Monday, August
2nd
Time
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Location: Hofburg
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Opening Ceremony
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Chair: R. Castle |
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Queen's |
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The Directed ortho Metalation -
Cross Coupling Symbiosis in Heteroaromatic Synthesis |
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Chair: D. Black |
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Asymmetric
Synthesis and Synthetic Utility of 2,3-Dihydro-4-pyridones |
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Break |
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B. Stanovnik |
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Chair: J. Fröhlich |
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The University of |
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Cycloaddition
Approaches to Oxygen Heterocycles Applied to Natural Product Synthesis |
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Lunch |
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Time
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HS 1
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HS N |
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Section A M. Begtrup and T. Kappe |
Section B J. Bremner and G. Kollenz |
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M. Mori IL-1
Hokkaido University, Japan |
A. Stoller IL-2 Novartis Crop Protection AG, Switzerland |
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Synthesis of Heterocycles from
Molecular Nitrogen as Nitrogen Source |
Synthesis of New Substituted 1l4-[1,2,4,6]-Thiatriazines
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J.-H. Sun OP-1 DuPont Pharmaceuticals |
E. Skibo OP-7 |
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Practical Syntheses of Oxazolidinone Antibacterial Agents |
Development of the Pyrrolo[1,2-a]benzimidazole Antitumor Agents |
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R. Dodd OP-2
CNRS, France |
H. Szczepanski OP-8 Novartis Crop Protection AG, |
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Ortho-Metallation Studies of 5-Phenylcarboxamide Derivatives of Indole and Indoline |
A Novel Production Process for Thiamethoxam |
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G. Hoornaert OP-3 |
E. Turos OP-9 |
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A New Class of b-Lactam Antibacterials |
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Break
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Poster Session 1 (PO-1 – PO-200) P. Gärtner |
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Section A G. Bernáth |
Section B M. Potacek |
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M.
Tokuda OP-4 |
S.
Pyne OP-10 The University of |
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The Development of a Novel Immunosuppressive Agent Isolated from Caramel Colour III |
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K. Banert OP-5
Technical |
H. Kotsuki OP-11 |
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Synthesis of New Heterocycles via Unsaturated Azides |
A New Enantioselective Total Synthesis of AI-77-B |
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H. Abd El-Nabi OP-6 |
M. Yokoyama OP-12 |
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1-Aryl-5-methoxy-2,3-dihydropyrrole- 2,3-diones as Synthons for 1,3-Dipolar Cycloaddition Reactions
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Synthesis
and Biological Activity of C-Azanucleosides |
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HS 5 |
HS 6 |
Time
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Section
C J. Cavaleiro and G. Kirsch |
Section
F W. Friedrichsen and |
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G. Bernáth IL-3 Szent-Györgyi Medical Univ., |
R. Wife IL-4 SPECS and BioSPECS b.v., Netherlands |
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Finding Drug
Candidates in Virtual and Lost Chemistry |
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N. Kanomata OP-13 RIKEN, Japan |
T. Nabeshima OP-19 |
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Stereocontrol of Molecular
Jump-Rope Amplification of Planar Chirality |
Positive and Negative Allosteric
Effects on Ion Binding with a Pseudocryptand |
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F. Davis OP-14 |
H.-J. Wu OP-20 |
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Synthesis, Chemistry, and
Applications of Heterocyclic Cage Compounds |
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M. Sakamoto OP-15 |
V. Bakulev OP-21 |
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Rearrangements of
1,2,3-Thiadiazoles |
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Break
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Poster Session 1 (PO1 – PO200) P.Gärtner |
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Section
D C. Szantay |
Section
E G. Cignarella |
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B.Fischer OP-16 |
M. Oda OP-22 |
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Intertwining Synthesis, Mechanism,
and Properties of Fluorescent Adenine Nucleotides |
Synthesis and Properties of
p-Quinones Extended with 1,3-Thiazole(s) |
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O. Rusin OP-17 |
R. Glass OP-23 The |
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The novel Macrocyclic Receptors
for Saccharide Recognition |
Annulation of an Aminopyrimidine
Ring to Ferrocene |
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H. van der Deen OP-18 |
F. Ogura OP-24 |
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Synthetic Studies of a New Organic
Electron Donor: Cyclohepta[de]naphtho |
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Tuesday, August
3rd
Time
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Location: Hofburg
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Chair: M. Tisler |
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Progress in the Synthesis
of Chiral Heterocyclic Natural Products: Epothilone B and Tartrolon B |
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Chair: L. Brandsma |
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Russian
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Reactions of Unsaturated Carbanions with Isothiocyanates: a New Avenue
to Fundamental Heterocycles |
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Break |
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J. Cavaleiro Announcement of the forthcoming 19th ECHC |
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Chair: P. Stanetty |
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Lunch |
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Time
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HS
1 |
HS
N |
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Section
A W. Kantlehner and G. Queguiner |
Section
B F. Marsais and M. Yus |
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V.
Nair IL-5 Regional Research |
O.
Meth-Cohn IL-6 |
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Novel Heterocyclic Construction via Dipolar
Cycloadditions to 1,2-Dicarbonyl Compounds |
New Synthetic Methodology en Route to Asymmetric
Piperidine Alkaloids |
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C.-K. Sha OP-25 |
R. Bobrovsky OP-31 Sanochemia Pharmazeutika AG, |
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Total Synthesis of Amaryllidaceae
Alkaloids: How to Prepare |
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E. Schaumann OP-26 |
M. Ikeda OP-32 |
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Markovnikov vs. Anti-Markovnikov
Cyclization of 4-Alkenols |
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R. Kumar OP-27 |
T. Inaba OP-33 Japan Tobacco Inc., Japan |
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Sterecontrolled Electrophilic
Additions Upon 1,4-Dihydropyridines: Access to Azasugars and Alkaloids |
Catalytic Asymmetric
Aminolysis of 3,5,8-Trioxa-bicyclo[5.1.0]octane and its Application to Practical
Synthesis of Nelfinavir, an HIV Protease Inhibitor |
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Break
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Poster Session 2
(PO201 – PO400) C. Hametner |
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Section
A V.
Charushin |
Section
B Y. Thebtaranonth |
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M. Iwao OP-28 |
A. M. Almerico OP-34 Università degli Studi, Italy |
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Directed C-7 Lithiation of
1-(2,2-Diethylbutanoyl)indoles |
Pyrazolo[1,2-a]benzotetrazines with
Antitumor Activity |
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J. Podlech OP-29 Universität
Stuttgart, Germany |
T. Fukuyama OP-35 |
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Diazoketones from
a-Amino Acids: Versatile Building Blocks for
Diastereoselective
b-Lactam Synthesis |
A Novel
Synthesis of 2,3-Disubstituted Indoles |
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G. Mlostoñ OP-30 |
J. Large OP-36 |
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Reactions of some Nitrogen
Heterocycles with Sterically Crowded
a-Chloro Sulfenylchlorides |
Radical Approaches to Cyclic Amino
Acids |
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HS
5 |
HS
6 |
Time
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Section
C G. Hoornaert and H.-U. Reissig |
Section
G L. Klemm and V. Lee |
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V.
Jäger IL-7 |
I.
Ugi IL-8 |
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New
Heterocyclic Structures from Unsaturated Aldehyde Derivatives. Inhibition of
a-L-Fucosidases |
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J. Hunt OP-37 |
E. Savin OP-43 Russian |
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Application of Oxime Ethers in the
Asymmetric Synthesis of Heterocycles |
New Four-Points-Diversity Pyranes:
Synthetic and Combinatorial Aspects |
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W.-S. Chung OP-38 |
A.
Kiselyov OP-44 Amgen Inc.,
USA |
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Solid Support Synthesis of
Macrocycles and Oxazocines via the SNAr Methodology |
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T. Patonay OP-39 |
J. Vanden Eynde OP-45 |
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Stereoselective
a-Hydroxylation of Benzo(hetera)cyclanones by
Dimethyldioxirane |
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Break
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Poster Session 2
(PO-201 – PO-400) C. Hametner |
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Section
C E.-S.
El-Ashry |
Section
D |
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R. Batey OP-40 |
J. Konopelski OP-46 |
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T. Kataoka OP-41 |
N. Katagiri OP-47 Health Sciences |
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Chalcogen Heterocycles as a New
Catalyst of Baylis-Hillman Reaction |
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F. Palacios OP-42 Universidad del País Vasco, Spain |
A. Attia OP-48 National Research |
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Asymmetric Synthesis of
2H-Azirines Derived from Phosphine Oxides and Phosphonates |
Synthesis of some Cyclic
Pyridine-Carboxamides as Potential |
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Wednesday,
August 4th
Time
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Location:
Freihaus |
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Invited Lectures
IL-9 – IL-32 see next table for
the program |
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Lunch |
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Excursions: "Kahlenberg – Klosterneuburg" or ”Mödling
– Heiligenkreuz” |
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”Heuriger" |
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Time
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HS 1 |
HS N |
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Section
A1 O.
Meth-Cohn |
Section
A2 M. Bachi |
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N.
De Kimpe IL-9 |
J.
Schantl IL-15 Universität
Innsbruck, Austria |
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Synthesis of Azaheterocycles by Electrophile-induced Cyclisations of Alkenylimines |
Diazene-derived Cyclic Azomethine
Imines |
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H. Heimgartner IL-10 Universität
Zürich, Switzerland |
C. Ramsden IL-16
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Heterocyclic Chemistry using Hypervalent Reagents of Te,
I and Xe. |
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Section A1 N.
Haider |
Section A2 J.
Bergman |
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R.
Jones IL-11 The Open University, |
R.
Varma IL-17 |
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Chiral Nitrone Reagents for Cycloaddition
Reactions |
Solvent-free Synthesis of Heterocyclic
Compounds using Microwaves |
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B. Stanovnik IL-12 University of Ljubljana, Slovenia |
G.
Queguiner IL-18 IRCOF Rouen, France |
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2-Substituted 3-Dimethylamino- and
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Break
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Section A1 G. Hajos |
Section
A2 R.
Neidlein |
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R.
Prager IL-13 |
E.
Babaev IL-19 |
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Carbene versus Radical Pathways in Pyrolysis of
Benzisoxazolones and Benzotriazoles |
Fused Munchnones in Recyclization
Tandems |
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T. Shioiri IL-14
Nagoya
City Univ. Tanabedori, |
O. Attanasi IL-20 Università di Urbino, Italy |
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Silylketenes as a Useful Building Block for
Heterocycles |
Heterocyclic Systems from 1,2-Diaza-
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Lunch
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HS
5 |
HS
6 |
Time
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Section B L.
Fišera |
Section
C S.
Gronowitz |
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M.
Nakagawa IL-21 |
T.
Hudlicky IL-27 |
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Enantioselective
Total Synthesis of Marine Alkaloids, Manzamine A and Related Compounds |
Recent Progress in Efficient
Syntheses of Amaryllidaceae and Morphine Alkaloids |
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Y. Thebtaranonth IL-22 NSTDA, |
H.-U. Reißig IL-28
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Synthetic and Naturally Occuring
Antimalarials |
Stereoselective Syntheses of
Heterocycles with Lithiated Methoxyallene |
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Section
B K |
Section C D. Döpp |
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R.
Neidlein IL-23 |
C. Nájera IL-29 Universidad de Alicante, Spain |
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New Porphyrinoids – Syntheses and
Potential Photodynamic Therapeutics |
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J. Cavaleiro IL-24
University of Aveiro, Portugal |
J. Liebscher IL-30 |
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Porphyrin Derivatives: Synthesis
and Potential Applications |
Synthetic Application of Chiral
Pool Derived Heterocycles |
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Break |
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Section F G.
Heinisch |
Section D F.
Schmidtchen |
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M. Kayser IL-25 |
H.
van der Plas IL-31 |
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Designer Yeast a New Enantioselective Reagent for
Organic Synthesis |
Degenerate Ring Transformations in Heterocyclic
Systems |
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R. Neier IL-26 The University of |
J. de Mendoza IL-32 Universidad Autónoma de Madrid, Spain |
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A Novel Synthesis of
Porphobilinogen. Synthetic and Biosynthetic Studies |
Self-Assembling Cavities through
Hydrogen Bonds and Metals |
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Lunch
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Thursday, August 5th
Time
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Location:
Hofburg
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Chair: C. Moody |
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A. Padwa AL-1 |
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The Evolution of a Heterocyclic
Chemist. From Photochemistry to Alkaloids |
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Chair: S. Lang |
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T. Gallagher AL-2
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The Azomethine Ylid Strategy for
b-Lactam Synthesis
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Break |
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M. Shibasaki Announcement of the forthcoming 18th ICHC |
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Chair: M. Shibasaki |
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M. Ciufolini PL-7 Université Claude Bernard Lyon, France
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Lunch |
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Time
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HS 1 |
HS N |
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Section A S. Pyne and C.-K. Sha |
Section B J. de Mendoza and B.
Zwanenburg |
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E. Scriven IL-33
Reilly Industries, |
M.
Bachi IL-34 The Weizmann Institute of |
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Achieving Selectivity in Pyridine Synthesis |
Synthesis and Reactions of
Antimalarial Bicyclic Peroxides |
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K. Kim OP-49 |
S. Kobayashi OP-55 Sankyo Co. Ltd., |
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Trials for the Synthesis of
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N. Haider OP-50 |
W. Murphy OP-56 |
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Pyridazine Analogs of
Pyridocarbazole Alkaloids: 3‑Azaolivacine and
3-Azaellipticine
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The shortest |
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O. Chupakhin OP-51 Institute of Organic |
T.
Nakata OP-57 RIKEN,
Japan |
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Transformations of 1,2,4-Triazines
Resulting from a Nucleophilic Attack on Unsubstituted Ring Carbon |
Synthetic Studies on Marine
Polycyclic Ethers |
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Break
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Poster Session 3
(PO401 – PO579) M. Mihovilovic |
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Section A E. Babaev |
Section B A. Fahmy |
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J. Pawlas OP-52 Royal Danish |
D. Ma OP-58 Chinese |
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Facile Synthesis of New Tricyclic
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Stereoselective Synthesis of
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V. Nenajdenko OP-53 |
R. Funk OP-59 The |
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A New Synthetic Approach to
Thiophenes |
Retrocycloadditions of Substituted
Dioxins Application in Natural Product Synthesis |
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K.
Takeuchi OP-54 Eli Lilly and Company, |
N. Almstead OP-60 Procter & Gamble |
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Design, Synthesis and Biological
Evaluation of Potent Thiazepine Based MMP Inhibitors |
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Congress Banquet
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HS 5 |
HS 6 |
Time
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Section
C W. Holzer and H. Neunhoeffer |
Section
G D. Aitken and U. Jordis |
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L.
Fišera IL-35 Slovak |
P.
Hermkens IL-36 N.V. |
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Stereoselective
1,3-Dipolar Cycloadditions to Heterocyclic Compounds |
Solid Phase Organic Chemistry: How
to Come to the Best Results? |
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P.
Zimmermann OP-61 Universität
Stuttgart, Germany |
A.
Dömling OP-67 Morphochem
AG, Germany |
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Furo[2,3-d]isoxazolines - Key
Intermediates in the Synthesis of Biologically Active Compounds |
New Reactions to Heterocycles by
MCR |
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C. Lee OP-62 Research Institute of Chem. |
V. Lee OP-68 Microcide Pharmaceuticals Inc., |
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Stereocontrolled Total Syntheses
of Tetracyclic
b,d–Lactams |
Total Synthesis and Stereochemical
Elucidation of Mureidomycins and Pacidamycins |
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M. Demeunynck OP-63 Université Joseph Fourier, France |
O. Kappe OP-69 Karl-Franzens-University Graz, |
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Aminoacridines as Precursors of
New Heterocycles of Biological Interest |
Efficient Solid-Phase Synthesis of
Biofunctional 4-Aryl-3,4-Dihydro-pyrimidin-2(1H)-ones |
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Break
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Poster Session 3 (PO401 – PO579) M. Mihovilovic
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Section
C B. Stanovnik |
Section
F C. Pedersen |
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M. Natchus OP-64 Procter & Gamble |
D. Döpp OP-70 G.-Mercator-Univ. |
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Piperazine based MMP Inhibitors:
Design, Synthesis and Biological Evaluation |
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C. Santi OP-65 Università di Perugia,
Italy |
G. Yranzo OP-71 Univ. Nacional de Córdoba, Argentina |
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Synthesis of Enantiomerically Pure
Oxazolines and Thiazolines Promoted by Camphorselenenyl Sulfate |
Flash Vacuum Pyrolysis (FVP) of
Pyrazoles over Zeolites |
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T. Nishikawa OP-66 |
W. Rom OP-72 |
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Stereocontrolled Synthesis of
(-)-5,11-Dideoxytetrodotoxin |
14C Accelerator Mass Spectrometry – an
Ultrasensitive Tool for the Detection of DNA Adducts |
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Congress
Banquet |
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Friday, August 6th
Time
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Location: Auditorium Maximum
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Chair: F. Sauter |
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The
Continuing Magic of Benzotriazoles
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Chair: H. van der Plas |
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Synthetic Studies Towards Natural Products
Containing bis-Spiroacetals |
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Break |
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E.-S. El-Ashry Announcement of the forthcoming 7th ISCHC |
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Chair: C. Rees |
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Metal Promoted Synthesis of
Heterocycles from Heteroacyclic Compounds
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Closing
Ceremony |
![Synthesis of New Substituted 1l4-[1,2,4,6]-Thiatriazines](99-IL-2.jpg){kind=link}
![Development of the Pyrrolo[1,2-a]benzimidazole Antitumor Agents](99-OP-7.jpg){kind=link}
![Synthetic Studies of a New Organic Electron Donor: Cyclohepta[de]naphtho [1,8-cd]dichalcogenole](99-OP-24.jpg){kind=link}
![Pyrazolo[1,2-a]benzotetrazines with Antitumor Activity](99-OP-34.jpg){kind=link}
![Modification of Calix[4]arenes in their Upper Rims: 1,3-Dipolar Cycloaddition Reactions of Benzonitrile Oxides with Mono- and A,C-Diallylcalix[4]arenes](99-OP-38.jpg){kind=link}
![Furo[2,3-d]isoxazolines - Key Intermediates in the Synthesis of Biologically Active Compounds](99-OP-61.jpg){kind=link}
