology, USA)
	Program No.: 2-OP-110 (B-29)

*2-PO-44*	Stereoselective Synthesis of Piperidones and Mannich-Type Products		461
	K. Ishimaru, T. Kojima (The National Defense Academy, Japan)
	Program No.: 2-OP-114 (B-30)

*2-PO-45*	Synthesis of New Benzodiazepines NNRT Inhibitors of HIV		462
	A. J. Cocuzza, D. M. Bilder, D. R. Chidester, J. D. Rodgers, C. S. Brosz, G. A. Cain, E. R. Holler, J. L. Hytrek, J.-H. Sun, J. -S. Yan, M. X. Xia, C. A. Teleha (DuPont Pharmaceuticals Company, USA)
	Program No.: 2-OP-117 (B-31)

*2-PO-46*	Crystallization-induced Asymmetric Transformation of Planar-chiral Pyridinophanes. Chirality Efficient Syntheses of (S)-and (R)-Bridged Nicotinic Acids
			512
	N. Kanomata (Meiji University / PRESTO / Japan Science and Technology Corporation (JST), Japan) S. Anada, M. Yamaguchi, Y. Ochiai (Meiji University, Japan)

*2-PO-47*	Novel and Efficient Synthesis for Perfluoroalkylated Heterocyclic Compounds
			513
	M. Yoshida, T. Muraoka, M. Ohkoshi, H. Matsuyama, M. Iyoda (Tokgo Metropolitan University, Japan)

*2-PO-48*	Synthesis of Isoindolinone Using Ir-catalyzed Reductive Amination of o-Formylbenzoic acids
			514
	T. Igarashi, K. Ooe, I. Shimizu (Waseda University, Japan)

*2-PO-49*	Convergent Synthesis of Six-Membered Polycyclic Ethers via Acetylenic Intermediates
			515
	Y. Mori, H. Hayashi (Meijo University, Japan)

*2-PO-50*	*Synthesis of Enantiomerically Enriched Oxazolidinones via* Nitrosation-Deamination Cyclization**
			516
	M. Suzuki, T. Sugai (Keio University, Japan)

*2-PO-51*	A Practical Synthesis of a Diltiazem Key Intermediate via Chiral Dioxirane-Mediated Catalytic Asymmetric Epoxidation
			517
	S. Yamada, T. Furutani, T. Kuroda, M. Seki (Tanabe Seigaku Co., Ltd., Japan)

*2-PO-52*	Development of New Synthetic Method of Indole Derivatives and Its Application to Natural Products Syntheses
			518
	K. Hiroya, S. Itoh, Y. Kanamori, T. Sakamoto (Tohoku University, Japan)

*2-PO-53*	The Control of Isocoumarin vs Phthalide Cyclization by Acid or Base Catalyst
			519
	M. Uchiyama (The University of Tokyo, Japan) H. Ozawa, T. Sakamoto (Tohoku University, Japan)

*2-PO-54*	Synthesis of a 1,6,6a λ⁴-Triselenapentalene and a 4H-Selenin-4-selone from d-Camphor p-Toluenesulfonyhydrazone
			520
	K. Shimada, M. Takiya, S. Aoyagi, Y. Takikawa (Iwate University, Japan)

*2-PO-55*	Synthesis of Cyclic Sulfones from Alkynyl Propargyl Sulfones by Treatment of an Amine or an Enamine
			521
	S. Aoyagi, J. Murakami, K. Shimada, Y. Takikawa (Iwate University, Japan)

*2-PO-56*	A Novel Regioselective Preparation of Substituted Indoles via Aromatic Pummerer-Type Reaction of p-Sulfinylanilines
			522
	S. Akai, N. Morita, N. Kawashita, Y. Nakamura, Y. Kita (Osaka University, Japan)

*2-PO-57*	Synthesis of 9,11-Diazapentacyclo[6.4.0.0^1.3.O^2.5.0^4.8]-dodecane-2,4-dione Derivatives
			523
	K. Ohkura, A. Sakushima, K. Seki (Health Sciences University of Hokkaido, Japan) K. Nishijima, Y. Kuge (Hokkaido University, Japan)

*2-PO-58*	Building Blocks in the Construction of Oligodibenzothiophenes		524
	T. Thiemann, K. Kumazoe, K. Arima, S. Mataka (Kgushu University, Japan)

*2-PO-59*	*Reaction of 2-Methoxy-5-tert-Butyl-3H-azepine with Sodium Alkoxide and Alkyllithium*
			525
	K. Satake, V. Kubota, H. Okamoto (Okagama University, Japan) M. Kimura (Kgushu University, Japan)

*2-PO-60*	Reaction of 2-Phenylpyrimido[4,5-d]pyridazines with Nucleophiles		526
	E. Oishi, C. Sugiyama, N. Inahashi, K. Iwamoto (University of Shizuoka, Japan)

*2-PO-61*	5-Nitro-2-pyridinesulfonic Acid as Substrate for 2,5-Substituted Pyridines		527
	J. M. Bakke, H. Gautun, E. Ranes, I. Sletvold (Norwegian University of Science and Technology, Norway) C. Rømming (University of Oslo, Norway)

*2-PO-62*	Carbamotelluroate-Mediated Radical Cyclization of Enynes		528
	Y. Shimizu, N. Kambe (Osaka University, Japan) T. Shin-ike, S. Fujiwara (Osaka Dental University, Japan)

*2-PO-63*	Vanadyl Triflate-Catalyzed Nucleophilic Acyl Substitutions of Anhydrides		529
	C.-T. Chen, J.-H. Kuo, C.-H. Li, N. B. Barhate (National Taiwan Normal University, Taiwan)

*2-PO-64*	The Rearrangement of Isoquinolines to Benzazepine Alkaloids		530
	V. Bhavakul (Chulabhom Research Institute) King Mongkut's University of Technology, Thonburi, Thailand) S. Ruchirawat (Chulabhom Research Institutel Mahidol University, Thailand)

*2-PO-65*	Further Development for the Synthesis of Lamellarin Alkaloids		531
	P. Ploypradith (Chulabhom Research Institute, Thailand) W. Jinaglueng, C. Pavaro (Mahidol University, Thailand) S. Ruchirawat (Chulabhom Research Institutel Mahidol University, Thailand)

*2-PO-66*	Radical Addition of p-Toluenesulfonyl Bromide and p-Toluenesulfonyl Iodide to Allenic Alcohols and Sulfonamides in the Presence of AIBN: Synthesis of Heterocyclic Compounds
			532
	S.-K. Kang, B.-S. Ko, Y.-H. Ha (Sungkgunkwan University, Korea)

*2-PO-67*	p-Toluenesulfonyl-Mediated Radical Cyclization of Bis(allenes) Utilizing p-TsBr and p-TsSePh
			533
	S.-K. Kang, Y.-H. Ha (Sungkgunkwan University, Korea)

*2-PO-68*	The Palladium Complex-Catalyzed Regio- and Stereoselective Carbocyclization of Bis(allenes) Using Reagents Involving Ge-Sn σ-Bond
			534
	S.-K. Kang, Y.-T. Hong (Sungkgunlaoan University, Korea)

*2-PO-69*	Asymmetric Addition of Silyl Enol Ethers of Allyltin Reagents to Aromatic C=N Bonds and Its Application to the Synthesis of Isoquinoline and Indole Alkaloids
			535
	T. Itoh, K. Nagata, M. Miyazaki, Y. Matsuya, A. Ohsawa (Showa University, Japan)

*2-PO-70*	Synthetic Study of Cocculolidine		536
	T. Kawasaki, H. Watanabe, T. Kitahara (The University of Tokyo, Japan)

*2-PO-71*	Design, Synthesis and Application of Chiral Spiro Bis(isoxazoline) Ligands(SPRIXs)		537
	M. Arai, T. Shinohara, M. Kuraishi, T. Arai, H. Sasai (The Institute of Scientific and Industrial Research (ISIR) Osaka University, Japan)

*2-PO-72*	*Synthetic Studies on Spectamine via* Pd(ll) Catalyzed Stereoselective Cyclization**
			538
	H. Makabe, L. K. Kong, K. Maehara, M. Hirota (Shinshu University, Japan)

*2-PO-73*	New Approches to Various Alkaloid Analogues by [3+3] Cyclisations		539
	P. Nemes, P. Scheiber (Szent István University, Hungary) J. Kovács, G. Tóth (Budapest University of Technology and Economics, Hungary)

*2-PO-74*	Palladium (II)-Catalyzed Asymmetric 1,3-Dipolar Cycloaddition of Nitrones		540
	K. Hori, N. Nishiwaki, Y. Tohda, M. Ariga (Osaka Kyoiku University, Japan) T. Ohta, I. Furukawa (Doshisha University, Japan)

*2-PO-75*	The Generation of Isobenzofuran and its Cycloaddition with Multiple Bond		464
	H. Ohmura, K. Mikami (Tokyo Institute of Technology, Japan)
	Program No.: 2-OP-91 (C-24)

*2-PO-76*	The Synthesis of b-Nitropyridines and Their Use in Organic Synthesis		465
	J. M. Bakke, I. Sletvold, H. Svensen (Norwegian University of Science and Technology, Norway)
	Program No.: 2-OP-95 (C-25)

2-PO-77	Enantioselective Acceleration in Kinetic Resolution with a Chiral Nucleophilic Catalyst
			466
	T. Kawabata, Y. Momose, K. Yamamoto, K. Fuji (Kyoto University, Japan)
	Program No.: 2-OP-99 (C-26)

*2-PO-78*	Stereoselective Cyclization Using Palladium (II) Catalyst via Hemiacetal Intermediates
			467
	M. Miyazawa, Y. Hirose, T. Nakano, H. Yokoyama, S. Yamaguchi, Y. Hirai (Toyama University, Japan)
	Program No.: 2-OP-103 (C-27)

*2-PO-79*	The Aza-ene Reaction of Heterocyclic Ketene Aminals		468
	Z.-T. Huang, M.-X. Wang, J.-H. Zhang, X.-P. Nie (The Chinese Academy of Sciences, China)
	Program No.: 2-OP-107 (C-28)

*2-PO-80*	Scale up Synthesis of Natural Compound Analogs from Acetylene, Ketones, Carbon Dioxide and Primary Amines
			469
	N. B. Chernysheva, I. Y. Titov, A. A. Bogolyubov, V. V. Semenov (Zelinsky Institute of Organic Chemistry / Chemical Block Ltd., Russia)
	Program No.: 2-OP-111 (C-29)

*2-PO-81*	Exoxides and Azirdines in Organic Synthesis: Total Synthesis of (‑)‑Boronolide and (-)-Muricatacin. A Simple Approach to Chiral Diamine and other related Ligands
			470
	V. K. Singh, M. Chandrasekhar, K. L. Chandra (Indian Institute of Technology Kanpur, India)
	Program No.: 2-OP-115 (C-30)

*2-PO-82*	*Site Directed DNA Cross-linking by Novel Nucleoside Analog via* Synchronous Activation within Duplex**
			471
	T. Kawasaki, F. Nagatsugi, N. Tokuda, M. Maeda, S. Sasaki (Kyushu University, Japan)
	Program No.: 2-OP-118 (C-31)

*2-PO-83*	Thermal Stability and Improved Synthesis of Fulleropyrrolidine Using Polymer-Supported Azomethine Ylide
			541
	Y. Kawamura, Y. Akai, M. Nishiuchi, M. Tsukayama (The University of Tokushima, Japan)

*2-PO-84*	Oxidative Rearrangement of 2'-Hydroxychalcones to Isoflavones Using Hypervalent Iodine(III) Reagent
			542
	Y. Kawamura, M. Maruyama, M. Nishiuchi, M. Tsukayama (The University of Tokushima, Japan)

*2-PO-85*	Synthesis of New Chiral N-[1-(2-Pyridinyl)ethyl]pyrrolidine Ligands for Asymmetric Reaction
			543
	J. Uenishi, M. Hamada (Kyoto Pharmaceutical University, Japan)

*2-PO-86*	Enantioselective Total Synthesis of 2-Arylbenzofuran Lignans, (+)‑Grossamide and (+)-Dehydrodiconiferyl Alcohol
			544
	M. Okazaki, Y. Shuto (Ehime University, Japan)

*2-PO-87*	Direct Platinum-Catalyzed Allylation of Anilines Using Allylic Alcohols		545
	S.-C. Yang, Y.-C. Tsai, Y.-J. Shue (Kaohsiung Medical University, Taiwan)

*2-PO-88*	Synthetic Study on Kaitocephalin, a Potent AMPA/KA Receptor Antagonist		546
	H. Kobayashi, M. Okue, H. Watanabe, T. Kitahara (The University of Tokyo, Japan)

*2-PO-89*	Syntheses, Structures and Reactions of Several "Cyclized" Thianthrene Derivatives
			547
	H. Morita, T. Nakajima, K. Kunimasa, Y. Oida, N. Kitao, T. Fujii (Toyama University, Japan)

*2-PO-90*	Convenient Synthesis of 2-Aminopyrrole Derivatives		548
	M. Yumoto, T. Kawabuchi, H. Sato, M. Takashima (Fuji Photo Film Co., Lid., Japan)

*2-PO-91*	Studies Toward the Total Synthesis of Scyphostatin: First Entry to the Highly Functionalized Cyclohexenone Segment
			549
	T. Katoh, T. Izuhara (Sagami Chemical Reserch Center, Japan)

*2-PO-92*	Synthesis of 5.5-bis(hydroxymethyl)-1,4-dideoxy-1,4-iminothreoitol		550
	E. Mironiuk, E. Kolaczkowska, W. Sas (Warsaw University of Technology, Poland)

*2-PO-93*	Synthesis of Polyhydroxylated Derivatives of Indolizidine and Quinolizidine by Intramolecular 1.3-Dipolar Cycloaddition of N-(3-alkenyllnitrones from 2,3:5,6-di-O-isopropylidene-D-mannofuranose
			551
	P. Gębarowski, W. Sas (Warsaw University of Technology, Poland)

*2-PO-94*	Anionic Cyclization with Triple Carbon-Carbon Bond under Phase Transler Catalysis Conditions (PTC)
			552
	K. Michalski, A. Jonczyk (Warsaw University of Technology, Poland)

*2-PO-95*	Enantioselective Lithiation of Azalerrocene Derivatives		553
	T. Fukuda, K. Imazato, M. Iwao (Nagasaki University, Japan)

*2-PO-96*	Stereoselective Total Synthesis of Tricyclic Terpenoid Chroman (+)-NG-121 Methyl Ether
			554
	S. Inoue, F. Iwasaki, C. Nakagawa, K. Honda (Yokohama National University, Japan)

*2-PO-97*	Single-Step Synthesis of Fused Hetero-polycyclic Compounds from Salicylaldehydes and Unsaturated Cyclic Alcohols of Their Sulfur Analogs
			555
	S. Inoue, M. Nagao, P. Wang, M. Yamada, K. Honda (Yokohama National University, Japan)

*2-PO-99*	Enantioselective Benzylation of the Lithium Enolate of 1-Tetralone Mediated by a Chiral Tetradentate Amine
			556
	K. Tanaka, T. Furuta, R. Shirai, K. Koga (Nara Institute of Science and Technology, Japan)

*2-PO-100*	*On the Synthesis of cis-* and trans- 5-Cyano-6-arylsulphonamido-1,3-dioxepanes**
			557
	M. Orešić, M. Dumić (PLIVA d.d., Croatia)

*2-PO-101*	Asymmetric Protonation of Lithium Enolate of Alanine Derivative Using Chiral Brønsted Acids
			558
	A. Yanagisawa (Chiba University, Japan) Y. Matsuzaki, H. Yamamoto (Nagoya University / CREST / Japan Science and Technology Corporation (JST), Japan)

*2-PD-102*	Catalytic Asymmetric 1,3-Dipolar Cycloadditions of Nitrones with Alkenoyl Oxazolidinones Catalyzed by Bis(oxazolyl)pyridine/Ni(II) Complex
			559
	S. Iwasa, S. Tsushima, K. Nishiyama, H. Nishiyama (Toyohashi University of Technology, Japan)

*2-PD-103*	*Simple Synthesis of Carbazoles from N,N-Diarylphthalimides with AlCl₃ via* Electron Delicient Nitrogen**
			560
	T. Sakamoto, Y. Aoki, Y. Kikugawa (Josai University, Japan)

*2-PO-104*	Solid Phase Synthesis of Oxazoles Via a Cyclization-Release Reaction		561
	M. Pulici, F. Quartieri (Pharmacia, Italy)

*2-PO-105*	Study on the Synthesis of Benzoxazole Derivatives by the Reaction of 2-Aminophenol with Aliphatic Acids and Acidic Catalysts
			562
	G. C. Penieres, A. O. Romero, E. P. Gómez, R. S. Rosas, C.T. Alvarez (Universidad Nacional Autónoma, Mexico)

*2-PO-106*	Synthesis of New Prido[2,3-d]pirimidine Derivatives by Phase Transfer Reaction
			563
	R. D. Yánez, E. T. Diaz, C. T. Alvarez, G. C. Penieres (Universidad Nacional Autónoma, Mexico)

*2-PO-107*	Chemoselective Reduction of Epoxide with Sml₂		564
	F. Matsuda, M. Sato (Hokkaido University, Japan)

*2-PO-108*	Synthesis of 3-Alkoxy-pyrimidines		565
	C. Goebel, D. Geffken (University of Hamburg, Germany)

*2-PO-109*	Synthesis of 4-Alkoxy-benzo[f]-1,4-thiazepine-3,5-diones		566
	K. Beck, D. Geffken (University of Hamburg, Germany)

2-PO-110	Palladium Catalysis in Carbohydrate Synthesis		567
	H. Kawabata, K. Yoshimoto, K. Yamada, M. Hayashi (Kobe University, Japan)

*2-PO-111*	Novel Heterocyclic Compounds from the Polyhalobutadienes and Polyhalobutenes
			568
	C. İBİŞ (Istanbul University, Turkey)

*2-PO-112*	New Approach in Synthesis of Heterocycles-Rearrangements of 1,2,3‑Triazoles and 1,2,3-Thiadiazoles
			473
	Y. Y. Morzherin, T. V. Glukhareva, V. A. Bakulev (Urals State Technical University, Russia)
	Program No.: 2-OP-92 (D-24)

*2-PO-113*	Selective Synthesis of New Tetrazine Derivatives		474
	J. Faragó, Z. Novák, A. Kotschy (Eötvös University, Hungary)
	Program No.: 2-OP-96 (D-25)

*2-PO-114*	Synthesis and Cycloaddition of Novel Zwitterionic Pyridine Derivatives		475
	G. Hajós, Z. Riedl, P. Kövér, A. Messmer (Chemical Research Center, Hungary)
	Program No.: 2-OP-100 (D-26)

*2-PO-115*	Preparation and Reactivity of D-heterocycle-triosmium Clusters		476
	Q. Lin, W. Leong (National University of Singapore, Singapore)
	Program No.: 2-OP-104 (D-27)

*2-PO-116*	Synthetic Applications of N-Phenacylpyridinium Salts Bearing Leaving Group at alpha-Position
			477
	E. Babaev (Moscow State University, Russia)
	Program No.: 2-OP-108 (D-28)

*2-PO-117*	Intramolecular 1,3-Dipolar Cycloaddition Initiated by, Microwaves		478
	M. Potáček, J. Pospíšil (Masaryk University of Brno, Czech Republic)
	Program No.: 2-OP-112 (D-29)

*2-PO-118*	Synthesisusing Unprotected Amno Acids; One-Step Synthesis of N-Acetyltryptophan from Indole and Serine
			479
	Y. Hiroki (Chiba University, Japan) Y. Yokoyama, M. Mitsuhashi, Y. Murakami (Toho University, Japan)
	Program No.: 2-OP-116 (D-30)

*2-PO-119*	New Class of DNA Binders Based on BisTHF, Bisfuran and Bispyrrole Scattold
			480
	T. Shibata, F. Nagatsugi, Y. Shibata, M. Maeda, S. Sasaki (Kyushu University, Japan) H. Torigoe (RIKEN (The Institute of Physical and Chemical Research), Japan)
	Program No.: 2-OP-119 (D-31)

*2-PO-120*	New Labdane-Type Diterpene Lactones with Antiinflammatory Activity, Hedychilactones A, B, and C, from Hedychium coronarium
			569
	H. Matsuda, T. Morikawa, I. Toguchida, M. Yoshikawa (Kyoto Pharmaceutical University, Japan)

*2-PO-121*	*Phytoestrogens from the Roots of Polygonum cuspidatum* (Polygonaceae): Structure-Requirement of Hydroxyanthraquinones for Estrogenic Activity**
			570
	H. Matsuda, H. Shimoda, T. Morikawa, M. Yoshikawa (Kyoto Pharmaceutical University, Japan)

*2-PO-122*	Synthesis and NMR Spectra of Furyl-and Thienyl Silacycloalkanes		571
	L. Ignatovich, J. Popelis, E. Lukevics (Latvian Institute of Organic Synthesis, Latvia)

*2-PO-123*	*Enantioselective Synthesis of (-)-(6R,7S)-Nitramine*		572
	K. A. Tehrani, M. Boelens, N. De Kimpe (Ghent University, Belgium) V. Yu (Institute of Chemical Sciences, Kazakhstàn)

*2-PO-124*	Regioselective Cyclization of 3-Acylindole Derivatives with Aluminum Chloride
			573
	T. Komoda, S. Nakatsuka (Gifu University, Japan)

*2-PO-125*	Study on Polymerization of N-acylindole		574
	K. Fujino, N. Tajima, S. Nakatsuka (Gifu University, Japan)

*2-PO-126*	Synthesis of Monomethyl Derivatives of Epigallocatechin Gallate (EGCg)		575
	E. Yanase, S. A. Sani, S. Nakatsuka (Gifu University, Japan)

*2-PO-127*	Palladium Charcoal Caralyzed Cross-Couplings: A Convenient Route to Ethynylpyridines and Arylpyridines
			576
	A. Torii, T. Tagata, M. Nishida (Koei Chemical Co., Ltd., Japan)

*2-PO-128*	Synthesis of Poly-functionalized Isoquinolone Derivatives Using 4-Methyl-4H-1,3-oxazin-4-ones
			577
	Y. Kawata, Y. Morita, H. Ouchi, Y. Saito, H. Takahata, Y. Yamamoto (Tohoku Pharmaceutical University, Japan)

*2-PO-129*	Synthetic Studies of Tedanolides by Taking Advantage of Convertible Protecting Groups, Six-membered 4-Methoxybenzylidene Acetals
			578
	S. Kusaka, K. Matsui, B.-Z. Zheng, H. Yamada, O. Yonemitsu (Okayama University of Science, Japan)

*2-PO-130*	Catalytic Asymmetric Synthesis of α,b-Epoxyesters via Darzens Reaction under Phase- Transfer Conditions
			579
	S. Arai, Y. Suzuki, K. Tokumaru, T. Shioiri (Nagoya City University, Japan)

*2-PO-131*	Preparation and Properties of A New Generation of Chiral Nucleophilic Catalysts Derived from 4-Hydroxyproline
			580
	T. Kawabata, R. Stragies, T. Fukaya, K. Fuji (Kyoto University, Japan)

*2-PO-132*	Design and Synthesis of New Optically Active Cyclic Phosphines.		581
	A. Ohashi, T. Sugiura, H. Hayashi, H. Danjo, T. Imamoto (Chiba University, Japan)

*2-PO-133*	Diels-Alder Reaction of 1-Imino Derivatives of 3,4-Di-t-butylthiophene		582
	T. Otani, J. Takayama, Y. Sugihara, A. Ishii, J. Nakayama (Saitama University, Japan)

*2-PO-134*	Pyrrolo[2,3-e][1,2,3]triazolo[1,5-a]pyrimidine. A New Tricyclic Ring System of Biological Interest
			583
	A. Lauria, P. Diana, P. Barraja, A. Montalbano, G. Dattolo, G. Cirrincione, A. M. Almerico (University of Palermo, Italy)

*2-PO-135*	Coloration and Crystal Structures of Phenyl-2-pyridinylborinic Acid Dimer Complex
			584
	T. Murafuji, H. Nakamura, T. Iwakiri, Y. Sugihara (Yamaguchi University, Japan) K. Takakura (The University of Tokyo, Japan)

*2-PO-136*	1,3-Dithian-2yl-arylmethanols: Acid Catalyzed Rearrangement, Cycloaromatization and Dimerization
			585
	C.W. Ong, C. Y. Yu (National Sun Yat Sen University, Taiwan)

*2-PO-137*	Formation of Fused Rings using Palladium-Catalyzed Intramolecular Benzannulation Strategy
			586
	T. Kawasaki, SoSaito, Y. Yamamoto (Tohoku University, Japan)

*2-PO-138*	Novel Synthetic Analogues of Coformycin Containing the Imidazo[4,5-e] [1,2,4]triazepine Ring System as Inhibitors of Adenosine Deaminase
			587
	A. Reayi, R. S. Hosmane (University of Maryland, USA)

*2-PO-139*	Inhibition of MIF Bioactivity by Rational Design of Pharmacological Inhibitor of the MIF Tautomerase Activity
			588
	A. Dios, R. A. Mitchell, B. Aljabari, C. N. Metz, R. Bucala, Y. Al-Abed (The Picower Institute for Medical Research, USA)

*2-PO-140*	Synthesis and Pharmacological Evaluation of Piperidyl- and Tetrahydroisoquinolyl Containing Thiazoles
			589
	E. Lukevics, A. Zablotskaya, I. Segal (Latvian Institute of Organic Synthesis, Latvia) A. Geronikaki (Aristotelian University of Thessaloniki, Greece)

*2-P0-141*	Synthesis and Antitumor Activity of Silylbenzimidazole Derivatives		590
	E. Lukevics, P. Arsenyan, I. Shestakova, O. Pudova (Latvian Institute of Organic Synthesis, Latvia)

*2-PO-142*	Synthesis and Evaluation of Water-soluble Taxoids		591
	T. Mandai, H. Okumoto, T. Oshitari (Kurashiki University of Science and the Arts, Japan) K. Nakanishi, K. Mikuni, K. Hara, K. Hara (Bio Research Corportion of Yokohama, Japan) W. Iwatani, T. Amano, K. Nakamura, Y. Tsuchiya (Kaken Pharmaceutical Co., LTD., Japan)

*2-PO-143*	*Molecular Design of a New Class of Spin-labeled Ribonucleosides with N‑tert-Butylaminoxyl Radicals*
			592
	M. Aso, T. Ikeno, K. Norihisa, N. Koga, H. Suemune (Kyushu University, Japan)

*2-PO-144*	Synthesis and Structure-activity Relationship Study of Antimicrotubule Diketopiperazines, Phenylahistin and Its Derivatives
			593
	Y. Hayashi, S. Orikasa, K.Tanaka, Y. Kiso (Kyoto Pharmaceutical University, Japan) K. Kanoh (Marine Biotechnology Institute, Japan)

*2-PO-145*	Direct Proton NMR Chirality Quantitaiton for Chiral Aldehyde Analogues		594
	K. Nagasawa, M. Gotoh, M. Hasegawa (Hokkaido College of Pharmacy, Japan)

*2-PO-146*	Synthesis of 3-Alkyl(aryl)-5-(alkylsulfanyl)-[1,3]thiazolo[4',5':4,5]pyrimido[1,6-a]benzimidazole-2(3H)-thiones
			595
	A. Ivachthenko, S. Kovalenko, A. Parkhomenko (Chemical Diversity Labs, Inc., USA)

*2-PO-147*	New Heterocyclic Scaffolds Containing the 2-Fluoronitrophenyl Moiety		596
	A. Ivachtchenko, A. Khizhan (Chemical Diversity Labs, Inc., USA)

*2-PO-148*	Nitrile in Heterocyclic Synthesis: New Routes for the Synthesis of Novel 9-Fluorenone, Indenopyridazine, Indenopyridine and Indenopyrazolotriazine Derivatives
			453
	A. Z. A. E. -B. Hassanien (Suez Conal University, Egypt) Z. E. Kandeel (Cairo University, Egypt)
	Program No.: 2-OP-120 (A-31)

*2-PO-149*	Dopamine-selective Membrane Potential Changes by Hexahomotrioxacalix[3]arene Hosts Equipped with a Defined Structure for Tripodal Hydrogen Bonding

			481
	K. Odashima, N. Shirai, R. Tanaka, Y. Murakami, J. Miyake, Y. Wasada-Tsutsui (Nagoya City University, Japan) K. Ozaku, S. Amemiya (The University of Tokyo, Japan)
	Program No.: 2-OP-121 (D-32)

*2-PO-150*	Selectivity Control During the Nucleophilic Opening of Epoxides as Key Step in the Syntheses of Pharmaceuticals
			454
	A. K. Chakraborti (National Institute of Pharamaceutical Education and Research, India)
	Program No.: 2-OP-122 (A-32)

*2-PO-151*	An Efficient Method for Syntheses of Thiazoles, Oxazoles and Imidazoles		597
	A. K.Chakraborti, G. Kaur, L. Sharma, C. Selvam (National Institute of Pharmaceutical Education and Research (NIPER), India)

*2-PO-152*	A Novel Imidazole Ring Transformation		598
	A. A. Tolmachev, V. V. Ivanov, A. A. Yurchenko, A. M. Pinchuk (National Academy of Sciences of Ukraine, Ukraine)

*2-PO-153*	Synthesis of Morpholines Polysubtited		599
	H. Harkat, M. Benkhaled, M. Laabassi (University of Batna, Algeria) R. Gree, D. Gree (Universiy of Rennes I. Rennes, France)

*2-PO-154*	New Approaches to Polycyclic Piperazindiones		600
	S. Jin, J. Liebscher (Humboldt-University, Germany)

*2-PO-155*	*Novel Strategies for Heterocyclic Construction via* Multicomponent Reactions**
			463
	V. Nair, A. U. Vinod, S. Bindu, L. Balagopal, C. Rajesh (Regional Research Laboratory, India)
	Program No.: 2-OP-123 (B-32)

*2-PO-156*	Transfer Reagents: The Synthesis of 3,6-Di(2-Pyridyl)-Pyridazino Norbornadiene and its Use in the Synthesis of bis-dppn Ligands
			472
	D. Margetic, D. N. Butler, R. N. Warrener (Central Queensland University, Australia)
	Program No.: 2-OP-124 (C-32)

*2-PO-157*	2,3,4-Triphenyl-3-azabicyclo[3.2.0]hepta-1,4-diene. Facile Ring Opening by Nucleophiles and Novel Reactions with Dimethyl Acetylenedicarboxylate
			601
	K. Matsumoto, S. Goto, J. C. Kim, N. Hayashi (Kyoto University, Japan) T. Uchida (Fukui University, Japan) A. Kakehi (Shinshu University, Japan)

*2-PO-158*	Novel Synthetic Route to Allyl Cyanamides: Palladium-Catalyzed Coupling of Isocyanides, Allyl Carbonate, and Trimethylsilyl Azide
			602
	S. Kamijo, T. Jin, Y. Yamamoto (Tohoku University, Japan)

*2-PO-159*	Transition Metal-Catalyzed Allylation of Aldehyde Using the Coordination Effect of Alkyne
			603
	K. Takahashi, N. Asao, Y. Yamamoto (Tohoku University, Japan)

*2-PO-160*	*Regiospecifically Substituted Oligothiophenes via* Structurally Defined Building Blocks**
			604
	F. Von Kieseritzky, J. Hellberg Asao (Royal Institute of Technology, Sweden)

B. Li, J. Xie, H. Yu, G. Xing, S. Lu, Y. Hui

C.J. Borths, W.S. Jen, J. S. Wiener, N.A. Paras, R. Wilson

G.T. Hwang, V.J. Vun, S.K. Kim Pohang University of Science and Technology, Korea

ORAL AND POSTER SESSION PROGRAM

July 30 (Mon)

Oral Presentation

D-1

C-Phosphorylation of Heteroaromatic Compounds in Synthesis of Novel Phosphorus-Containing Heterocycles

D-3

Formation of Iminosubstituted Propadienethiones by Thermal (FVP) and Electron Impact Induced Fragmentation of Multisulfur Heterocycles

July 30 (Mon)

Poster Presentation

30-PO-2

30-PO-8

July 31 (Tue)

Oral Presentation

July 31 (Tue)

Poster Presentation

August 2 (Thu)

Oral Presentation

Transfer Reagents: The Synthesis of 3,6-Di(2-Pyridyl)-Pyridazino Norbornadiene and its Use in the Synthesis of bis-dppn Ligands

472

August 2 (Thu)

Poster Presentation

2-PO-18

Synthesis and Reaction of Indolizine-1,2-dicarboxylic Anhydride

492

2-PO-20

Synthesis and Reaction of Indolo[1,2-b]indazoles

494