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SCIENTIFIC PROGRAM |
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August 7, Monday |
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Opening
Ceremony |
Hall, TICC |
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PLENARY LECTURES
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August 7, Monday
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Hall, TICC
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Chairman:
J Bergman |
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PL-1 |
R.
Noyori, |
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Chairman:
T -S. Chou |
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PL-2 |
C.-H.
Wong, The Scripps Research Institute, U.S.A |
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INVITED
LECTURES
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August 7, Monday
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201BC, TICC
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Session
Ia: Organic Synthesis in Heterocyclic Chemistry
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Chairman: |
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J.
Barluenga, Universidad de Oviedo, Spain |
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IL-Ia-1 |
Synthesis
of Heterocycles Mediated by Metal and Metalloid Species |
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M. D. Bachi, A Melman, The Weizmann Institute
of |
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IL-Ia-2 |
Stereocontrolled Synthesis of
(±)-Kainic Acid Based on Free-Radical Key Reactions |
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August 7, Monday
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101B, TICC
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Session
Ib: Organic Synthesis in Heterocyclic Chemistry
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Chairman: K. -T
Liu |
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Y.
Thebtaranonth, |
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IL-Ib-1 |
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H. N. C.
Wong, The Chinese |
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IL-Ib-2 |
Regiospecific
Synthesis of Polysubstituted Furans, Thiophenes and Pyrroles |
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August 7, Monday
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201DE, TICC
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Session
II: Asymmetry and Heterocycles
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Chairman: T-K. Yang |
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F.
Effenberger, |
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IL-II-1 |
Enzyme
Catalyzed Preparation of Chiral Educts for the Synthesis of Optically Active
Heterocycles |
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J.
Campbell, B. Filippini, D. J. Hart, S. Lacoutiere, The |
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IL-II-2
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New Syntheses of Functionalized Perhydroisoquinolines and
Perhydroindoles
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August 7, Monday
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101A, TICC
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Session
III: Heterocyclic Pharmaceuticals and Agrochemicals
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Chairman:
Y Kita |
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P. N. Confalone, L. Anzalone, G. Harris, P. K.
Jadhav, R Kaltenbach, P. Y. S. Lam, Y. S. Lo, L. Radesca, J.
D. Rodgers, L. T. Rossano, S. P. Seitz, T. E. Smyser, R. E. Waltermire, The
DuPont Merck Pharmaceutical Co., U.S.A |
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IL-III-1 |
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The
Synthesis of Cyclic Urea Diols as Inhibitors of HIV Protease |
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Y.-I. Lin, P Bitha, S. M. Sakya, T. W. Strohmeyer, Z.
Li, V. J. Lee, S. A Lang, Jr., K. Bush, R. T. Testa, Wyeth-Ayerst Research, U.S.A
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IL-III-2
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August 7, Monday
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103, TICC
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Session
VI: New Heterocyclic Materials
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Chairman:
C. T. Pedersen |
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T. Shimidzu, |
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IL-VI-1 |
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M. Hanack, Universität Tubingen, Germany |
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IL-VI-2
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Phthalocyaninato
Transition Metal Coordination Polymers and Their Applications in Materials Design |
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ORAL PRESENTATIONS
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August 7, Monday
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201BC, TICC
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Session
Ia: Organic Synthesis in Heterocyclic Chemistry
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Chairman:
L. F. Tietze |
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F.
Beaulieu, P. Moreau, O. B. Familoni, L Ionica, M. Gray, J. A Glanzer, V.
Snieckus, |
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OP-Ia-1 |
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M. Regitz, |
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OP-Ia-2 |
Azacyclobutadienes - Remarkable
Building Blocks in Heterocyclic Synthesis |
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W.
Eberbach, E. Lopez-Calle, |
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OP-Ia-3 |
Studies
on the Reactivity of 4-Oxazolines: The Photochemical Route to Azomethine
Ylides |
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16:20
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T. Kitamura, M.-a. Miyaji, S.-i.
Soda, H. Taniguchi, Kyushu University, Japan |
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OP-Ia-4 |
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C. O.
Kappe, J. E. Cochran, A Padwa, |
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OP-Ia-5 |
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August 7, Monday
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101H, TICC
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Session
Ib: Organic Synthesis in Heterocyclic Chemistry
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Chairman: V Sipido |
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D. E. Justice, J. R. Malpass,
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OP-Ib-1 |
Synthesis of Natural Epoxytropanes
and Novel Non-Natural Analogues and Homologues |
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T. Toda, M. Karikomi, M. Watanabe, |
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OP-Ib-2 |
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K. Vijayakumaran, Chimique Laboratories ( |
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OP-Ib-3 |
Enolate Formation in
Tetrahydropyran-3-ones. Regioselectivity and Directing Effect of Ring Oxygen |
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M
Nakagawa, Y. Torisawa, Y. Koide, M. Arisawa, T. Rino, |
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OP-Ib-4 |
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J.-S.
Pan, D.-D. Hsiao, Y.-M. Tsai, |
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OP-Ib-5 |
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August 7, Monday
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201DE, TICC
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Session
II: Asymmetry and Heterocycles
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Chairman: W Pearson |
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T.
Kercher, T. Livinghouse, |
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OP-II-1 |
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E. Wada, U.
Chin, H. Kawamoto, H. Yasuoka, S. Kanemasa, Kyushu University, Japan |
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OP-II-2 |
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B. Zwanenburg, L.
Gentilucci, L. Thijs, G. J. A. Ariaans, M. M. H. Verstappen, |
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OP-II-3 |
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M. Ikeda, H. Ishibashi, |
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OP-II-4 |
Asymmetric Synthesis of
b-Lactams by Radical Cyclization of N-Vinylic
α- Haloacetamides |
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D. Ma, J. Ma, W. Ding, Chinese |
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OP-II-5 |
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August 7, Monday
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101A, TICC
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Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
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Chairman:
D. |
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J.-H.
Sun, R. F. Kaltenbach, M. R. Kirshenbaum, L. M. Papp, M. P. Stafford, R
J. McRipley, P. M. Czemiak, R J. Diamond, J. L. Miller, R J. Page, S.-P.
Chen, D. L. Dexter, J. L. Gross, C. H. Behrens, S. P. Seitz, The DuPont Merck
Pharmaceutical Company, |
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OP-III-1 |
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M.
Daneshtalab, D. Q. Nguyen, A. B. Oreski, R G. Micetich, SynPhar
Laboratories Inc., |
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OP-III-2 |
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H.-Y.
Mei, M. Cui, A. A. Galan, N. S. Halim, D. P. Mack, D. W. Moreland, K. B.
Sanders, H. N. Truong, A. W. Czarnik, Warner-Lambert Company, |
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OP-III-3 |
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Inhibition
of an HIV-1 Tat-Derived Peptide Binding to TAR RNA by Aminoglycoside Antibiotics |
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16:20 |
A. M. Almerico, G. Cirrincione, F.
Mingoia, S. Grimaudo, P. Diana, P. Barraja, G. Dattolo, E. Aiello, A. G. Loi,
P. La Colla, Università degli Studi, Italy |
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OP-III-4 |
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Glycosidopyrroles
and Related Acyclic Derivatives as Potential Antiviral and Anticancer Agents |
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A.
Gutcait, H-W. Liu, J.-W. Chern, |
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OP-III-5 |
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August 7, Monday
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103, TICC
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Session
VI: New Heterocyclic Materials
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Chairman: A. B.
Holmes |
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R. A.
Aitken, L. Hill, |
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OP-VI-1 |
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R. Gompper, A. Ehmann, H.
Engel, J. Einsiedler, O. Freundel, H.-J. Mair, W. Sammer, C. Schnock,
University of München, Germany |
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OP-VI-2 |
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H.-H. Horhold, A. Lux, F. Leonhardt, R Stockmann,
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OP-VI-3 |
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F.
Ogura, Y. Shibata, A. Kashihara, K. Takimiya, Y. Aso, T.
Otsubo, Kinki University, Japan |
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OP-VI-4 |
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POSTER SESSION I
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August 7, Monday
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201AF, TICC
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PO1-001 |
V. A. Alfonsov, G. S. Stepanov, D. A. Pudovik,
I. A. Litvinov, O. N. Kataeva, Russian |
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Heterocyclization
of
b-Oxyethylamide
of 5-Methoxyindolyl-2-carbonic Acid |
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PO1-002 |
H.
Kiljunen, K. Wähälä, T. A. Hase, |
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PO1-003 |
C.-H. Yang, H.-J. Shen,
S.-J. Chen, R-S. Wang, |
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2,3,7-Triazabicyclo[3.3.0]octenes,
Their Syntheses, Chemical Properties and Applications |
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PO1-004 |
T.
Kataoka, T. Iwama, |
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Selective
C-S Bond Cleavage of 1,2-Thiazetidine 1,1-Dioxides by Lewis Acids |
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PO1-005 |
H. Togo, T. Muraki, M.
Yokoyama, Chiba University, Japan |
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Use of
(Diacyloxyiodo)benzene for Organic Synthesis: Lactones and Cyclic Ethers |
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PO1-006 |
Y.
Murakami, T. Watanabe, |
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PO1-007 |
B. I.
Drevko, M. L Smoushkin, L A. Fomenko, O. L Zhukov, V. G.
Kharchenko, The |
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PO1-008 |
K.
Dikovskaya, T. Mazure, L Turovskis, M. Gavars, J. Freimanis,
Latvian Institute of Organic |
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Synthesis
of Bicyclic
b-Oxyaminovinyl
and
b-Oxavinyl
Lactones |
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PO1-009 |
L.-W. Chuang, L-C. Row,
M.-C. P. Yeh, |
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Synthesis
of N-Containing Heterobicyclic and -tricyclic Skeletons Mediated by Irontricarbonyls |
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PO1-010 |
I. L.
Yudin, A. B. Sheremetev, Russian |
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Diagonally
Substituted Pyrazines Based on 2,5-Dioxopiperazine |
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PO1-011 |
M. Iwao, O. Motoi, |
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Methodology for the Highly
Efficient Synthesis of 3,4-Differentially Substituted Indoles |
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PO1-012 |
L.
Ferris, C. J. Moody, D. Haigh, |
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PO1-013 |
M. El-Ghanam, |
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Synthesis, Reactions and Spectral Properties of
3-Chloro-2,6-diaryltetrahydro-4H-thiopyran-4-ones |
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PO1-014 |
R. F.
Ambartsumova, L P. Kosmacheva, Academy Science |
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PO1-015 |
M.-K.
Hu, D. H. Rich, |
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Design
and Synthesis of Suitable Precursors for Photoaffinity Labeling of Cyclosporin
A |
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PO1-016 |
V. M.
Berestovitskaya, |
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The
Problem of Regioselectivity in the Chemistry of Nitrothiolene-l,l-dioxides |
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PO1-017 |
I. E. Eftemova, V. M. Berestovitskaya, E. V. Trukhin, G. A.
Berkova, State Pedagogical
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Allyl-Vinylic Isomerization in the
Series of Nitro Group Containing Thiolene-l,1-dioxides |
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PO1-018 |
A. P. Halverson, R. N. Castle, L.
W. Castle, |
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PO1-019 |
J.-K.
Luo, R. F. Federspiel, R. N. Castle, |
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PO1-020 |
O.
Tsuge, T. Hatta, M. Kuwata, Kumamoto Institute of |
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PO1-021 |
Q. Chen, T. Jian, |
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PO1-022 |
Q. Chen, Z.
Wang, |
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Photocatalysed Additions of Cyclic
Amines to 5-Alkoxy-2-(5H)-furanones |
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PO1-023 |
M. Yeung, B. Fraser-Reid, H. D.
Banks, U. S. Army, Edgewood Research, U.S.A. |
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Novel Approach to a Potent
Synthetic Opioid by Means of an Aza-Claisen Rearrangement |
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PO1-024 |
A. P. Fonseca, A. M. Lobo, S. Prabhakar,
Sintor-Vninova, Portugal |
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PO1-025 |
V. Brovarets, R. Vydzhak, K. Ziouz, E.
Romanenko, B. Drach, National Academy of Sciences of the |
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PO1-026 |
M. Kiyoshi, |
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Reactions of 3a,6a-Diazapentalenes
with Dimethyl Acetylenedicarboxylate: Formation of 1:2 Adduct |
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PO1-027 |
A. M. F.
Oliveira-Campos, M. M. M. Raposo, P. V. R. Shannon, Universidade do
Minho, Portugal |
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Synthesis
of Cyanocarbazoles Precursors of Anti-Cancer Ellipticines |
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PO1-028 |
S. P. G.
Costa, M. M. Oliveira, A. M. F. Oliveira-Campos, M. J.R. P. Queiroz,
J. Seita, Universidade do Minho, Portugal |
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Light
Sensitive Compounds Derived from Carbazoles and Indoles |
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PO1-029 |
Y.-H. Chen, T.-Y. Luh, |
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PO1-030 |
S. R.
Fletcher, M. S. Chambers, S. C. Hobbs, L. A. McNeill, Merck,
Sharp and Dohme Research Laboratories, |
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Epibatidine
and Analogues: Unexpected Formation of exo-7-Methyl-7-azabicyclo[2.2.1]heptan-2-ol |
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PO1-031 |
T. Okano, T Sakaida, S. Eguchi,
Nagoya University, Japan |
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Synthesis
of Trifluoromethyl-Group-Containing Fused Nitrogen-Heterocycles |
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PO1-032 |
B. M.
Ginzburg, V. I. Kovalenko, V. V. Nurgatin, |
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PO1-033 |
V. I.
Kovalenko, L. V. Anisimova, V. L. Furer, Kazan State
Technology University, |
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The
Interpreted Vibrational Spectra of 1,2,5-Oxadiazole N-Oxyde |
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PO1-034 |
V. Murugesan, A. Pandurangan, Anna University, India |
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Heterocyclic Halochromates: Mild
but Potential Oxidants in Organic Synthesis |
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PO1-035 |
Y. Terao, |
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PO1-036 |
T. J. Chow, J.-J. Hwang, |
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On the Iron-Promoted Deamination
Reactions of N-Substituted 7- Azanorbornadiene Derivatives |
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PO1-037 |
T.
Choshi, S. Yamada, E. Sugino, T. Kuwada, S. Hibino, Fukuyama
University, Japan |
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PO1-038 |
S. K. Dewan, S. D. Malik,
Maharshi Dayanand Univeristy, |
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Clay-Mediated
Synthesis of Enamines from Acyclic Ketones and Secondary Cyclic Amines |
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PO1-039 |
M. K. Mao, R. K. Webber,
Monsanto Co., U.S.A. |
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PO1-040 |
T. K. O'Leary, R. W. Read,
The |
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Selectivity in the Synthesis of
Substituted 1,3,6,8- Tetraazadecalins |
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PO1-041 |
K.
Vijayakumaran, T. Balasubramanian, Chimique Laboratories ( |
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Efficient
Oxidation of Alcohols Using Imidazolium Dichromate under Heterogeneous
Conditions |
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PO1-042 |
W. Tian, J. Li,
Chinese |
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PO1-043 |
S.
Kaban, Z. Turgut, N. Öcal, |
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PO1-044 |
G. N. Lipunova, G. A. Mokrushina, O. M.
Chasovskikh, E. V. Granovskaya, V. N. Charushin, Ural |
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Cyclizations of
3-Hetarylhydrazino-2-polyfluorobenzoyl Substituted Ethyl Acrylates |
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PO1-045 |
P. Stanetty, M. D. Mihovilovic,
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PO1-046 |
P.
Stanetty, B. Krumpak, M. D. Mihovilovic, |
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PO1-047 |
P. Stanetty, M. Kremslehner, M. D.
Mihovilovic, |
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Synthesis of Annelated
1,2,3-Thiadiazoles via the Hurd-Mori-Reaction |
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PO1-048 |
Y. Chang, S.-C.
Lin, F.-D. Yang, J.-M. Fang, |
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PO1-049 |
I. I.
Ismail, A. H. Abd El-Aleem, A. Abdel-Megied, H. Abd
El-Bary, National Research |
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Reactions
with Sultones IV,
synthesis of 1,3,4-Oxadiazolyl and 1,3,4-Triazolyl Sultam
Derivatives |
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PO1-050 |
I.
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PO1-051 |
Y.
Kitahara, F. Tamura, S. Watanabe, H. Onikura, A. Kubo, |
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Synthesis
of Polycyclic Aromatic Marine Alkaloids Possessing Iminoquinolinequinone Structure |
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PO1-052
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T.
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Synthesis
of 1,2-Dihydro-2-allylindol-3-ones Using in situ Claisen Rearrangement
of 1,2-Dihydroindol-3-ones with Allyl Alcohols |
|
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PO1-053 |
M.
Kotera, K. Ishii, O. Tamura, M. Sakamoto, |
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1,3-Dipolar
Cydoadditions of Photoinduced Carbonyl Ylides from α,b-Unsaturated
γ,δ‑Epoxy Dinitriles |
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PO1-054 |
S.-J. Shieh, J.-S. Lie,
T-C. Tarny, R.-S Liu, |
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Preparation
of Five-Membered Oxygented Compounds by Tungsten-Promoted Intramolecular
Cyclization |
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PO1-055 |
M. P.
Meyyappan, C. S. Venkatachalam, K. K. Balasubramanian, Intran
Institute of |
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PO1-056 |
M. A. J.
Miah, M. Tsukazaki, M. Wicki, T Nguyen, M. Kerr, V. Snieckus, |
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PO1-057 |
V. Snieckus, M. Campbell, |
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Preparation and Complexation
Studies of Macrocydic Hosts for the Complexation of Aromatic Pollutants |
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PO1-058 |
M. Komatsu, S. Minakata, I. Ryu,
Y. Ohshiro, Osaka University, Japan |
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Novel
Generation of Azomethine Ylide by Fluorosilylation of Azaallyl Anion |
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PO1-059 |
T. Konoike, Y. Kanda, Y. Araki, Shionogi & Co., Ltd.,
Japan |
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Ortho-Directed Metalation of
Isoxazole: Synthesis of 4-Substituted Aminoisoxazoles |
|
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PO1-060 |
Y.-L. Liu, G.-H. Hsiue, Y.-S. Chili, |
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Ring Opening Reaction of Oxetane
Rings: Polymerization and Polymer Modification |
|
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PO1-061 |
D.
Prajapati, J. S. Sandhu, A. C. Ghosh, Regional Research |
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PO1-062 |
F. Fülop, L.
Lázár, G. Bernáth, F. G. Riddell, |
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Synthesis and
Characterization of Multicomponent Ring-Chain Tautomeric Mixture |
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PO1-063 |
E.
Gudriniece, M. Jure, A. Gutcait, S. Belyakov, |
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Condensed
Systems of Pyridine from Fluorinated 1,3-Diketones |
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PO1-064 |
E. Gudriniece, M. Jure,
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PO1-065 |
R. Martinez, E. Angeles, F. Martinez,
Universidad Nacional Autónoma de México, México |
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PO1-066 |
F. Fülöp, H. Warnhoff, P. Sohár, |
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PO1-067 |
C.-K.
Sha, T.-S. Jean, N.-T. |
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Synthesis
of Heterocyclic and Carbocyclic Structures by Radical Cyclization |
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PO1-068 |
H. R.
Kim, E. K. Ryu, Korea Research Institute of Chemical |
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PO1-069 |
K. Tanaka, Y. Shogase, H.
Osuga, H. Suzuki, K. Nakamura, Kyoto University, Japan |
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PO1-070 |
R.-S. Liu, K.-W. Liang, |
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PO1-071 |
A. Lightfoot, C. J. Moody, P. T.
Gallagher, Loughborough |
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PO1-072 |
M. N.
Preobrazhenskaya, E. I. Lazhko, A. M. Korolev, |
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PO1-073 |
C. W. Jefford, D. Misra, A. P.
Dishington, J. C. Rossier, G. Bernardinelli, G. Timari, Hungarian
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Asymmetric
Dihydroxylation of cis-Fused Cyclopentano-1,2,4-trioxanes |
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PO1-074 |
Y. Yuasa, J.
Ando, S. Shibuya, Tokyo University of Pharmacy & Life Science, Japan |
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|
|
Enantioseletive
Synthesis of Pyrrolidine and Piperidine Derivatives by Radical Cyclization |
|
|||
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PO1-075 |
H.
Ishibashi, C. Kameoka, K. Kodama, M. Ikeda, |
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|
Radical
Cyclization Approach to a Chiral 1b-Methylcarbapenem
Key Intermediate |
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PO1-076 |
Y. Aoyagi, A. Ohta, |
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PO1-077 |
G. Galley, M. Pätzel,
Humboldt-Universität zu Berlin, Germany |
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PO1-078 |
J. Uenishi, S.
Hata, T. Hiraoka, K. Nakamura, S. Oae, O. Yonemitsu, |
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Preparation
of Optically Active Pyridines and Oligopyridines |
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PO1-079 |
N. N. Romanova, V. V. Dunina, Moscow State University, Russia |
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PO1-080 |
H. Waldmann, G.
Schmidt, A. Flohr, E. BHiser, R. Lock, M. Braun, Universität Karisruhe,
Germany |
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PO1-081 |
S. Bausch, P.
H. Laur, A. Scharsich, S. Vonderbank, PWTH Aachen University of Technology,
Germany |
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|
Preparation
and Stereochemistry of Some Novel Cyclic Organic Esters of Selenic and
Telluric Acids |
|
|||
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|
PO1-082 |
R. N.
Yadava, N. Jain, Dr. |
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|
|
Isolation
and Characterization of a New Steroidal Glycoside from Setaria Italica |
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PO1-083 |
C.-C.
Han, R.-C. Jeng, |
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PO1-084 |
V. F.
Ivanov, A. A. Nekrasov, O. L. Gribkova, A. V. Vannikov, A.
N. Frumkin, Russian Academy of Sciences, Russia |
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PO1-085 |
Y.-X. Lou, Q. Wu, J.-S. Bao,
Z.- T. Huang, Academia Sinica, China |
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PO1-086 |
A. B.
Sheremetev, V. O. Kulagina, E. A. Ivanova, Russian Academy of
Sciences, Russia |
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|
|
Zoro-Hydrogen
Furazan-Macrocycles with Oxy and Diazo Bridges |
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PO1-087 |
R. N. Warrener, M. A. Houghton, S. Wang, |
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PO1-088 |
J.-J.
Chen, I.-L. Tsai, W.-S. Sheen, I.-S. Chen, |
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PO1-089 |
J W
Brown, D. T. Hurst, J. P. O'Donovan, |
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|
|
The
Synthesis of Some Alkoxy(aryl)pyrazines and Aryl-pyrazinyl Esters as Heterocyclic
Mesogens |
|
|||
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|
PO1-090 |
V. Efimov, M. Makova, Russian |
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|
|
Influence of Superconductor
Transition on Kinetic Coefficients of k-(ET)2CU[N(CN)2]Br
(k-Br) |
|
|||
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|
PO1-091 |
W.-L.
Chia, S.-P. Tzeng, Fu |
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|
PO1-092 |
T. V.
Vernitskaya, O. N. Efimov, Russian |
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|
||
|
|
Synthesis
of Polypyrrole Films in the Presence of FeCl4- and
PolymolybdateAnions |
|
|||
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|
PO1-093 |
N. G.
Spitsina, V. N. Semkin, A. Graja, Russian Academy of
Sciences, Russia |
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Single
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PO1-094 |
T. L.
Tong, J.-i. Tanaka, T. Higa, K. Suwanborirux, University of the Ryukyus, |
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|
PO1-095 |
J.
Tamaki, J.-i. Tanaka, T. Higa, University of the Ryukyus, |
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|
||
|
|
Unusual Reactions of the Sulfinyl Indoles Isolated from the Seaweed Laurencia Brongniartii |
|
|||
|
PO1-096 |
C.-L.
Wang, Taiwan Forestry Research Institute |
|
|
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|
|
Investigation
on the Stability and Tocopherol, Sterol Compositions of Oiltea's Oil |
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|
PO1-097 |
S. Ya. Melnik, A. A. Bakhmedova, L.
V. Ektova, L. D. Garaeva, T. D. Miniker, I. L. Plikhtyak, I. V. Yartseva,
Cancer Research Center, Russia |
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|
PO1-098 |
D.-F.
Tai, C.-T. Lai, L.-C. Chiu, Da-Yeh Institute of |
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|
||
|
|
Alcalase
Catalyzed Esterification of N-Protected Amino Acids with Secondary Alcohols |
|
|||
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|
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|
PO1-099 |
R. S. Wu, M. Ghoshal,
L. Liu-Allison, K. Schwenzer, Roche Diagnostic Systems, U.S.A. |
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|
||
|
|
Synthesis
and Evaluation of 6-Hydroxycinchonine Derivatives by Fluorescence Polarization |
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|
PO1-100 |
D.-H.
Chin, M.-C. Tseng, National Changhua |
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|
|
Abnormal
Cycloaromatization of Neocarzinostatin Chromophore in Holoprotein Induced by
Sugar Thiols |
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PO1-101 |
J. Ohkanda, A. Katoh, Seikei University, Japan |
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|
PO1-102 |
H.-M. Yu, S.-T.
Chen, C.-L Ho, H.-P. Juan, K.- T. Wang, Academia |
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PO1-103 |
W. Hübsch, BAYER AG, Pharma-Research, Germany |
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|
|
Reactions of Sterically Hindered
Phenoles with Pyridine and Trifluoromethane-sulfonic Anhydride |
|
|||
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|
PO1-104 |
H.-W. Huang, K.-T. Wang,
Academia Sinica, Taiwan, R.O.C. |
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|
PO1-105 |
E.
Lukevics, J. Popelis, O. Pudova, Latvian Institute of Organic |
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||
|
|
Nucleophilic
Reactions of Silyl Substituted Thiophene-1,1-dioxides |
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||
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|
PO1-106 |
L-C
Chen, H.-M. Wang, |
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||
|
|
Palladium-Catalyzed
Synthesis of Carbazoles and
b-Carbolines |
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||
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|
PO1-107 |
S.-S. P.
Chou, Y.-J. Yu, Fu |
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|
|
Intramolecular
l,3-Dipolar Cycloaddition of Sulfur-Substituted l,3-Dienes with Nitrones |
|
|||
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|
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|
PO1-108 |
V.
A. Makarov, N. P. Solov'eva, O. S. Anisimova, Centre for Drug Chemistry, Russia |
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PO1-109 |
M. Watanabe, Y. Matsumura, |
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|
PO1-110 |
C. J.
Moody, D. A. Riddick, |
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|
||
|
|
A Novel
Double Diels-Alder Reaction as a Route to Annelated Bipyridyls |
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|
||
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|
||||
|
August 8, Tuesday
|
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|
|||
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|
|||
|
PLENARY
LECTURES
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|
|||
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|
|||
|
August 8, Tuesday
|
101, TICC
|
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||
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|
|||
|
|
Chairman: H. van der Plas |
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|
||
|
PL-3 |
E. Vogel, |
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|||
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|
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|
|
Chairman: A. Dondoni |
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|
||
|
PL-4 |
K. Mori, Science |
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||
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|
|||
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|
||||
|
INVITED LECTURES
|
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|
|||
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|
|||
|
August 8, Tuesday
|
101, TICC
|
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|
||
|
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|
|||
|
Session
Ia: Organic Synthesis in Heterocyclic Chemistry
|
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|
|||
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|
|||
|
|
Chairman: S-S Chou |
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|
||
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|
|||
|
|
J.-M.
Fang, |
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|
||
|
IL-Ia-3 |
Samarium(II)
lodide Promoted Coupling Reactions of Aromatic and Carbonyl Compounds |
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|
||
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|
|||
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|
|||
|
|
M.
Lautens, |
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|
||
|
IL-Ia-4 |
Synthetic
Approaches to Polycyclic Compounds via Heterocyclic Intermediates |
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|
||
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|
||||
|
August 8, Tuesday
|
102, TICC
|
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|
||
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|
|||
|
Session
II: Asymmetry and Heterocycles
|
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|
|||
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|
|||
|
|
Chairman: H.-J Liu |
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|
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|||
|
|
H. Hiemstra, |
|
|
||
|
IL-II-3 |
Synthetic Applications of
Enantiopure, Heterocyclic, Highly Electrophilic Iminium Intermediates |
|
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||
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|
|
D. H. Kim, |
|
|
||
|
IL-II-4 |
|
|
|||
|
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|
||||
|
August 8, Tuesday
|
201BC, TICC
|
|
|
||
|
|
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|
|||
|
Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
|
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|
|||
|
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|
|||
|
|
Chairman: M Regitz |
|
|
||
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|
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|
|
N. De
Kimpe, M. Boelens, |
|
|
||
|
IL-III-3 |
New
Synthesis of Azaheterocycles by Electrophile-Induced Cyclizations |
|
|
||
|
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|
|||
|
|
G.-Q. Lin, Shanghai Institute of |
|
|
||
|
IL-III-4 |
Two Useful Synthons for the
Synthesis of the Homochiral Heterocyclic Compounds |
|
|
||
|
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||||
|
August 8, Tuesday
|
103, TICC
|
|
|
||
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|
|||
|
Session
VI: New Heterocyclic Materials
|
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|
|||
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|
|
Chairman: M Banwell |
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||
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|
|
B. Ganem, |
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||
|
IL-IV-1 |
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|
|
D. S.
Black, M. C. Bowyer, A. J. Ivory, N. Kumar, D. B. McConnell, The University
of |
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|
IL-IV-2 |
|
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||||
|
August 8, Tuesday
|
201DE, TICC
|
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|
Session
VI: New Heterocyclic Materials
|
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|||
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|||
|
|
Chairman:
R. Gompper |
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|
|
R. L.
Elsenbaumer, H. Cheng, Y. Fu, The |
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IL-VI-3 |
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||||
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|
11:30 |
A. B. Holmes, X.-C. Li, S. C. Moratti, K.A.
Murray, T.-M. Yong, F. Cacialli, J. Grüner, R H. Friend, |
|
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|
IL-VI-4 |
|
|
|||
|
|
Applications
of Conjugated Heteroaromatic Polymers in Light Emitting Devices |
|
|
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|
||||
|
ORAL
PRESENTATIONS
|
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|||
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|||
|
August 8, Tuesday
|
101, TICC
|
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||
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|
|||
|
Session
Ia: Organic Synthesis in Heterocyclic Chemistry
|
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|||
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|||
|
|
Chairman:
R. Glass |
|
|
||
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|||
|
|
R Neidlein, M.
Bergemann, H.G. Krug, M. Jochheim, Universität Heidelberg, Germany |
|
|
||
|
OP-Ia-6 |
Isocyano-acetonitril
and Derivatives New Potential Synthons for Syntheses of Heterocycles |
|
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|||
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|||
|
|
D.
Cartwright, J. R. Ferguson, T. Giannopoulos, G. Varvounis, B.
J. Wakefield, |
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|
OP-Ia-7 |
|
|
|||
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|
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|
|||
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|
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|
|
U. Zoller, Haifa Univerisity-Oranim, Israel |
|
|
||
|
OP-Ia-8 |
In Pursuit of Stable, Strained
Three-Membered Ring Sulfur Heterocycles |
|
|
||
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|
|||
|
|
B.
Stanovnik, J. Svete, A. Hvala, J. Smodis, M, Kmetic, L.
Kralj, L. Selic, G. Sorsak, S. Strah, R. Toplak, |
|
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|
OP-Ia-9 |
|
|
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|
||||
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|
|||
|
|
K. K. Balasubramanian, G. Bhavani, Indian Institute of |
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|
||
|
OP-Ia-10 |
|
|
|||
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|
|||
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|
|||
|
|
S. Ostrowski, Polish |
|
|
||
|
OP-Ia-11 |
New
Approach to Fused Pyrirnidine Derivatives. Synthesis of Purines. |
|
|
||
|
|
|
||||
|
August 8, Tuesday
|
201DE, TICC
|
|
|
||
|
|
|
|
|||
|
Session
Ib: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
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|
|||
|
|
Chairman: J Barluenga |
|
|
||
|
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|
|||
|
|
R. H.
Prager, J. Smith, B. Weber, C. M. Williams, |
|
|
||
|
OP-Ib-6 |
Heterocyclic
Synthesis by Photolysis or Pyrolysis of Isoxazol-5-ones |
|
|
||
|
|
|
|
|||
|
|
S.
Eguchi, Y. Yu, M. Ohno, |
|
|
||
|
OP-Ib-7 |
Synthesis
of Homoadamantane-Fused Nitrogen Heterocycles Based on Nitrone Cycloadditions |
|
|
||
|
|
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|
|||
|
|
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|
|||
|
|
L. Abmann, T. Debaerdemaeker, O. Peters, C.
Pli.ig, S. Reck, W. Friedrichsen |
|
|
||
|
OP-Ib-8 |
|
|
|||
|
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|
||||
|
|
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|
|||
|
|
L.
Strekowski, S.-Y.
Lin, A. S. Kiselyov, R. L. Wydra, J. Nguyen, N. P. Redmore, J. C. Mason,
|
|
|
||
|
OP-Ib-9
|
|
|
|||
|
|
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|
|||
|
|
|
|
|||
|
|
G.
Himbert, O. Gerulat, E. Pierron, |
|
|
||
|
OP-Ib-10 |
Five
Membered Betaines from the Reaction of(1-Alkynyl)hydrazines with Aryl Isocyanates |
|
|||
|
|
|
|
|||
|
|
J. Reiter, J. Reiter
Jr., J. Brlik, EGIS Pharmaceuticals, Hungary |
|
|
||
|
OP-Ib-11 |
Synthesis,
Alkylation and Rearrangements of Triazolo[1,5-a]pyrimidin-5-one Oximes |
|
|
||
|
|
|
||||
|
August 8, Tuesday
|
102, TICC
|
|
|
||
|
|
|
|
|||
|
Session
II: Asymmetry and Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: R. A. Aitken |
|
|
||
|
|
|
|
|||
|
|
Y. Kita, H. Fujioka,
|
|
|
||
|
OP-II-6 |
|
|
|||
|
|
|
|
|||
|
|
J. Liebscher, A. Bartels,
J. Bohrisch, M. Patzel, H. Faltz, W. Wohlauf, Humboldt-University Berlin,
Germany |
|
|
||
|
OP-II-7 |
|
|
|||
|
|
Synthesis
of Functionalized Alkylheterocycles by Asymmetric Michael-Like Additions |
|
|||
|
|
|
|
|||
|
|
M. Somei, K.
Nakagawa, F. Yamada, S. Hamamoto, |
|
|
||
|
OP-II-8
|
The First and Simple Total Syntheses of Ergot Alkaloids,
(-)- Isochanoclavine-I and (-)-Agro-Clavine, and
Their (+)-Enantiomers
|
|
|
||
|
|
|
|
|||
|
|
I.-q. Wang, W.-s. Tian,
Chinese |
|
|
||
|
OP-II-9 |
|
||||
|
|
|
|
|||
|
15:20
|
T.
Benincori, E. Brenna, F. Sannicolò, L. Trimarco, P. Antognazza, E.
Cesarotti, T. Filati, Dip. Chimica Organica e Industriale, Italy |
|
|
||
|
OP-II-10 |
|
|
|||
|
|
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|
|||
|
|
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|
|||
|
|
J. S.
Yadav, Indian Institute of Chemical |
|
|
||
|
OP-II-11 |
|
|
|||
|
|
|
||||
|
August 8, Tuesday
|
201BC, TICC
|
|
|
||
|
|
|
|
|||
|
Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: C. O-Yang |
|
|
||
|
|
|
|
|||
|
|
M. G.
Banwell, B. D. Bissett, C. T. Bui, G. W. Simpson, The
Australian National |
|
|
||
|
OP-III-6 |
|
|
|||
|
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|
|||
|
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|
|||
|
|
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|
|||
|
|
C.-K.
Chen, T. Arunachalam, E. Delaney, P. deMena, R. Deshpande, J. Grosso, O.
Hass, G. Kodersha, D. Lust, E. Marinelli, M. Miller, K. Natalie, S. Prasad, R.
Ranganathan, T. Sedergran, A. Singh, N. Soundararjan, K. Tse, Bristol-Myers
Squibb, U.S.A. |
|
|
||
|
OP-III-7 |
|
||||
|
|
Process
Development for the Synthesis of Iopiperidol:A Non-Ionic Contrast Agent |
|
|
||
|
|
|
|
|||
|
|
H. Szczepanski, Ciba-Geigy
AG, Switzerland |
|
|
||
|
OP-III-8 |
|
|
|||
|
|
|
|
|||
|
|
K.-C. Lin, D. P. Getman, M. Clare, Biogen
Inc., |
|
|
||
|
OP-III-9 |
The Syntheses of the Two Key
Cyclic Epoxides for the Syntheses of the Cyclic HIV Protease Inhibitors |
|
|
||
|
|
|
|
|||
|
|
|
|
|
||
|
OP-III-10 |
|
||||
|
|
|
||||
|
|
|
|
|||
|
|
G. W.
Rewcastle, A. M. Thompson, B. D. Palmer, W. A. Denny, A. J.
Bridges, D. R. Cody, D. W. Fry, A. McMichael, H. Zhou, University of Auckland
Medical School, New Zealand |
|
|
||
|
OP-III-11 |
|
||||
|
|
|||||
|
|
|
||||
|
August 8, Tuesday
|
103, TICC
|
|
|
||
|
|
|
|
|||
|
Session
IV: Bioorganic Chemistry of Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: J S. Bradshaw |
|
|
||
|
|
|
|
|||
|
|
M. P.
Groziak, Z.-W. Huan, A. D. Ganguly, Southern |
|
|
||
|
OP-IV-1 |
Development
of Imidazo[4,5-e][2,4,1]oxaza- and Diazaborine Purine Analogs |
|
|
||
|
|
|
|
|||
|
|
M. J.
Wanner, G. J. Koomen, |
|
|
||
|
OP-IV-2 |
|
|
|||
|
|
|
|
|||
|
|
H. Neunhoeffer, J. Gante, A. Schmidt, Technische Hochschule
Darmstadt, Germany |
|
|
||
|
OP-IV-3 |
1,4,5,6-Tetrahydro-1,2,4-triazin-3-ones
- Cyclic Azapeptides |
|
|
||
|
|
|
|
|||
|
|
Y. L. Chen, J. Collins, D. Costello, M.
Corman, A. Dunaiskis, S. Faraci, J. Heym, R. Mansbach, A. Schrnidt, D.
SchuIz, T. Seeger, P. Seymour, D. TingIey, E. Winston, Pfizer
Inc., U.S.A. |
|
|
||
|
OP-IV-4 |
|
||||
|
|
|
|
|||
|
|
|
|
|||
|
|
P.
Pradhan, A. Banerji, Bhabha Atomic Research |
|
|
||
|
OP-IV-5 |
|
|
|||
|
|
|
||||
|
POSTER SESSION II
|
|
|
|||
|
|
|
||||
|
August 8, Tuesday
|
201AF, TICC
|
|
|
||
|
|
|
|
|||
|
PO2-111 |
M. G. Marei, Alexandria
University, Egypt |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-112 |
K.
Imafuku, N. Ishida, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-113 |
T.-H. Duh, M.-J. Wu, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-114 |
H.
|
|
|||
|
|
Synthesis
and Reaction of 2- Thianaphthalenes Bearing an Electron-Withdrawing Group at
3-Position |
|
|||
|
|
|
|
|||
|
PO2-115 |
M.
Yokoyama, T. Akiba, M. Nomura, H. Toyoshima, H. Togo, Chiba University, Japan |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-116 |
T. Sano, Y.
Niimura, J. Toda, |
|
|
||
|
|
Synthesis
of Erythrina Alkaloid via Ring Formation by Pummerer Reaction |
|
|
||
|
|
|
|
|||
|
PO2-117 |
I. V.
Alabugin, V. K. Brel, N. S. Zefirov, Russian Academy of
Science, Russia |
|
|
||
|
|
First
Heterocytlic Phosphorus-Containing Unsaturated Sulfenylchlorides |
|
|
||
|
|
|
|
|||
|
PO2-118 |
I. V.
Alabugin, G. A. Sereda, V. K. Brel, N. V. Zyk, N. S.
Zefirov, Russian Academy of Science, Russia |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-119 |
V. K.
Brel, E. V. Abramkin, I. V. Alabugin, Russian Academy of Science, Russia |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO2-120 |
C.-Y.
Cheng, J.-P. Liou, H.-L. Wei, |
|
|
||
|
|
Synthesis
of Spiro [benzofuran-3(2H),4'-piperidines] via Intramolecular Radical
Cyclization |
|
|||
|
PO2-121 |
R.
Valters, G. Karlivans, J. Gulbis, M. Utinans, A. Bace, |
|||||
|
|
A
General Method for the Synthesis of Trichloro-l,4-benzoquinonylsubstituted Heterocycles |
|
|||
|
PO2-122 |
P. Kolar, A. Pizzioli, M. Tisler, University of Ljubljana, Slovenia |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO2-123 |
V. N.
Bulavka, O. N. Tolkachev, Ukrainian Acad. of Agric. Sci.,
Ukraine |
|
|
||
|
|
Synthesis
of Benzofuro[3a,3,2-ef][2]benzazepines by the Barton Reaction
Oxidation of Norbelladine Amides in Homogenic Medium |
|
|
||
|
|
|
|
|||
|
PO2-124 |
H.
Fujiwara, C. Suzuki, |
|
|
||
|
|
Synthesis
and Reaction of Novel Spirolactones of 9H-Xanthenes |
|
|
||
|
|
|
|
|||
|
PO2-125 |
C.-P. Chuang, S.-F. Wang, |
|
|
||
|
|
Manganese(III) Acetate Initiated
Oxidative Free Radical Reaction of 1,4‑Naphthoquinones |
|
|||
|
PO2-126 |
M. I. García Trimiñio, D. Moya Argilagos, A. Macias
Cabrera, R. Pérez Perera, H. Heimgartner, A. Linden, National Center for
Scientific Research, Cuba |
|
|
||
|
|
|
|
|||
|
|
3,3-Diamino-2-nitrothioacrylamides,
Useful Tools in Synthetic Chemistry |
|
|
||
|
|
|
|
|||
|
PO2-127 |
M.
I. García
Trimiñio, A. Macias Cabrera, D. Moya Argilagos, R. Pérez
Perera, H. Heimgartner, A. Linden, National Center for Scientific Research,
Cuba |
|
|
||
|
|
|
||||
|
|
|
||||
|
|
|
|
|||
|
PO2-128 |
O. Muraoka, H. Aoyama, G.
Tanabe, |
|
|
||
|
|
Synthesis of 2-Substituted
2-Thiazolines via the Reductive Cyclization of N,N'‑Diacylcystamines |
|
|||
|
|
|
|
|||
|
PO2-129 |
M. Takahashi, M. Oba, |
|
|
||
|
|
Synthesis of 1,3-Benzothiazoles
and 1,4-Benzothiazines via Aza-Wittig Reaction |
|
|
||
|
|
|
|
|||
|
PO2-130 |
H. Neunhoeffer, V. Rusinov,
O. Chupakhin, Technische Hochschule Darmstadt, Germany |
|||||
|
|
Direct
Introduction of Aromatic C-Nucleophiles into 1,2,4-Triazin-5(2H)-ones |
|
|
||
|
|
|
|
|||
|
PO2-131 |
V. I.
Saloutin, Z. E. Skryabina, |
|
|
||
|
|
|
|
|||
|
|
Interaction
of 2-Ethoxycarbonyl-5,6,7,8-tetrafluorochromone with N-di- and Trinucleophiles |
|
|||
|
|
|
|
|||
|
PO2-132 |
S. Jin,
J. Xu, Q. Xing, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-133 |
V. I. Timokhin, |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO2-134 |
M. Nishikawa, Y. Murai, O.
Onomura, Y. Veda, Daicel Chemical Industries, Ltd.,
Japan |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-135 |
N. Nishiwaki, Y. Tohda, M. Ariga,
Osaka Kyoiku University, Japan |
|
|
||
|
|
Cine-Substitution
of 1-Methyl-3,6,8-trinitroquinolin-2(1H)-one |
|
|
||
|
|
|
|
|||
|
PO2-136 |
R H.
Schlessinger, Y.-J. Li, |
|
|
||
|
|
Total
Synthesis of Virginiamycin M2 Using Vinylogous Urethane
Methodologies |
|
|
||
|
|
|
|
|||
|
PO2-137 |
H.
Ogasawara, T. Shiohara, M. Suzuki, O. Hoshino, Science |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-138 |
Y. Tominaga, N.
Yoshioka, S. Kataoka, T. Hata, N. Aoyama, T. Masunari, A. Miike, R N.
Castle, Nagasaki University, Japan |
|
|
||
|
|
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
PO2-139 |
T.-J. Lu, L-J. Sheu, |
|
|
||
|
|
1,3-Dipolar Cycloaddition
Reactions of α,b-Unsaturated Acetals with
Nitrile Oxides |
|
|
||
|
|
|
|
|||
|
PO2-140 |
A.
Miyashita, Y. Suzuki, N. Kuriyama, E. Oishi, T. Higasino, University
of Shizuoka, |
|||||
|
|
Catalytic Activities of Azolium
Salts for Benzoin Condensation and Related Reaction |
|
|
||
|
|
|
|
|||
|
PO2-141 |
E. Oishi, K.
Yahagi, A. Miyashita, K.-i. Iwamoto, T. Higasino, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
PO2-142 |
B. Puodziunaite, R. Janciene, L.
Kosychova, Z. Stumbreviciute, Institute of Biochemistry, Lithuania |
|
|
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Interaction
of Tetrahydro-l,5-benzodiazepin-2-ones (or-thiones) with Nucleophiles |
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PO2-143 |
G. Hajós, G.
Timári, Zs. Riedl,
A. Messmer, W. Ritzberger, J. G. Schantl, Central Research Institute
for Chemistry, |
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PO2-144 |
Z.-T. Huang, J.-C. Wang, C.-Y.
Yu, L.-B. Wang, Acadenia Sinica, China |
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PO2-145 |
S. Arai, K. Sato, T.
Yamagishi, Tokyo Metropolitan University, Japan |
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Synthesis
and Reactivity of Thieno-Fused Analogues of Benzo[a]Quinolizinium Salt |
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PO2-146 |
S. Arai, M. Koyama, T.
Yamagishi, Tokyo Metropolitan University, Japan |
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PO2-147 |
V. K. Yu, R E.
Meirmanova, E. E. Fomicheva, National Academy of Sciences, Republic |
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PO2-148 |
K. Teng, R.
Bharadwaj, P. D. Cook, |
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Study the Synthetic
Utility of
1-(3-Benzyloxy-(4'-benzoyl-5'-acetoxy)tetrahydrofuran-2'-yl)thymine for
Furanoid Nucleoside Analogues Synthesis |
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PO2-149 |
W. Franek, |
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PO2-150 |
S.-M.
Yang, J.-M. Fang, |
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PO2-151 |
S.
Yasuike, S. Shiratori, J. Kurita, T. Tsuchiya, |
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Synthesis of Novel
1-Benzometallepines Containing Group 14, 15 and 16 Elements |
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PO2-152 |
Y. Miki, Y.
Tada, K.-i. Matsushita, H. Hachiken, |
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PO2-153 |
K. Oda, H.
Tsujita, M. Sakai, M. Machida, Health Sciences |
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PO2-154 |
Y. Komatsu, N. Minami, Eisai Co., Ltd., Japan |
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PO2-155 |
Y. Kondo, T.
Matsudaira, T. Sakamoto, Tohoku University, Japan |
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Syntheses
of Heterocycles Using Ate Complexes of Aromatic Metal Derivatives |
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PO2-156 |
H.-H.
Tso, N.-c. Yang, Y.-M Chang, Academia Sinica, Taiwan,
R.O.C. |
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PO2-157 |
K. Orito, M. Miyazawa, M.
Tokuda, Hokkaido University, Japan |
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PO2-158 |
A.-B.
Hörnfeldt, S. Gronowitz, P. Bjork, |
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Synthesis
of Nitrogen and Sulfur Containing Tricycles and Their Reactivity |
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PO2-159 |
S. M.
Anand, S. M. Jain, R. S. Kapil, Regional Research |
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PO2-160 |
D. Pandyo, M. Rao, K. B. Nair, M. S.
University of Baroda, |
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PO2-161 |
B. A. J.Clark, H. McNab, C. C.
Sommerville, The |
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Gas Phase Pyrolysis of
1-(2-Azidophenyl)azoles Leading to Condensed Heterocyclic Systems |
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PO2-162 |
R-S. Liu, L-H. Shiu,
H.-G. Shu, |
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Tungsten-η1-propargyl
Compounds for Synthesis of Five-Membered Oxygen Heterocycles |
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PO2-163 |
G.
Stájer, A E. Szabó, G. Bermith, P. Sohar, Albert
Szent-Gyorgyi Medical University, |
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Saturated
Heterocycle-Condensed Isoindolone Isomers Prepared from Aroylcyclohexanecarboxylic
Acids |
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PO2-164 |
S. Z. Vatsadze, |
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Intramolecular Interactions in
3,7-Diazabicyclo[3.3.1]nonanes and Their Complexes |
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PO2-165 |
A. I. Kotov, R. V. Pisarev, E. B.
Yagubskii, C. Faulmann, P. Cassoux, Russian Academy of Sciences, Russia |
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PO2-166 |
E. V. Tretyakov, S. F. Vasilevsky, Siberian
Division of the Russian |
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The Unknown Nitrodeiodination of
Polyiodopyrazoles: A New, General Entry to 4-Nitroiodopyrazoles |
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PO2-167 |
L.
Petrulanis, G. Veinberg, N. Grigan, D. Zeile, D. Musels, E. Lukevics,
Latvian Institute of Organic |
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PO2-168 |
Yu. S. Andreichikov, S. N. Shurov, E. Yu.
Pavlova, P. A. Manakov, |
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PO2-169 |
L. M. Gornostaev, N.
A. Timoshkova, V. T. Sakilidi, State Pedagogical University, Russia |
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Synthesis of Nitrogencontaining
Heterocycles Using 1,4-Naphtoquinon Derivatives |
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PO2-170 |
M. S. Shvartsberg, I. D. Ivanchikova,
I. L. Barabanov, M. A. Mzhelskaya, A. V. Piskunov, L. G. Fedenok, Russian
Academy of Sciences, Russia |
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Novel
Syntheses of Condensed Heterocyclic Quinone Derivatives |
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PO2-171 |
L.-M. Yang, National Research Institute of
Chinese |
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Synthesis of Acyclic Pyrrolo[2,3-d]pyrimidine
Nucleoside Analogue |
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PO2-172 |
A. V. Tkachev, Novosibirsk Institute of |
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Chiral Heterocycls Derived from
Natural Terpenes: Syntheses and Application. |
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PO2-173 |
S. A. Popov, A. V. Tkachev,
Novosibirsk Institute of |
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Tricyclic Pyrazole- and
Pyrazolinol-Type Heterocycles Based on the (+)-3-Carene Molecule |
|
|||
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PO2-174 |
C.-K.
Sha, C.- Y. Shen, R.-S. Lee, S.-R. Lee, W.-H.
Tseng, |
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PO2-175 |
A. M.
Chibiryaev, S. A. Popov, A. V. Tkachev, Novosibirsk Institute
of |
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PO2-176 |
A. Ohta, M.
Maeda, F. Okazaki, Y. Aoyagi, |
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Total
Synthesis of Pyrrolidine Alkaloids via 1,3-Dipolar Cycloaddition
Reaction |
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PO2-177 |
A. J.
Wood, P. R. Jenkins, |
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PO2-178 |
N. Maezaki, M.
Soejima, M. Takeda, A. Sakamoto, I. Sakamoto, Y. Matsumori, T. Tanaka, C.
Iwata, Osaka University, Japan |
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PO2-179 |
C.-C. Chen, J.-S. Fan, R-S. Liu, |
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PO2-180 |
C.
Kashima, K. Takahashi, K. Fukusaka, |
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PO2-181 |
R. Pellicciari, B. D. Giacomo, B.
Natalini, M.-H. Ni, R Luneia, Università degli
Studi, Italy |
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|
Enantioselective
Synthesis and Properties of New Potent and Metabolically Stable Terfenadine Analogs |
||||||
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PO2-182 |
V. P. Morgaluk, B. M. Arshava, A. A. Nikitenko,
L. L. Zil'berg, Y. E. Raifeld, |
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|
Transition
Metal Containing Nucleophilic Reagents for Regioselective Oxirane Ring
Cleavage |
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|||
|
PO2-183 |
P. A. Nadar, T. R Prabakaran,
Annamalai University, India |
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|
|
Synthesis
and Mass Spectral Study of Substituted 2-Phenylthiazolidines |
|
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PO2-184 |
V. B.
Kurochkina, P. S. Nys, G. S. Libinson, National Research
Centre for Antibiotics, |
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|
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|
Biocatalysis
in Production of Ureidopenicillins and Ureidocephalosporins |
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PO2-185 |
V. B. Kurochkina, G. S. Libinson, P. S. Nys,
National Research Centre for Antibiotics, |
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Acyl Transfer Synthesis of
Aminopenicillins and Aminocephalosporins |
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PO2-186 |
J. B. Hansen, B. Christensen, Novo Nordisk A/S,
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PO2-187 |
P.
Jakobsen, A. Kanstrup, J. Lundbeck, P. Faarup, Novo Nordisk
A/S, |
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Synthesis
and Biological Activity of New Thieno[2,3-b]indoles |
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PO2-188 |
M. Gruttadauria, P. L. Meo, R. Noto,
A. Pace, G. Werber, Università di Palermo, Italy |
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Hindered
Rotation about C-N Bond in 2,3-Dihydro-4(1H)-quinazolinones |
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|
PO2-189 |
F.
Hadizadeh, A. Ghanbarpour, The Medical Seiences |
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Synthesis
and Antidepressant Activity of a Series of Benzamides |
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PO2-190 |
Z.-Y.
Zhang, N. Zou, |
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PO2-191 |
S.-F.
Lee, G. W. Luehr, C. R. Scott, R. J. Anderson, Sandoz Agro, Inc., |
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|
||
|
|
Synthesis
and Herbicidal Activity of Substituted Benzoyl-2H-pyran-3,5-(4H,6H)-dione
Derivatives |
|
|||
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|
PO2-192 |
K. Sasaki, A. S. S. Rouf, T.
Matsushita, M. Yoshida, T. Hirota, Okayama University, Japan |
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|
Reaction
of 4-[o-Cyanoarylthio( or oxy) ]butyronitrile with Base |
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PO2-193 |
F. Boers, G.
Lemière, J. A. Lepoivre, R Dommisse, A. D. Groot, F. Alderweireldt, |
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PO2-194 |
Y. Morita, M. Abel, M. Ono, M.
Daneshtalab, R. Micetich, Y. Yamamoto, Tohoku College of Pharmacy, Japan |
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|
|
Modifications
of 6,8- Dihydroxy-4-ethoxycarbonyl-isoquinolone Derivatives |
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PO2-195 |
A. K. LY, H.-P.
Husson, K. Camara, Université de Conakry, West Africa |
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|
PO2-196 |
A. Shalmashi, Iranian Research Organic for |
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||
|
|
Synthesis and Pharmacological
Evaluation of Indole Derivatives as Antidepressants |
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|
||
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|
PO2-197 |
O. N.
Kataeva, I. A. Litvinov, V. A. Naumov, Russian Academy of
Sciences, Russia |
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||
|
|
Molecular
Structure of Eight-Membered Heterocyclic Compounds in Crystalline Phase |
|
|||
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PO2-198 |
T.-C.
Chien, C.-S. Chen, J.-Y. Yeh, K.-C. Wang, J.-W. Chern, |
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PO2-199 |
G. P.
Kalena, P. Pradhan, A. Banerji, Bhabha Atomic Research |
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|
PO2-200 |
R. Xu, W.
Pang, S. Qiu, |
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||
|
|
The Role
of Heterocyclic Nitrogen Compound in the Crystallization of Microporous
Materials |
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|
PO2-201 |
I. A. Litvinov, Russian |
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|
PO2-202 |
K. N.
Rajasekharan, K. V. D. Babu, E. Samuel, M. M. Samuel, |
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||
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|
|
Synthesis
of Anchorable 1,3,5-Triaryl-2-pyrazoline Flurophores |
|
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|
PO2-203 |
H. Hara, S.-i.
Watanabe, O. Hoshino, Science |
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|
PO2-204 |
V. Ch. Christov, C. M
Angelov, |
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||
|
|
Synthesis of Heterocyclic
Phosphorus Compounds from Unsaturated Phosphonates |
|
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|
PO2-205 |
M.
Velasco, E. Angeles, B. Villaneda, R. Martinez, Universidad Nacional
Autonoma de México, México |
|
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|
PO2-206 |
H. Wu, X.
Huang, Chinese |
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|
PO2-207 |
J.
Bloxham, C. J. Moody, Loughborough |
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|
PO2-208 |
H.-J. Tien, J.-T. Chern,
National Cheng Kung University, Taiwan, R.O.C. |
|
|
||
|
|
Oxidation
of 4-(1'-Hydroxyethyl)-3-(4'-substitutedphenyl)sydnone |
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|
||
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|
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|
PO2-209 |
M. S.
Roy, G. D. Sharma, Defence Laboratory |
|
|
||
|
|
Electrical
and Photoelectrical Properties of Furazano(3,4-b)piperazine (FP) Thin Film |
|
|||
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|
PO2-210 |
A. V.
Sereda, O. N. Tolkachev, Ukrainian Acad. Agr. |
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|
PO2-211 |
S. Mataka, H. Moriyama, T.
Sawada, M. Tashiro, Kyushu University, Japan |
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|
PO2-212 |
D. Zhu,
P. Wu, Y. Liu, Y. Xli, Y. Li, W. Qin, B. Zhang, S. Liu, Y. Yao,
Academia |
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PO2-213 |
N. N. Tonkih, A Ya. Strakovs, O. Ya. Neilands, |
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|
||
|
|
2-Isonicotinoyl-,
2-nicotinoylhydrazinomethylene-1,3-cyclandiones and Theirs Polychrome |
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|
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|
PO2-214 |
D.-S.
Lee, P.-W. Yang, |
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|
||
|
|
Synthetic
Study of Azulenocrown Ethers a New High Dilution Technique and Another
Improving Method |
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PO2-215 |
B. Sener, F. Bingöl, A. H.
Gilani, Gazi University, Turkey |
|
|
||
|
|
New
Anticholinergic Heterocyclic Compounds from Fritillaria Species |
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|
PO2-216 |
A. V. Popov, E. L. Luzina, N. B. Bespalova,
M. A. Bovina, Russian Academy of Sciences, |
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PO2-217 |
A. V. Popov, A. V. Shastin, Russian |
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PO2-218 |
A. M.
Sipyagin, I. V. Efremov, A. V. Popov, Russian Academy of
Sciences, Russia |
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|||
|
PO2-219 |
A. V.
Popov, A. N. Pushin, E. L. Luzina, Russian Academy of Sciences, Russia |
|
|
||
|
|
A New
Way Towards Tritluoromethyl-Containing Heterocycles Using Polytluorinated
Enamines |
|
|
||
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|
PO2-220 |
A. V.
Popov, E. L. Luzina, Russian |
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|||
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|
||||
|
August 9, Wednesday
|
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|
|||
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|
|||
|
PLENARY
LECTURES
|
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|
|||
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|
|||
|
August 9, Wednesday
|
101,
TICC
|
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||
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|
|||
|
|
Chairman: V. Snieckus |
|
|
||
|
PL-5 |
S. V. Ley, J. A. Clase, I. C. Lennon, D. J.
Mansfield, University of Cambridge, U.K. |
|
|
||
|
|
Synthesis and Chernistry of the
Ionophore Antibiotic Tetronasin |
|
|
||
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|
|||
|
|
Chairman: F. Alderweireldt |
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|
||
|
PL-6 |
Y. Ito, |
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|
|||
|
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|
||||
|
INVITED LECTURES
|
|
|
|||
|
|
|
|
|||
|
August 9, Wednesday
|
101, TICC
|
|
|
||
|
|
|
|
|||
|
Session
Ia: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
M Ikeda |
|
|
||
|
|
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|
|||
|
|
G. S. R. Subba Rao, Indian Institute of |
|
|
||
|
IL-Ia-5 |
|
|
|||
|
|
|
|
|||
|
|
C. J. Moody, Loughborough |
|
|
||
|
IL-Ia-6 |
|
|
|||
|
|
|
||||
|
August 9, Wednesday
|
102,
TICC
|
|
|
||
|
|
|
|
|||
|
Session
II: Asymmetry and Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: T Kappe |
|
|
||
|
|
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|
|||
|
|
A. G.
Schultz, Zo Guo, T.
J. Guzi, P. R. Guzzo, S. J. Kirincich, R. Rahm, Rensselaer Polytechnic
Institute, U.
|
|
|
||
|
IL-II-5
|
|
|
|||
|
|
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|
|||
|
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|
|||
|
|
|
|
|||
|
|
T.
Hudlicky, |
|
|
||
|
IL-II-6 |
|
|
|||
|
|
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|
|||
|
|
|
||||
|
August 9, Wednesday
|
201BC, TICC
|
|
|
||
|
|
|
|
|||
|
Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: N De Kimpe |
|
|
||
|
|
|
|
|||
|
|
G.
Bernáth, |
|
|
||
|
IL-III-5 |
|
|
|||
|
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|
|||
|
|
|
|
|||
|
|
M.
Tisler, P. Kolar, A Pizzioli, R. Zupet, |
|
|
||
|
IL-111-6 |
|
|
|||
|
|
|
||||
|
August 9, Wednesday
|
103,
TICC
|
|
|
||
|
|
|
|
|||
|
Session V: Molecular
Recognition by Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: |
|
|
||
|
|
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|
|||
|
|
W. Verboom, |
|
|
||
|
IL-V-1 |
|
|
|||
|
|
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|
|||
|
|
E. Kimura, |
|
|
||
|
IL-V-2 |
|
|
|||
|
|
|
||||
|
August
10, Thursday
|
|
|
|||
|
|
|
|
|||
|
PLENARY LECTURES
|
|
|
|||
|
|
|
|
|||
|
August 10, Thursday
|
101, TICC
|
|
|
||
|
|
|
|
|||
|
|
Chairman:
B. Stanovnik |
|
|
||
|
PL-7 |
G. R.
Newkome, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: A. Padwa |
|
|
||
|
|
C. W. Rees, |
|
|
||
|
|
|
|
|||
|
|
|
||||
|
INVITED LECTURES
|
|
|
|||
|
|
|
|
|||
|
August 10, Thursday
|
101,
TICC
|
|
|
||
|
|
|
|
|||
|
Session
Ia: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
R. Neidlein |
|
|
||
|
|
|
|
|||
|
|
L. F. Tietze, W. Buhr, O.
Burkhardt, T. Grote, T. Raschke, R Schimpf, Georg-August- |
|
|
||
|
IL-Ia-7 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
T.-S. Chou, Academia Sinica, Taiwan, R.O.C. |
|
|
||
|
IL-Ia-8 |
Generation of Heteroaromatic ortho-Quinodimethanes
via 3-Sulfolenes |
|
|
||
|
|
|
||||
|
August 10, Thursday
|
201DE, TICC
|
|
|
||
|
|
|
|
|||
|
Session
Ib: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: T Livinghouse |
|
|
||
|
|
|
|
|||
|
|
E. Block, State |
|
|
||
|
IL-Ib-3 |
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
|
S. Kim, C. M.
Cho, |
|
|
||
|
IL-Ib-4 |
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
102,
TICC
|
|
|
||
|
|
|
|
|||
|
Session
II: Asymmetry and Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: C-C Liao |
|
|
||
|
|
|
|
|||
|
|
H. J.
Liu, W. L. Yeh, |
|
|
||
|
IL-II-7 |
|
|
|||
|
|
|
|
|||
|
|
W. H. Pearson, |
|
|
||
|
IL-II-8 |
2-Azaallyl Anion Chemistry:
Application to the Stereoselective Synthesis of Heterocyclic Compounds |
|
|
||
|
|
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
20lBC, TICC
|
|
|
||
|
|
|
|
|||
|
Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: J. G. Schantl |
|
|
||
|
|
|
|
|||
|
11:00 |
R. Pellicciari, Università degli Studi, Italy |
|
|
||
|
IL-III-7 |
|
|
|||
|
|
|
|
|||
|
|
F.-W.
Yeng, J.-Y. Chili, P.-H. Yang, P.-L. Lee, S.-Y. Chou, S.-S. Chen C.-L. J.
Wang, |
|
|
||
|
IL-III-8 |
|
|
|||
|
|
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
103, TICC
|
|
|
||
|
|
|
|
|||
|
Session V: Molecular
Recognition by Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
|
|
|
||
|
|
|
|
|||
|
|
J. S. Bradshaw, K. E. Krakowiak, R. L.
Bruening, M. L. Bruening, A. V. Bordunov, V. N. Pastushok, P. C. Hellier, X.
X. Zhang, and R. M. Izatt, Brigham Young University, U.S.A. |
|
|
||
|
IL-V-3 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
R. J.-R. Hwu, |
|
|
||
|
IL-V-4 |
Development and Computer Modeling
of Organic Compounds as Photo-Induced DNA‑Cleaving Agents |
|
|
||
|
|
|
|
|||
|
|
|
||||
|
ORAL PRESENTATIONS
|
|
|
|||
|
|
|
|
|||
|
August 10, Thursday
|
101, TIC C
|
|
|
||
|
|
|
|
|||
|
Session
Ia: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
Z-T. Huang |
|
|
||
|
|
|
|
|||
|
|
J. B.
Bremner, R. J. Smith, G. J. Tarrant, |
|
|
||
|
OP-Ia-12 |
A
Meisenheimer Rearrangement Approach to Bridgehead Hydroxylated Tropane Alkaloid
Derivatives |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
S.
Gronowitz, A.-B. Homfeldt, E. Temciuc, |
|
|
||
|
OP-Ia-13 |
Cyclication
Reactions of Some Dithienopyridine Derivatives with Dimethyl Acetylenedicarboxylate |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
J. G. Schantl, H.-T. Cam-Hoai, |
|
|
||
|
OP-Ia-14 |
Synthesis of Pyridazines Using
Diazenium Ions and Diazonium Ions |
|
|
||
|
|
|
|
|||
|
|
T. Kappe, P. Roschger,
B. Schnell, B. D. Schober, University of Graz, Austria |
|
|
||
|
OP-Ia-15 |
Rearrangement
Reactions of Heterocycles via α-Oxoketene Intermediates |
|
|
||
|
|
|
|
|||
|
|
S. T.
Abu-Orabi, L. Al-Momany, |
|
|
||
|
OP-Ia-16 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
V. A. Bakulev, Ural |
|
|
||
|
OP-Ia-17 |
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
201DE, TICC
|
|
|
||
|
|
|
|
|||
|
Session
Ib: Organic Synthesis in Heterocyclic Chemistry
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
G. Roos |
|
|
||
|
|
|
|
|||
|
|
Q. Yao, W.
Pfleiderer, University of Konstanz, Germany |
|
|
||
|
OP-Ib-12 |
|
|
|||
|
|
|
|
|||
|
|
C. Th.
Pedersen, N. Svenstrup, |
|
|
||
|
OP-Ib-13 |
The
Reaction of 1,2-Dithiole-3-thiones with Trivalent Phosphorus Compounds |
|
|
||
|
|
|
|
|||
|
|
T. H. Ngoi, D. H. Reid, University of the |
|
|
||
|
OP-Ib-14 |
New Syntheses of Five- and
Six-Membered Heterocycles Using 3-Chloropropenylidene Iminium Salts |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
R. S.
Glass, M. Sabahi, Sanaullah, W.P. Singh, G.S. Wilson, The |
|
|
||
|
OP-Ib-15 |
|
|
|||
|
|
Synthesis,
Structure and Redox Properties of a Conformationally Restricted 1,5‑Dithiocane |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
C.-S. Li, N.
Mayes, Merck Frosst Canada Inc., |
|
|
||
|
OP-Ib-16 |
|
|
|||
|
|
|
|
|||
|
|
V.V.
Samoshin, E.I. Troyansky, |
|
|
||
|
OP-Ib-17 |
|
|
|||
|
|
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
102, TICC
|
|
|
||
|
|
|
|
|||
|
Session
II: Asymmetry and Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: C. O. Kappe
|
|
|
||
|
|
|
|
|||
|
|
T.
Koizumi, T. Takahashi, Y.N. Yamakoshi, W.-Y. Ge, J. Sugita,
K. Okayama, |
|
|
||
|
OP-II-12 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
P. Q.
Huang, X. S. Fei, Y. P. Ruan, |
|
|
||
|
OP-II-13 |
An
Unified Strategy for the Asymmetric Synthesis of Pyrrolidine Alkaloids |
|
|
||
|
|
|
|
|||
|
|
T.
Kiguchi, M. Ikai, Y. Yuumoto, T. Naito, |
|
|
||
|
OP-II-14 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
15:00 |
M.
Sato,
S. Sunami, M. Murakami, C. Kaneko, T. Furuya, H. Kurihara, Tohoku University, Japan |
|
|
||
|
OP-II-15 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
A. van
Oeveren, C. W. Leung, E. M. Geertsema, B. L. Feringa, |
|
|
||
|
OP-II-16 |
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
|
V. I.
Sokolov, N. V. Abramova, N. M. Loim, M. A. Kondratenko, |
|
|
||
|
OP-II-17 |
|
|
|||
|
|
|
||||
|
|
|
||||
|
August 10, Thursday
|
201BC, TICC
|
|
|
||
|
|
|
|
|||
|
Session
III: Hetrocyclic Pharmaceuticals and Agrochemicals
|
|
|
|||
|
|
|
|
|||
|
|
Chairman: K. K. Balasubramanian |
|
|
||
|
|
|
|
|||
|
|
R. R.
Gupta, P. K. Dev, C. M. Rajoria, M. K. Nyati, A. Gupta, University of
Rajasthan, |
|
|
||
|
OP-III-12 |
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
|
H.-J.
Federsel, G. Glasare, C. Högström, J. Wiestål, B. Zinko, C.
Ödman, Astra Production Chemicals AB, |
|
|
||
|
OP-III-13 |
|
|
|||
|
|
An
Expedient Two-Step Transformation of Thiazoles to Medium- and Large-Sized N,S‑Heterocycles |
|
|||
|
|
|
|
|||
|
|
P.-P.
Kung, A. Fraser, C. Guinosso, K. Weiler, P. Wheeler, V. Mohan, P. D. Cook,
ISIS Pharmaceuticals, Inc, |
|
|
||
|
OP-III-14 |
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
|
L.-C.
Hwang, C.-C. Tzeng, |
|
|
||
|
OP-III-15 |
|
|
|||
|
|
|
||||
|
August 10, Thursday
|
103, TICC
|
|
|
||
|
|
|
|
|||
|
Session V: Molecular
Recognition by Heterocycles
|
|
|
|||
|
|
|
|
|||
|
|
Chairman:
G. J Koomen |
|
|
||
|
|
|
|
|||
|
|
M. Berger, W.
Peschke, F. P. Schmidtchen, Technische Universität München, Germany |
|
|
||
|
OP-V-1 |
Recognition
of Anionic Substrates Using Bicyclic Guanidinium Receptors |
|
|
||
|
|
|
|
|||
|
|
A. Katoh, Y.
Kitamura, J. Ohkanda, |
|
|
||
|
OP-V-2 |
Synthesis
of New Bipyridines Bearing the Carboxyl Group and Properties of Their Ru(II)
Complexes |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
G.
Kollenz, W. Heilmayer, C. O. Kappe, C. Wentrup,
KF-University of Graz, Austria |
|
|
||
|
OP-V-3 |
|
|
|||
|
|
|
|
|||
|
|
B.
Zwanenburg, N. A. J. M. Sommerdijk, P. ten Holte, D. G.
Geurts, C. J. Booij, M. H. L.
Lambermon, P. J. J. A Buynsters, R J. M. Notte, |
|
|
||
|
OP-V-4 |
|
|
|||
|
|
|
|
|||
|
|
Molecular
Recognition by Imidazole and Aziridine Derived Surfactants |
|
|
||
|
|
|
||||
|
POSTER SESSION III
|
|
|
|||
|
|
|
|
|||
|
August 10, Thursday
|
201AF,
TICC
|
|
|
||
|
|
|
|
|||
|
PO3-221 |
W.-J. Xiao, B.-G. Huang, L.-L.
Shi, Z.-C. Chen, Z.-W. Guo, Y.-Z. Hui, S. A. Lang, Chinese |
|
|
||
|
|
|
|
|||
|
|
Synthesis
of 1,4-Dideoxy-l,4-imino-L-lyxitol and Its N-Alkyl
Derivatives |
|
|
||
|
|
|
|
|||
|
PO3-222 |
K.
Hirota, H. Kuki, R. Totani, M. Sako, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO3-223 |
V.
K. Khlestkin, D. G. Mazhukin, A. Ya. Tikhonov, Yu. V.
Gatilov, |
|
|
||
|
|
|
|
|||
|
|
|
||||
|
|
|
|
|||
|
PO3-224 |
S.
Kanemasa, T. Tsuruoka, |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO3-225 |
A. P.
Halverson, R. N. Castle, L. W. Castle, |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO3-226 |
G. Cirrincione, A. M. Almerico, A.
Passannanti, P. Diana, F. Mingoia, Istituto Farmacochimico dell'Università, Italy |
|
|
||
|
|
|
||||
|
|
|||||
|
|
|
|
|||
|
PO3-227 |
D. W. M.
Liang, J.-H. Wang, L.-J. Liu, C.-J. Peng, |
|
|||
|
|
|
||||
|
|
|
|
|||
|
PO3-228 |
T. Oshima, Y.-i. Nakajima, T.
Nagai, Osaka University, Japan |
|
|
||
|
|
|
||||
|
|
|
|
|||
|
PO3-229 |
A. Kotschy, G. Hajós, G. Jones, A. Messmer,
Central Research Institute for Chemistry, |
|
|||
|
|
Synthesis and Ring Opening of
Tricyclic Fused s-Triazolium Salts |
|
|
||
|
|
|
|
|||
|
PO3-230 |
O.
Smolii, D. Shakhnin, S. Panchishin, E. Romanenko, B.
Drach, National Academy of Sciences of |
|
|
||
|
|
|
||||
|
Heterocyclization
of Products of Cyanomethylenetriphenylphosphorane Addition to
Acylisothiocyanates |
|
||||
|
|
|
|
|||
|
PO3-231 |
J.
Bergman, J. Tholander, |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
PO3-232 |
N. N.
Nagibina, L P. Sidorova, O. M. Chasovskikh, V. N. Charushin, Ural
State |
|
|||
|
|
1,3-Dipolar
Cycloaddition Reactions of 7-Azido-6-fluoro-4-quinolones |
|
|
||
|
|
|
|
|||
|
PO3-233 |
V. I.
Vysokov, T. K. Pashkevich, V. N. Charushin, O. N. Chupakhin, Ural
State |
|
|
||
|
|
|
|
|||
|
|
|
|
|||
|
|
|
|
|||
|
PO3-234 |
C.-P. Wu, L- Y.
Cheng, P.-W. Yang, |
|
|
||
|
|
Synthesis
of Cyclopent[c,d]azulene Derivatives by Vilsmeier Reaction |
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PO3-235 |
M. H. Elnagdi, E.
A. A. Hafez, A. W. Erian, Cairo University, Egypt |
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PO3-236 |
M.
Henriksen, K. J. Klabunde, R. G. Hazell, F. K. Larsen, K. V. Mikkelsen, T.
Schultz, K. Sylvester-Hvid, A. Senning, Technical |
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Synthesis
of trans-(±)-1,2,3,3a,4a,5,6,7-Octaphenyl-3aH,4aH-dicyclopenta[b,e][1,4]dithiin |
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PO3-237 |
H.
Takahata, S.-i. Kouno, T. Momose, |
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PO3-238 |
Y.-G.
Pan, M.-I. Lim, Clairol Inc., |
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An
Economical Synthesis of 5,6-Dihydroxyindole, a Biosynthetic Precursor to Melanin |
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PO3-239 |
L. Lu, J.-M.
Fang, |
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PO3-240 |
T.
Konakahara, C. Fukuda, |
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Synthesis
of Trifluoromethylisoxazoles from
b-Diketones
and the Reaction Mechanism |
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PO3-241 |
Y. Sugita, S. Inoue, Y. Shirataki, I.
Yokoe, Josai University, Japan |
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Diels-Alder Reaction of
3-Substituted Benzopyrons as a Dienophile and a Heterodiene |
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PO3-242 |
Y. Koseki, T. Nagasaka, |
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PO3-243 |
T. Sone, K. Sato, Yamagata University,
Japan |
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Aluminum
Chloride-Catalyzed Reactions of Dichlorothiophenes with Aromatic Compounds |
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PO3-244 |
T. Ibata, M. Himori, K.
Fukushima, Osaka University, Japan |
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PO3-245 |
H.-T.
Wang, J.-K. Yang, Z.-T. Huang, Academia Sinica, China |
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The
Reaction of Heterocyclic Ketene Aminals with Isothiocyanates |
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PO3-246 |
L. Fodor, J.
Szabó, G. Bermith, P. Sohar, |
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Synthesis
of 1,4-Benzothiazepins via Ring Transformations of 1,3-Benzothiazine Derivatives |
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PO3-247 |
M. J. Bordoloi, S.
Mohan, N. C. Barua, S. C. Dutta, R K. Mathur, A. C. Ghosh, Regional
Research Laboratory, India |
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Structure
of a Meroisoprenoid with an Unusual Carbon Framework |
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PO3-248 |
C.-K. Sha, J.-F. Yang, |
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Diels-Alder and Retro Diels-Alder
Reactions of 2,4-Dihydropyrrolo[2,3-c]indoles |
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PO3-249 |
D.
Korakas, A. Kimbaris, G. Varvounis, |
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PO3-250 |
J. Kurita, Y. Hashikawa, T. Tsuchiya, |
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Cobaltaindens; Syntheses and
Transformations into 5- and 6-Membered Heterocyclic Systems |
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PO3-251 |
C.-C.
Lin, S.-H. Tsai, J.-H. Chen, C.-I. Wu, H.-J. Wu, |
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Synthesis,
Structure, Formation Mechanism and Chemical Nature of Novel Oxa- Cage
Compounds |
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PO3-252 |
N.
Kakusawa, K. Inui, J. Kurita, T. Tsuchiya, |
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PO3-253 |
V. V.
Kiselev, V. S. Zyabrev, A. V. Kharchenko, B. S. Drach, |
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Regioselective
Heterocyclizations Based on Imidoylalkylating Agents and Their Analogs |
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PO3-254 |
T. Nishio, |
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PO3-255 |
N.
Palani, K. K. Balasubramanian, K. Vijayakumaran, Indian Institute of |
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PO3-256 |
N.
Palani, K. K. Balasubramanian, Indian Institute of |
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PO3-257 |
W.-S.
Chung, W.-J. Lin, W.-D. Liu, L.-G. Chen, |
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Synthesis
of Furan- Thiophene- and Pyrrole-Sultines and Their Application in Diels-Alder
Reactions |
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PO3-258 |
M. Kocevar, S. Polanc, P.
Trebse, University of Ljubljana, Slovenia |
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Pyrano[3,2-c]azepines
as Building Blocks in Heterocyclic Synthesis |
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PO3-259 |
A.
Rykowski, T. Lipinska, Agricultural University at |
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A
Concise Route to a Key Intermediate in the Total Synthesis of Sempervirine |
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PO3-260 |
N. Romanov, E.
Mikitenko, |
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PO3-261 |
N.
Romanov, E. Mikitenko, Y. Kovtun, National Academy of
Sciences of Ukraine, |
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PO3-262 |
C. A. Obafemi, W. Ptleiderer, Obafemi
Awolowo University, Nigeria |
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A Novel
Synthesis of Bibenzimidazoles and 2-Heterylbenzimidazoles |
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PO3-263 |
T. Okawara, Y. Okamoto,
T. Yamasaki, M. Furukawa, |
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Preparation of
Polyheteropolycycles and Prediction of Their Stereochemistries by AM1 |
|
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PO3-264 |
G.-P. Xue, C.-T. Wu, |
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PO3-265 |
G.-P.
Xue, C.-T. Wu, B.-S. Luo, |
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Synthesis
of 3,7-Dihydroxyl-1,5-diazacyclooctane and the Crystal Structure of Complex
with Cu(II) |
|
|||
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PO3-266 |
R. Zniber, E. M.
Essassi, M. Regragui, R. Achour, Université Mohammed V, Maroc |
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Synthesis
of New Heterocyclic Systems from Benzimidazol-2-thione |
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PO3-267 |
V. D. Pokhodenko, V. G. Koshechko, L. A.
Kiprianova, L. I. Kalinina, National |
|
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Electrochemical
Synthesis of Phenothiazine Derivatives Containing Nitrous Bases in the
Aromatic Ring |
|
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PO3-268 |
S. F. Vasilevsky, M. S. Shvartsberg, Siberian
Division of the Russian |
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PO3-269 |
L. I.
Belen'kii, |
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PO3-270 |
G.
Penieres, C. Alvarez, K. Franco, O. Garcia, Ciudad
Universitaria, Mexico |
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PO3-271 |
J.
G. Penieres C., J. F. Delgado R. J. M. Aceves H., J. G. Garcia E., Facultad
de Estudios Superiores Cuautithin-UNAM, Mexico |
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PO3-272 |
S. F.
Vasilevsky, T. A. Prikhodko, M. S. Shvartsberg, Siberian
Division of the Russian |
|
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A Cyclization of Vicinal
Acetylenic Derivatives of Phenyl- and Pyrazolylhydrazines |
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PO3-273 |
C.-K.
Jow, M. Cheung, T. Fukuyama, |
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PO3-274 |
I. Iovel, G. Oehme,
E. Lukevics, Latvian Institute of Organic |
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PO3-275 |
S. A.
Bakunov, A. V. Tkachev, Novosibirsk Institute of |
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New
Optically Active Isoquinuclidine Derivatives from Limonene |
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PO3-276 |
J.-S.
Lee, H.-P. Wang, |
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Studies
on Prevention of Δ3 → Δ2 Isomerization
along the Synthesis of Cephalosporin Prodrugs |
|
|||
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PO3-277 |
C. E.
Raab, G. H. P. Roos, M. P. Doyle, |
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PO3-278 |
R. A.
Aitken, K. Ali, S. T. E. Mesher, |
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|
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Applications
of a Proline-Derived Chiral Bicyclic Iminium Salt in Asymmetric Synthesis |
|
|||
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|
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PO3-279 |
R. A.
Aitken, A. H. Cowley, F. P. Gabbai, W. Masamba, University
of St. Andrews, U.K. |
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PO3-280 |
Y. Kita, S.
Kitagaki, M. Kondo, S. Okamoto, R. Imai, H. Fujioka, Osaka University, Japan |
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PO3-281 |
L.-B. Wang, C.- Y. Yu, Z.-J. Li, Z.-X. Ren, Z.- T. Huang,
Academia Sinica, China |
|
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|
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Regiospecific Nucleophilic Alkylation
and Glycosidation of Heterocyclic Ketene Aminals |
|
|||
|
PO3-282 |
H. Fujioka, H.
Kitagawa, N. Matsunaga, Y. Nagatomi, Y. Kita, Osaka University, Japan |
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PO3-283 |
Y.
Abrokina, B. Oksengendler, S. Rashidova, A. Razumnyi, N.
Nikiforova, Polymers of Academy of Sciences, Republic of Uzbekistan |
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|
|
Electronical
Spectrum of Long Qusi-1D Molecular Chains with Loops of Different Topology |
|
|||
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PO3-284 |
S. M. Bayomi, H. A. Al-Khamees, |
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Synthesis of N-[[4-(1H-Tetrazolo-5-yl)methyl]benzensulfonyl]-N'-Substituted
Ureas as
Potential Antidiabetic Agents |
|
|||
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PO3-285 |
L.-Y.
Hsu, C.-H. Lin, |
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PO3-286 |
P. S.
Nys, A. V. Sklyarenko, V. B. Kurochkina, G. S. Libinson, National
Research Centre for Antibiotics, |
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Enzymatic
Approach to Synthesis of Semisynthetic Betalactams |
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PO3-287 |
A. V.
Sklyarenko, P. S. Nys, National Research Centre for
Antibiotics, |
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PO3-288 |
V. Gupta, A.
Gupta, |
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PO3-289 |
P. H.
Olesen, P. Sauerberg, M. J. Sheardown, P. D.
Suzdak, M. D. B. Swedberg, C. H. Mitch, J. S. Ward, F. P. Bymaster, H. E.
Shannon, Novo Nordisk A/S, Denmark |
|
|||
|
|
Synthesis
of 3-Alkylthio-1,2,5-thiadiazol-1-azabicycles. A New
Class of
Antinociceptive
Agents |
|
|||
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|
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|
PO3-290 |
J.-A.
Mahling, G. M. Blackburn, |
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|
||
|
|
Synthesis
of New Bioactive 1,2,3,4-Tetrahydroisoquinoline Derivatives for Cytochrome P450 2D6 |
|
|||
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|
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|
PO3-291 |
T-S. Bai, O.
Lee, K.-D. Ker, H.-P. Wang, |
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|
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|
PO3-292 |
A.
Shafiee, M. Khazen, F. Poormorad, Medical Sciences |
|
|
||
|
|
Synthesis
of New 2-Imidazolylquinoline Derivatives as Fungicidal and Acaricidal Agents |
|
|||
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|
|||
|
PO3-293 |
Yu. N.
Bulychev, N. I. Zimakova, M. L. Gershanovich, |
|
|||
|
|
Synthesis
of 14C-CRC-87, Preclinical Pharmacokinetics and Phase I of
Clinical Trials |
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PO3-294 |
I. Maeba, Y.
Nishiyama, |
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PO3-295 |
J. Van
hemel, E. L. Esmans, F. C. Alderweireldt, |
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||||
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PO3-296 |
S. Peng, M.
Guo, M. Zhao, E. Winterfeldt, |
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|
PO3-297 |
B. L.
Mylari, C. E. Aldinger, T. A. Beyer, M. J. Peterson,
R. Sarges, P. J. Scott, Pfizer Inc., |
|
|||
|
|
N-1
Substituted 1,2,4-Triazine 3,5-Diones: A Novel Series of Aldose Reductase Inhibitors |
|
|||
|
PO3-298 |
H. S. Andersen, Novo Nordisk A/S, Denmark |
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|
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|
|
A Convenient Synthesis of 3-(1H-Imidazol-4(5)-yl)prop-1-yl-amine |
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|
PO3-299 |
A. Duflos, J. C.
Tristani, J. Fahy, C. Etievant, J. Lhomme, M. Demeunynck, N. Fixler, D. C. H.
Bigg, Centre de Recherche Pierre FABRE, France |
|
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|
PO3-300 |
W. J.
Houlihan, K. Prasad, O. Repic, R. Underwood, P.G. Munder, C.-P. Chen,
Bristol- Myers Squibb Research Institute, |
|
|||
|
|
Synthesis
and Antitumor Activity of the R- & S-Enantiomers of the
Phospholipid SRI 62-834 |
|
|||
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|
|||
|
PO3-301 |
A. B.
Reitz, M. Goodman, B. Pope, D. Argentieri, S. C. Bell, L. E. Burr, E. Chourmouzis,
J. Come, J. H. Goodman, D. Klaubert, B. E. Maryanoff, M. E. McDonnell, M. S.
Rampulla, M. R. Schott, R. Chen, The R. W. Johnson Pharmaceutical
Research Institute, U.S.A. |
|
|||
|
|
Guanosine
Derivatives as Immunostimulants. Discovery of Loxoribine |
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|
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|
PO3-302 |
C.-S. Chen, J.-W. Chem, |
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|
PO3-303 |
A. Monge, J. A.
Palop, A. L. de Ceráin, V. Senador, F. J. Martínez, Y. Sainz, S. Narro, E. García, C. de Miguel, M.
González, E. Hamilton, A. J. Barker, E. D. Clarke, D. T. Greenhow, CIFA, |
|
|||
|
|
Hypoxia-Selective
Agents Derived from Quinoxaline-N1,N4-dioxides |
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|
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|
|||
|
PO3-304 |
M. Jain, M. A.
Alabdalla, R. R. Gupta, |
|
|
||
|
|
Synthesis
of Substituted 4H-1,4-Benzothiazines and Their Conversion into
Sulfones |
|
|
||
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|
|||
|
PO3-305 |
D. Abou El
Ella, E. Goessnitzer, W. Wendelin, Karl-Franzens-University Graz,
Austria |
|
|
||
|
|
Synthesis,
Structure, Stereochemistry and Tautomerism of Dodecahydrobenzimidazo[2,1-b]quinazolines |
|
|||
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|
|||
|
PO3-306 |
D. Abou El Ella, E. Goessnitzer, W.
Wendelin, Karl-Franzens-University Graz, Austria |
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||||
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|
|||
|
PO3-307 |
A. Shafiee, M. Khazen, The
Medical Sciences |
|
|
||
|
|
Synthesis of New
2-Imidazolyl-quinoline 4-Carboximides as Potential Antitumor Agents |
|
|||
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|
|||
|
PO3-308 |
H.
Petersen, P. O. Sørensen, M. S. Chorghade, E. C. Lee, Novo
Nordisk A/S, |
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||||
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|
PO3-309 |
K.
Achiwa, H. Ebiike, |
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||||
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|
PO3-310 |
A.
Foroumadi, A. Sharifian, S. Emami, A. Davood, Y. Tabatabaiee,
Gh. Sepehri, A. Shafiee, |
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|
||
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|
|||
|
|
Synthesis
and Antimicrobial Activity of N-(2-Oxyimino-2-phenyl ethyl)quinolone Derivatives |
|
|||
|
PO3-311 |
V. Ambrogi, L.
Feriali, G. Grandolini, Università degli Studi di Perugia, Italy |
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||||
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|
|||
|
PO3-312 |
J. Li, G. Chen, J. M.
Webster, Simon Fraser University, Canada |
|
|
||
|
|
Antimicrobial
Metabolites from the Bacterium, Xenorhabdus Bovienii |
|
|
||
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|
|||
|
PO3-313 |
C.-Y.
Wei, Z. Slanina, P.-T. Chou, L. Adamowicz, |
|
|||
|
|
Complexes
of 2-Piperidinone and 7-Azaindole: A Computational Study |
|
|
||
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|
|||
|
PO3-314 |
W. Löwe, S. Bischoff,
M. Weber, G. Perpetuo, P. Luger, Freie Universität Berlin, Germany |
|
|||
|
|
Studies on the
Reactivity and Structure of Phenyl 7-Fluoro-4-chromone-3-sulfonate |
|
|
||
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|
|||
|
PO3-315 |
N. N.
Nikiforova, D. T. Alimov, B. L. Oksengendler, V. M. Kosov,
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|
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|
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PO3-316 |
C.-C. Feng, M. Nandi, C.-H.
Cheng, |
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PO3-317 |
G. N.
Nikonov, A. S. Balueva, A. A. Karasik, A. E. Arbuzov,
Russian Academy of Sciences, |
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Intramolecular
Interactions in Functional Substituted Phosphines |
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PO3-318 |
A.N.
Pankratov, A. N. Stepanov, N. G |
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PO3-319 |
A. N.
Pankratov, |
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PO3-320 |
Z.
Abdullah, N. Mohd Tahir, M. R. Abas, B. K. Low, |
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Synthesis
and Fluorescence Study of Selected 2-X Pyrimidines and Related Compounds |
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PO3-321 |
T.-Y.
Ssieh, S.-T. Liu, |
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Synthesis
and Metal Complexation of Thia-Macrocycle with Phosphines as Side-Arm Donors |
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PO3-322 |
T.
Eswara Yuvaraj, N. Sundaram, Indian Institute of |
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PO3-323 |
N. N.
Madikizela, N. Nkente, A. M. Sipamla, |
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PO3-324 |
V. V. Plemenkov, N. P.
Artemova, I. V. Fedunina, L. E. Nikitina, Medical University, |
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August 11, Friday
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PLENARY
LECTURES
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August 11, Friday
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101,
TICC
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Chairman:
K-C. Liu |
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PL-8 |
S. M.
Weinreb, The |
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Synthetic
Applications of a Novel Pericyclic Imino Ene Reaction of Allenyl Silanes |
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Chairman: H. Neunhoeffer |
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PL-9 |
C. H. Heathcock, |
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Chairman:
C.-K Sha |
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PL-10 |
D. A.
Blank, S. W. North, Y.-T. Lee, Academia |
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The Ultraviolet
Photodissociation Dynamics of Pyrrole and Other Small Heterocyclic Compounds |
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Closing
Ceremony (Announcement of the 16th ICHC) |
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